
Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.542 prodotti)
- Apoptosi(5.816 prodotti)
- Ciclo cellulare/Checkpoint(4.466 prodotti)
- Cromatina/Epigenetica(2.252 prodotti)
- Segnalazione citoscheletrica(1.381 prodotti)
- Danno al DNA/Riparazione del DNA(2.830 prodotti)
- Endocrinologia/Ormoni(3.518 prodotti)
- Enzima(3.640 prodotti)
- Proteina G/GPCR(8.362 prodotti)
- Immunologia e infiammazione(3.540 prodotti)
- Virus dell'influenza(296 prodotti)
- Segnalazione JAK/STAT(405 prodotti)
- Segnalazione MAPK(1.201 prodotti)
- Trasportatore di membrana/canale ionico(2.809 prodotti)
- Metabolismo(9.462 prodotti)
- Microbiologia/Virologia(7.003 prodotti)
- Neuroscienza(9.942 prodotti)
- Altri inibitori(37.827 prodotti)
- Ossidazione-riduzione(40 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.399 prodotti)
- Proteasi/Proteasoma(1.598 prodotti)
- Cellule staminali e Derivati(830 prodotti)
- Adattatori Tirosin-chinasi(2.012 prodotti)
- Ubiquitinazione(1.651 prodotti)
Mostrare 16 più sottocategorie
Trovati 66618 prodotti di "Inibitori"
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5'-Azido-5'-deoxy-2'-O-(2-methoxyethyl)-5-methyluridine
CAS:<p>5'-Azido-5'-deoxy-2'-O-(2-methoxyethyl)-5-methyluridine is a Nucleoside Derivative - 5'-Modified nucleoside; Azido-nucleoside; 2'-Modified nucleoside.</p>Formula:C13H19N5O6Colore e forma:SolidPeso molecolare:341.32Hippuryl-His-Leu-OH
CAS:<p>Hippuryl-His-Leu-OH tests for angiotensin I enzyme activity, allowing His-Leu detection by fluorescence.</p>Formula:C21H27N5O5Colore e forma:SolidPeso molecolare:429.473-Acetamidocoumarin
CAS:<p>3-Acetamidocoumarin is vital in biology, medicine, treating burns, brucellosis, rheumatic diseases, and cancer.</p>Formula:C11H9NO3Colore e forma:Light Yellow Amorphous PowderPeso molecolare:203.19Yadanziolide B
CAS:<p>Yadanziolide B, a bitter wood bittersweet analog from the stem of Brucea mollis, is cytotoxic with an IC50 value of 3.00-5.81 μM.</p>Formula:C20H26O11Purezza:99.76%Colore e forma:SolidPeso molecolare:442.41EHMT2-IN-1
CAS:<p>EHMT2-IN-1: potent EHMT inhibitor, for blood disorders/cancer research; IC50s <100 nM for EHMT1/2 peptides and cellular EHMT2.</p>Formula:C18H23N7OColore e forma:SolidPeso molecolare:353.422-(2,4-Dichlorobenzyl)thioadenosine
CAS:<p>2-(2,4-Dichlorobenzyl)thioadenosine is a Nucleoside Derivative - 2-Modified purine nucleoside.</p>Formula:C17H17Cl2N5O4SColore e forma:SolidPeso molecolare:458.32N2-(Isopropylphenoxyacetyl)-2'-O-propargylguanosine
CAS:<p>Nucleoside Derivatives - 2’-Modifed Nucleosides</p>Formula:C24H27N5O7Colore e forma:SolidPeso molecolare:497.5BRD5529
CAS:BRD5529 selectively blocks CARD9/TRIM62, disrupting ubiquitinylation; IC50 is 8.6 μM.Formula:C25H31N5O4Colore e forma:SolidPeso molecolare:465.54Bis-PEG9-acid
CAS:<p>Bis-PEG9-acid, a cleavable PEG-based linker, is utilized for PROTACs and ADCs synthesis.</p>Formula:C22H42O13Colore e forma:SolidPeso molecolare:514.56PEG8-Tos
CAS:PEG8-Tos is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.Formula:C23H40O11SPurezza:98%Colore e forma:SolidPeso molecolare:524.62NS 383
CAS:<p>ASIC blocker with varying IC50: 0.12 μM in hASIC1a, and ineffective on hASIC2a/3; <5 μM on rASIC1a/2a/3; alleviates pain in inflamed/CCI rats.</p>Formula:C19H19N3O2Colore e forma:SolidPeso molecolare:321.37IBT6A hydrochloride
CAS:IBT6A hydrochloride: Ibrutinib impurity, Btk inhibitor IC50: 0.5 nM, used in dimer/adduct synthesis.Formula:C22H23ClN6OColore e forma:SolidPeso molecolare:422.912'-O-Methyl-5-methylcytidine
CAS:<p>2'-O-Methyl-5-methylcytidine is a 2'-O-Methyl nucleoside.</p>Formula:C11H17N3O5Colore e forma:SolidPeso molecolare:271.272-Amino-6-chloropurine
CAS:<p>2-Amino-6-chloropurine: used to create antiviral drugs for EBV and HHV-6.</p>Formula:C5H4ClN5Colore e forma:SolidPeso molecolare:169.57β-Anomer
CAS:<p>β-Anomer shows antiviral properties.</p>Formula:C10H13N3O6Purezza:98.68% - 99.81%Colore e forma:SolidPeso molecolare:271.234-Chloro-7-(2-b-C-methyl-β-D-ribofuranosyl)-7H-pyrrolo[2,3-d] pyrimidine
CAS:<p>4-Chloro-7-(2-b-C-methyl-β-D-ribofuranosyl)-7H-pyrrolo[2,3-d] pyrimidine is a Nucleoside Derivative - 7-Deaza-purine nucleoside; 2'-Modified nucleoside; Halo-</p>Formula:C12H14ClN3O4Colore e forma:SolidPeso molecolare:299.71IMP2-IN-1
CAS:<p>IMP2-IN-1 effectively inhibits IMP2 (IC50: 81.3-127.5 μM), reduces IMP2 in SW480 cells, and hinders Huh7 cell activity.</p>Formula:C21H14F3NO4Colore e forma:SolidPeso molecolare:401.34Balaglitazone
CAS:Balaglitazone is a PPARγ agonist that regulates blood glucose and is used in studies of heart failure and myocardial infarction.Formula:C20H17N3O4SPurezza:99.74%Colore e forma:SolidPeso molecolare:395.434-Deoxy-3'-deoxy-3'-fluoro uridine
<p>Nucleoside Derivatives - 3’-Modified nucleosides, 4-Deoxy pyrimidine nucleosides, Fluoro-modified nucleosides</p>Colore e forma:SoildAripiprazole (D8)
CAS:<p>Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).</p>Formula:C23H27Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:456.441-(3'-O-[4,4'-Dimethoxytrityl]-α-L-threofuranosyl)-thymine
CAS:<p>Nucleoside Derivatives - L-Nucleosides; Protected nucleosides w/NH2/OH open</p>Formula:C30H30N2O7Colore e forma:SolidPeso molecolare:530.57Profluralin
CAS:Profluralin is a effective herbicide.Formula:C14H16F3N3O4Purezza:98%Colore e forma:Yellow-Orange Crystals SolidPeso molecolare:347.29N6-Bz-5'-O-DMTr-3'-deoxyadenosine-2'-O-CED-phosphoramidite
CAS:<p>N6-Bz-5'-O-DMTr-3'-deoxyadenosine-2'-O-CED-phosphoramidite is an adenine nucleoside analog with potential vasodilator activity and anticancer activity.</p>Formula:C47H52N7O7PPurezza:98.59%Colore e forma:SolidPeso molecolare:857.933-b-D-Ribofuranosyl-6-hydroxymethyl-furano[2,3-d]-pyrimidin-2-one
CAS:<p>Nucleoside; Used for nucleoside and nucleic acid modification</p>Formula:C12H14N2O7Colore e forma:SolidPeso molecolare:298.25Hoechst 33258 analog 5
CAS:<p>Hoechst 33258 analog 5 is an analog of Hoechst stains which are part of a family of blue fluorescent dyes used to stain DNA.</p>Formula:C29H26N6Colore e forma:SolidPeso molecolare:458.56Boc-C16-NHS ester
CAS:<p>Boc-C16-NHS ester, an alkyl/ether-based PROTAC linker, enables the synthesis of PROTACs[1].</p>Formula:C26H45NO6Colore e forma:SolidPeso molecolare:467.64N1-(tert-Butoxycarbonylmethyl)-6-[2-(N-Cbz-amino)ethoxy)]-phenoxazine
CAS:<p>N1-(tert-Butoxycarbonylmethyl)-6-[2-(N-Cbz-amino)ethoxy)]-phenoxazine is a PNA-related Derivative; Heterocyclic Compound - Fused polyheterocycle.</p>Formula:C26H28N4O7Colore e forma:SolidPeso molecolare:508.525'-Deoxy-5'-iodouridine
CAS:<p>Nucleoside Derivatives - Halo-nucleosides, 5’-Modified nucleosides</p>Formula:C9H11IN2O5Colore e forma:SolidPeso molecolare:354.1m-PEG7-Amine
CAS:<p>m-PEG7-Amine is a cleavable ADC linker used in the synthesis of antibody-drug conjugates (ADCs)[1].</p>Formula:C15H33NO7Purezza:98%Colore e forma:SolidPeso molecolare:339.422-Methoxy-2'-deoxy-2'-fluoro-β-D-arabinoadenosine
CAS:<p>Fluoro-modified nucleoside; 2/6/8-Modified purine nucleoside; Arabino-nucleoside</p>Formula:C11H14FN5O4Colore e forma:SolidPeso molecolare:299.262'-O-Methyl-5'-O-dmt-inosine-3'-CE-phosphoramidite
CAS:<p>2'-O-Methyl-5'-O-dmt-inosine-3'-CE-phosphoramidite is a Nucleoside Phosphoramidite.</p>Formula:C41H49N6O8PColore e forma:SolidPeso molecolare:784.842-Amino-N6,N6-dimethyl-2'-O-methyladenosine
CAS:<p>Nucleoside Derivatives - 2’-Modified nucleosides, 6-Modified purine nucleosides; N-Methylated nucleosides</p>Formula:C13H20N6O4Colore e forma:SolidPeso molecolare:324.34THZ-P1-2
CAS:<p>THZ-P1-2 is a PI5P4K inhibitor with anti-leukemic activity and can be used in the study of leukemia.</p>Formula:C31H29N7O2Colore e forma:SolidPeso molecolare:531.61Carpalasionin
CAS:<p>Carpalasionin is a natural product from Rabdosia lasiocarpa.</p>Formula:C22H28O8Purezza:98%Colore e forma:SolidPeso molecolare:420.458UBP608
CAS:<p>UBP608 selectively inhibits NMDA GluN1/GluN2A receptors, 23x more than GluN1/GluN2D.</p>Formula:C10H5BrO4Colore e forma:SolidPeso molecolare:269.05Batatasin I
CAS:Batatasin I is a natural product from Dioscorea batatasFormula:C17H16O4Purezza:98%Colore e forma:SolidPeso molecolare:284.31Mal-NH-Boc
CAS:<p>Mal-NH-Boc is a alkyl/ether-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>Formula:C11H16N2O4Colore e forma:SolidPeso molecolare:240.262'-O-(2-Methoxyethyl) inosine
CAS:<p>2'-O-(2-Methoxyethyl) inosine is a Nucleoside Derivative - 2'-Modified nucleoside.</p>Formula:C13H18N4O6Colore e forma:SolidPeso molecolare:326.313-[(6-Iodohexyl)oxy]-(3b)-cholest-5-ene
CAS:<p>Bio-reagents and Conjugation Reagents; Intermediates and Building Blocks - Electrophiles</p>Formula:C33H57IOColore e forma:SolidPeso molecolare:596.71Dodecanedioic acid
CAS:Dodecanedioic acid is a dicarboxylic acid used in the synthesis of plastics.Dodecanedioic acid is used as a base oil for industrial production.Formula:C12H22O4Purezza:98.1%Colore e forma:SolidPeso molecolare:230.3Clothiapine
CAS:Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.Formula:C18H18ClN3SPurezza:99.93%Colore e forma:SolidPeso molecolare:343.877-Deazaguanosine
CAS:<p>Nucleoside Derivatives - 7-Deaza-purine nucleosides; Drugs and Inhibitors; Antiviral agent, anti-HCV</p>Formula:C11H14N4O5Colore e forma:SolidPeso molecolare:282.255-Benzylaminocarbonyl-3'-O-acetyl-2'-O-methyluridine
CAS:<p>5-Benzylaminocarbonyl-3'-O-acetyl-2'-O-methyluridine is a 5-modified pyrimidine nucleoside; 2'-O-Methyl nucleoside.</p>Formula:C20H23N3O8Colore e forma:SolidPeso molecolare:433.41DMT-dI Phosphoramidite
CAS:<p>Phosphoramidite (a modified phosphoramidite monomer) is utilized in the synthesis of oligonucleotides.</p>Formula:C40H47N6O7PColore e forma:SolidPeso molecolare:754.81Angiotensin II (3-8), human
CAS:Angiotensin II (3-8), human is a less effective agonist at the angiotensin AT1 receptor.Colore e forma:Solid(S)-GNA-A(Bz)-phosphoramidite
CAS:<p>(S)-GNA-A(Bz)-phosphoramidite is a Nucleoside Phosphoramidite.</p>Formula:C45H50N7O6PColore e forma:SolidPeso molecolare:815.9Methyl-PEG3-bromide
CAS:<p>Methyl-PEG3-bromide is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>Formula:C7H15BrO3Colore e forma:SolidPeso molecolare:227.15-(Methoxymethyl)-2,4(1H, 3H)-pyrimidinedione
CAS:<p>Intermediates and Building Blocks - Nucleoside base; Heterocyclic Compounds - Pyrimidine</p>Formula:C6H8N2O3Colore e forma:SolidPeso molecolare:156.14(±)-1,2-Diolein
CAS:(±)-1,2-Diolein (1,2-Dioleoyl-rac-glycerol) (1,2-Dioleoyl-rac-glycerol) is a PKC activator. (±)-1,2-Diolein could increases myotubes Ca 2+ influx.Formula:C39H72O5Colore e forma:SolidPeso molecolare:620.993-Deoxy-1,2;5,6-di-O-isopropylidene-D-glucofuranose
CAS:<p>3-Deoxy glucofuranose: used in drug glycosylation, custom synthesized, antiviral against Epstein-Barr virus.</p>Formula:C12H20O5Colore e forma:SolidPeso molecolare:244.28
