
Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.523 prodotti)
- Apoptosi(5.792 prodotti)
- Ciclo cellulare/Checkpoint(4.449 prodotti)
- Cromatina/Epigenetica(2.238 prodotti)
- Segnalazione citoscheletrica(1.383 prodotti)
- Danno al DNA/Riparazione del DNA(2.825 prodotti)
- Endocrinologia/Ormoni(3.507 prodotti)
- Enzima(3.640 prodotti)
- Proteina G/GPCR(8.333 prodotti)
- Immunologia e infiammazione(3.526 prodotti)
- Virus dell'influenza(296 prodotti)
- Segnalazione JAK/STAT(404 prodotti)
- Segnalazione MAPK(1.202 prodotti)
- Trasportatore di membrana/canale ionico(2.790 prodotti)
- Metabolismo(9.448 prodotti)
- Microbiologia/Virologia(6.981 prodotti)
- Neuroscienza(9.926 prodotti)
- Altri inibitori(37.926 prodotti)
- Ossidazione-riduzione(41 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.400 prodotti)
- Proteasi/Proteasoma(1.597 prodotti)
- Cellule staminali e Derivati(831 prodotti)
- Adattatori Tirosin-chinasi(2.016 prodotti)
- Ubiquitinazione(1.650 prodotti)
Mostrare 16 più sottocategorie
Trovati 66641 prodotti di "Inibitori"
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2,5-Dihydroxybenzaldehyde
CAS:<p>2,5-Dihydroxybenzaldehyde (Gentisaldehyde) has antioxidant activity against Mycobacterium avium subsp.</p>Formula:C7H6O3Purezza:99.55% - 99.75%Colore e forma:SolidPeso molecolare:138.12HG-10-102-01
CAS:<p>HG-10-102-01 is an inhibitor of leucine-rich repeat kinase 2 (LRRK2, IC50 of 20.3 nM).</p>Formula:C17H20ClN5O3Purezza:99.59%Colore e forma:SolidPeso molecolare:377.83M4284
CAS:<p>M4284 (M 4284) is a selective and orally active biphenyl mannoside FimH antagonist.</p>Formula:C23H28N2O8Purezza:97.43%Colore e forma:SolidPeso molecolare:460.48m-Chlorophenylbiguanide hydrochloride
CAS:<p>m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.</p>Formula:C8H11Cl2N5Purezza:99.43% - 99.87%Colore e forma:SolidPeso molecolare:248.11Anecortave Acetate
CAS:<p>Anecortave Acetate (NSC-24345), an angiostatic steroid, is used for proteomics research.</p>Formula:C23H30O5Purezza:99.88%Colore e forma:SolidPeso molecolare:386.48D-Leucine
CAS:<p>D-Leucine stops seizures post-onset and lessens long-term potentiation without affecting basal synaptic transmission.</p>Formula:C6H13NO2Purezza:99.67%Colore e forma:SolidPeso molecolare:131.17Ginsenoside C-K
CAS:<p>Ginsenoside C-K (Ginsenoside K) is a bacterial metabolite of G-Rb1 exhibiting anti-inflammatory effects by reducing iNOS and COX-2.</p>Formula:C36H62O8Purezza:99.65% - 99.97%Colore e forma:SolidPeso molecolare:622.878-CHLOROQUINAZOLIN-4(1H)-ONE
CAS:<p>8-CHLOROQUINAZOLIN-4(1H)-ONE is inhibitor of Poly [ADP-ribose] polymerase 1 (human)</p>Formula:C8H5ClN2OPurezza:98.79%Colore e forma:SolidPeso molecolare:180.59NVP-TAE 684
CAS:<p>NVP-TAE 684 (TAE684) is a excellently effective and specific ALK inhibitor(IC50=3 nM).</p>Formula:C30H40ClN7O3SPurezza:98% - 99.82%Colore e forma:SolidPeso molecolare:614.2Theaflavin-3'-Gallate
CAS:<p>Theaflavin-3'-Gallate (Theaflavin 2B) usually comes from the leaves of Camellia sinensis (L.) O. Kuntze,which act as prooxidants and induce oxidative stress.</p>Formula:C36H28O16Purezza:99.21% - 99.89%Colore e forma:SolidPeso molecolare:716.6Pomolic acid
CAS:<p>Pomolic acid has anti-cancer, anti-inflammatory and apoptotic activities, it can induce apoptosis in SK-OV-3 cells, which is mediated by the mitochondrial-</p>Formula:C30H48O4Purezza:96.84% - 99.79%Colore e forma:SolidPeso molecolare:472.7Danofloxacin
CAS:<p>Danofloxacin (Danofloxacin free base) is a fluoroquinolone antibiotic used in veterinary medicine.</p>Formula:C19H20FN3O3Purezza:99.77% - 99.8%Colore e forma:SolidPeso molecolare:357.38Guanosine 5'-triphosphate trisodium salt
CAS:<p>5'-GTP trisodium salt activates G proteins, regulates cell proliferation/apoptosis, and aids DNA/RNA biosynthesis.</p>Formula:C10H13N5Na3O14P3Purezza:98.74% - 99.45%Colore e forma:White PowderPeso molecolare:589.13Fexaramine
CAS:<p>Fexaramine is a small molecule farnesoid X receptor (FXR) agonist with 100-fold increased affinity compared to natural compounds.</p>Formula:C32H36N2O3Purezza:98.87% - 99.61%Colore e forma:SolidPeso molecolare:496.64JNJ-7777120
CAS:<p>JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.</p>Formula:C14H16ClN3OPurezza:99.83% - 99.96%Colore e forma:SolidPeso molecolare:277.75(Z)-LFM-A13
CAS:(Z)-LFM-A13(IC50=2.5 μM), a specific Bruton's tyrosine kinase (BTK), is more than 100-fold specificity than other protein kinases, such as JAK1, JAK2, HCK, EGFR, and IRK.Formula:C11H8Br2N2O2Purezza:99.88%Colore e forma:SolidPeso molecolare:360PI-103
CAS:<p>PI-103 is a potent, cell-permeable, ATP-competitive inhibitor of PI3K family members (IC50s: 2/3/3/15/30/23 nM for p110α/β/δ/γ, mTOR, and DNA-PK).</p>Formula:C19H16N4O3Purezza:97.79% - 99.3%Colore e forma:SolidPeso molecolare:348.363-Methyltoxoflavin
CAS:<p>3-Methyltoxoflavin (3-methyl toxoflavin) is an effective inhibitor of protein disulfide isomerase (PDI) and its IC50 value is 170 nM.</p>Formula:C8H9N5O2Purezza:99.81%Colore e forma:SolidPeso molecolare:207.194μ8C
CAS:<p>4μ8C (IRE1 Inhibitor III)(IC50=76 nM) is an effective and specific IRE1 Rnase inhibitor.</p>Formula:C11H8O4Purezza:97.48% - 98.45%Colore e forma:SolidPeso molecolare:204.18SMIFH2
CAS:<p>SMIFH2 is formin homology 2 (FH2) domains inhibitor.</p>Formula:C15H9BrN2O3SPurezza:97.41%Colore e forma:SolidPeso molecolare:377.21[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
<p>[D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and</p>Formula:C76H103N21O18SPurezza:99.75%Colore e forma:SolidPeso molecolare:1630.82Methenamine Hippurate
CAS:<p>Methenamine Hippurate is a component of Hiprex, with antibacterial activity.</p>Formula:C15H21N5O3Purezza:99.69% - 99.72%Colore e forma:White Crystalline PowderPeso molecolare:319.36Lophanthoidin E
CAS:<p>Lophanthoidin E is a kind of natural product derived from the herbs of Rabdosia lophanthoides.</p>Formula:C22H30O7Purezza:98.00%Colore e forma:SolidPeso molecolare:406.47Nelociguat
CAS:<p>Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.</p>Formula:C19H17FN8O2Purezza:99.19%Colore e forma:SolidPeso molecolare:408.39Thalidomide-4-OH
CAS:<p>Thalidomide-4-OH, a Thalidomide-derived Cereblon binder, recruits CRBN and serves as a PROTAC linker.</p>Formula:C13H10N2O5Purezza:99.59%Colore e forma:SolidPeso molecolare:274.23Jervine
CAS:<p>Jervine inhibits Smoothened, blocking Hedgehog signaling and GLI1 transcription activation.</p>Formula:C27H39NO3Purezza:99.20% - 99.86%Colore e forma:Needles From Methanol + Water SolidPeso molecolare:425.6Pantoprazole sodium
CAS:<p>Pantoprazole sodium is a proton pump inhibitor that irreversibly blocks gastric acid secretion by bonding with H+/K+-ATPase.</p>Formula:C16H14F2N3NaO4SPurezza:96.92% - 99.81%Colore e forma:White To Off-White SolidPeso molecolare:405.35SU5205
CAS:<p>SU5205 is a VEGFR2 inhibitor.</p>Formula:C15H10FNOPurezza:99.62% - 99.67%Colore e forma:SolidPeso molecolare:239.24AMG-47a
CAS:<p>AMG-47a inhibits Lck, T cell growth, and degrades KRAS oncoprotein, affecting EGFP-KRASG12V but not EGFP.</p>Formula:C29H28F3N5O2Purezza:98%Colore e forma:SolidPeso molecolare:535.56PR-619
CAS:<p>PR-619 (2,6-Diamino-3,5-dithiocyanopyridine) is a DUB inhibitor. PR-619 induces endoplasmic reticulum stress and activates autophagy. Cost-effective and quality-assured.</p>Formula:C7H5N5S2Purezza:97.25% - >99.99%Colore e forma:SolidPeso molecolare:223.28Mandelic acid
CAS:<p>Mandelic acid is a metabolite of adrenaline and found in skincare, used as an analytical reagent, dye precursor, and linked to phenylketonuria.</p>Formula:C8H8O3Purezza:99.45% - 99.95%Colore e forma:White Solid SolidPeso molecolare:152.15Cefoperazone
CAS:<p>Cefoperazone (Medocef) inactivates PBPs, disrupting bacterial cell wall synthesis and division; inhibits rMrp2 [3H]E217βG uptake (IC50: 199 μM).</p>Formula:C25H27N9O8S2Purezza:98.99% - 99.76%Colore e forma:SolidPeso molecolare:645.67Glycinamide Hydrochloride
CAS:<p>Glycinamide Hydrochloride (2-Aminoacetamide hydrochloride) is a glycine pro-drug.</p>Formula:C2H7ClN2OPurezza:98% - 99.7%Colore e forma:White To Off-White SolidPeso molecolare:110.5416-Epivoacarpine
CAS:<p>16-Epivoacarpine is a natural product from Gelsemium elegans.</p>Formula:C21H24N2O4Purezza:98.12% - 99.98%Colore e forma:SolidPeso molecolare:368.43Epiberberine
CAS:<p>1.</p>Formula:C20H18NO4Purezza:98.52% - 99.59%Colore e forma:SolidPeso molecolare:336.36Ca-DTPA trisodium salt hydrate
CAS:<p>Ca-DTPA trisodium hydrate: metal chelator, antidote for cadmium poisoning, non-toxic CMV replication inhibitor.</p>Formula:C14H20CaN3NaO11Purezza:≥98%Colore e forma:SolidPeso molecolare:469.393Fasiglifam
CAS:<p>Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.</p>Formula:C29H32O7SPurezza:99.82% - 99.9%Colore e forma:SolidPeso molecolare:524.63Phellamurin
CAS:<p>Phellamurin blocks intestinal P-glycoprotein dose-dependently and it seriously interacts with cyclosporin; coadministration should be avoided.</p>Formula:C26H30O11Purezza:97.91%Colore e forma:SolidPeso molecolare:518.51DS-1971a
CAS:<p>DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.</p>Formula:C20H21ClFN5O3SPurezza:99.66%Colore e forma:SolidPeso molecolare:465.93Argireline
CAS:<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Formula:C34H60N14O12SPurezza:96.79% - 99.65%Colore e forma:White PowderPeso molecolare:888.99SU9516
CAS:<p>SU9516 is a potent CDK2 inhibitor, with an IC50 of 22 nM, and also has inhibitory effects on CDK1 and CDK4, with IC50s of 40 nM and 200 nM, respectively.</p>Formula:C13H11N3O2Purezza:99.34% - 99.87%Colore e forma:SolidPeso molecolare:241.25Fedratinib
CAS:Fedratinib (TG-101348) (TG101348) is an ATP-competitive inhibitor of JAK2 (IC50: 3 nM) with significantly less potent activity against JAK3.Formula:C27H36N6O3SPurezza:97.31% - 99.96%Colore e forma:SolidPeso molecolare:524.68Ibuprofen Lysine
CAS:<p>Ibuprofen Lysine (Neoprofen) is a non-steroidal anti-inflammatory drug.</p>Formula:C19H32N2O4Purezza:99.26%Colore e forma:CoaPeso molecolare:352.47Purpurogallin
CAS:<p>Purpurogallin: natural phenol from Quercus spp., xanthine oxidase inhibitor (IC50: 0.2μM), antioxidant, anti-inflammatory.</p>Formula:C11H8O5Purezza:96.44%Colore e forma:SolidPeso molecolare:220.187-Ethoxyresorufin
CAS:<p>7-Ethoxyresorufin (Resorufin ethyl ether) (7-ER) is a fluorometric substrate for and competitive inhibitor of cytochrome P450, especially CYP1A1.</p>Formula:C14H11NO3Purezza:99.09% - 99.62%Colore e forma:Red SolidPeso molecolare:241.24REVERSE T3
CAS:<p>Reverse T3 (3,3',5'-triiodo-L-thyronine) inhibits the increase of sodium current generated by other thyroid hormone analogs in neonatal rat myocytes.</p>Formula:C15H12I3NO4Purezza:95.99% - 97.89%Colore e forma:PowderPeso molecolare:650.97Isocurcumenol
CAS:<p>1. Isocurcumenol inhibits 5α-reductase which converts testosterone to dihydrotestosterone (DHT).</p>Formula:C15H22O2Purezza:99.29% - ≥95%Colore e forma:SolidPeso molecolare:234.332-Phenylethylamine hydrochloride
CAS:<p>2-Phenylethylamine hydrochloride (benzeneethanamine hydrochloride) acts as neuromodulator in the central nervous system.</p>Formula:C8H12ClNPurezza:99.94%Colore e forma:SolidPeso molecolare:157.64Deoxythymidine triphosphate
CAS:<p>Deoxythymidine triphosphate (dTTP) is one of the four nucleoside triphosphates that are used in the in vivo synthesis of DNA.</p>Formula:C10H14N2Na3O14P3Purezza:99.78%Colore e forma:White Amorphous PowderPeso molecolare:548.11Licochalcone C
CAS:<p>Licochalcone C: antioxidant, anti-bacterial, supports heart health, anti-inflammatory, fights cancer cells.</p>Formula:C21H22O4Purezza:95% - 99.93%Colore e forma:SolidPeso molecolare:338.4
