
Recettore degli oppioidi
I recettori degli oppioidi sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti degli oppioidi endogeni ed esogeni. Questi recettori svolgono un ruolo centrale nella modulazione del dolore, nella regolazione dell'umore e nei comportamenti di dipendenza. Gli agonisti e antagonisti dei recettori degli oppioidi sono ampiamente utilizzati nella gestione del dolore e nel trattamento delle dipendenze, nonché nella ricerca sui disturbi neurologici e psichiatrici. Presso CymitQuimica, offriamo una selezione completa di modulatori dei recettori degli oppioidi di alta qualità per supportare la tua ricerca in neurobiologia, gestione del dolore e terapia delle dipendenze.
Trovati 326 prodotti di "Recettore degli oppioidi"
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Asimadoline
CAS:Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.Formula:C27H30N2O2Colore e forma:SolidPeso molecolare:414.54BMS-986121
CAS:BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.Formula:C15H9Cl2N3O2SPurezza:99.67%Colore e forma:SolidPeso molecolare:366.22MCOPPB triHydrochloride
CAS:MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.Formula:C26H43Cl3N4Purezza:99.89% - 99.91%Colore e forma:SolidPeso molecolare:518.01Ref: TM-T2071
2mg34,00€5mg50,00€10mg87,00€25mg163,00€50mg255,00€100mg375,00€200mg535,00€1mL*10mM (DMSO)58,00€LY2940094 tartrate
CAS:LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.Formula:C26H29ClF2N4O8SColore e forma:SolidPeso molecolare:631.04GR103545
CAS:GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.Formula:C23H29Cl2N3O7Purezza:99.75%Colore e forma:SolidPeso molecolare:530.4Ref: TM-T9459
1mg87,00€2mg143,00€5mg188,00€10mg283,00€25mg509,00€50mg727,00€100mg1.017,00€1mL*10mM (DMSO)250,00€Ac-RYYRWK-NH2 acetate
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.Formula:C51H73N15O11Purezza:98.59%Colore e forma:SolidPeso molecolare:1072.22Naloxegol (NKTR-118)
CAS:Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].Formula:C34H53NO11Colore e forma:SolidPeso molecolare:651.78b-Casomorphin (1-3) Acetate
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.Formula:C25H31N3O7Purezza:98.99%Colore e forma:SolidPeso molecolare:485.53Ref: TM-T21660L
5mg44,00€10mg60,00€25mg93,00€50mg138,00€100mg202,00€200mg301,00€1mL*10mM (DMSO)58,00€Hemorphin-7 acetate(152685-85-3 free base)
Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.Formula:C51H68N12O13Purezza:99.66%Colore e forma:SolidPeso molecolare:1057.16BMS986187
CAS:BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.Formula:C31H34O4Purezza:99.09%Colore e forma:SolidPeso molecolare:470.6Nalmefene hydrochloride
CAS:Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.Formula:C21H26ClNO3Purezza:98% - 99.85%Colore e forma:SolidPeso molecolare:375.89EST73502 hydrochloride
CAS:EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.Formula:C19H27ClF2N2O2Colore e forma:SolidPeso molecolare:388.88Sec-O-Glucosylhamaudol
CAS:Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.Formula:C21H26O10Purezza:99.79%Colore e forma:SolidPeso molecolare:438.43GR 89696 free base
CAS:GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.Formula:C19H25Cl2N3O3Colore e forma:SolidPeso molecolare:414.33Naloxegol oxalate
CAS:Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.Formula:C36H55NO15Purezza:99.67% - >99.99%Colore e forma:SolidPeso molecolare:741.83N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.Formula:C30H39N5O8Purezza:>99.99%Colore e forma:SolidPeso molecolare:597.66Nociceptin
CAS:Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.Formula:C79H129N27O22Purezza:99.35%Colore e forma:SolidPeso molecolare:1809.04MCOPPB
CAS:MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.Formula:C26H40N4Colore e forma:SolidPeso molecolare:408.62Corydaline
CAS:<p>Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits CYP2C19 and CYP2C9.</p>Formula:C22H27NO4Purezza:98.97% - 99.86%Colore e forma:SolidPeso molecolare:369.45Dynorphin A 1-10 acetate(79994-24-4 free base)
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.Formula:C59H95N19O14Purezza:99.88%Colore e forma:SolidPeso molecolare:1294.53
