
Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.524 prodotti)
- Apoptosi(5.793 prodotti)
- Ciclo cellulare/Checkpoint(4.452 prodotti)
- Cromatina/Epigenetica(2.242 prodotti)
- Segnalazione citoscheletrica(1.382 prodotti)
- Danno al DNA/Riparazione del DNA(2.826 prodotti)
- Endocrinologia/Ormoni(3.507 prodotti)
- Enzima(3.640 prodotti)
- Proteina G/GPCR(8.333 prodotti)
- Immunologia e infiammazione(3.527 prodotti)
- Virus dell'influenza(296 prodotti)
- Segnalazione JAK/STAT(404 prodotti)
- Segnalazione MAPK(1.203 prodotti)
- Trasportatore di membrana/canale ionico(2.792 prodotti)
- Metabolismo(9.449 prodotti)
- Microbiologia/Virologia(6.981 prodotti)
- Neuroscienza(9.926 prodotti)
- Altri inibitori(37.921 prodotti)
- Ossidazione-riduzione(41 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.400 prodotti)
- Proteasi/Proteasoma(1.597 prodotti)
- Cellule staminali e Derivati(830 prodotti)
- Adattatori Tirosin-chinasi(2.015 prodotti)
- Ubiquitinazione(1.650 prodotti)
Mostrare 16 più sottocategorie
Trovati 66639 prodotti di "Inibitori"
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API-1
CAS:<p>API-1 (NSC-177223) is a potent inhibitor of Akt. It induces GSK3-dependent, β-TrCP- and FBXW7-mediated Mcl-1 degradation, resulting in induction of apoptosis .</p>Formula:C13H15N5O6Purezza:97.15%Colore e forma:SolidPeso molecolare:337.29Dipsacoside B
CAS:<p>Dipsacoside B is a major bioactive saponin used as a marker.</p>Formula:C53H86O22Purezza:99.03% - 99.81%Colore e forma:SolidPeso molecolare:1075.24Palmatine
CAS:<p>Palmatine, also known as Burasaine, inhibits dopamine production and may treat flavivirus, jaundice, dysentery, hypertension, and liver issues.</p>Formula:C21H22NO4Purezza:96.28% - 99.49%Colore e forma:SolidPeso molecolare:352.4Dimethyl-d6 Sulfoxide
CAS:<p>Dimethyl-d6 Sulfoxide (DMSO-d6) replaces H with deuterium; it's a solvent in NMR spectroscopy.</p>Formula:C2D6OSPurezza:98%Colore e forma:LiquidPeso molecolare:84.17Syrosingopine
CAS:<p>Syrosingopine is a dual inhibitor of MCT1 and MCT4, 60 times more potent against MCT4, preventing lactate and H+ efflux.Cost-effective and quality-assured.</p>Formula:C35H42N2O11Purezza:99.25% - 99.78%Colore e forma:SolidPeso molecolare:666.711-Stearoyl-sn-glycero-3-phosphocholine
CAS:<p>1-Stearoyl-sn-glycero-3-phosphocholine (L-ALPHA-LYSOPHOSPHATIDYLCHOLINE, STEAROY) is a chemical used in lipid metabolism studies</p>Formula:C26H54NO7PPurezza:99.61%Colore e forma:SolidPeso molecolare:523.68DDR1-IN-1 dihydrochloride
CAS:<p>DDR1-IN-1 dihydrochloride: potent DDR1 kinase inhibitor; IC50=105 nM; 4x less effective on DDR2 (IC50=413 nM).</p>Formula:C30H33Cl2F3N4O3Colore e forma:SolidPeso molecolare:625.51N2,N2-Dimethylguanosine
CAS:<p>Urinary N2,N2-Dimethylguanosine levels higher in colorectal cancer than in villous adenoma or healthy adults.</p>Formula:C12H17N5O5Purezza:98.01%Colore e forma:White SolidPeso molecolare:311.29Abz-FR-K(Dnp)-P-OH acetate
<p>Abz-FR-K(Dnp)-P-OH acetate is an excellent angiotensin I-converting enzyme (ACE) substrate with a Km value of 4.0 μM and a kcat value of 210s-1.</p>Formula:C41H53N11O12Purezza:>99.99%Colore e forma:SolidPeso molecolare:891.95Loureirin B
CAS:<p>Loureirin B suppresses fibrosis by modulating MMPs/TIMPs, hindering fibroblast growth, and targeting TGF-β1/Smad2/3 pathway.</p>Formula:C18H20O5Purezza:99.33% - 99.86%Colore e forma:SolidPeso molecolare:316.35Spermine tetrahydrochloride
CAS:<p>Spermine tetrahydrochloride, a polyamine in all eukaryotic cells, protects DNA from free radicals.</p>Formula:C10H26N4·4HClPurezza:99.75% - 99.82%Colore e forma:SolidPeso molecolare:348.18Nelfinavir Mesylate
CAS:<p>Nelfinavir Mesylate (Viracept) is an effective HIV protease inhibitor (Ki: 2 nM).</p>Formula:C33H49N3O7S2Purezza:95.81% - 98.51%Colore e forma:A White Or Almost White PowderPeso molecolare:663.89Metergoline
CAS:<p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>Formula:C25H29N3O2Purezza:99.83% - 99.97%Colore e forma:SolidPeso molecolare:403.523-hydroxymorindone
CAS:<p>3-hydroxymorindone is a natural product from Morinda citrifolia. 3-hydroxymorindone is a pigment.</p>Formula:C15H10O6Purezza:98.7% - 99.24%Colore e forma:SolidPeso molecolare:286.24γ-decalactone
CAS:<p>Gamma-decalactone (Decan-4-olide) is a food additive with a fruity peach flavor. Ricinoleic acid is used as a substrate in the production of γ-Decalactone.</p>Formula:C10H18O2Purezza:≥95%Colore e forma:LiquidPeso molecolare:170.25Canertinib
CAS:<p>Canertinib (CI-1033), a pan-erbB inhibitor, effectively targets esophageal cancer in vitro/vivo, altering metabolism and reducing growth and hypoxia.</p>Formula:C24H25ClFN5O3Purezza:98% - >99.99%Colore e forma:White Or Similar To White Crystalline PowderPeso molecolare:485.942-Methoxyestradiol
CAS:<p>2-ME2, an estradiol derivative, hinders angiogenesis and tumor growth, causes cell apoptosis, and stops mitosis.</p>Formula:C19H26O3Purezza:98% - 99.95%Colore e forma:Off-White SolidPeso molecolare:302.41Hordenine hydrochloride
CAS:<p>Hordenine hydrochloride is a biochemical that inhibits the activity of PDK3, inhibits quorum sensing, and acts as an antibiofilm agent against bacteria.</p>Formula:C10H16ClNOColore e forma:SolidPeso molecolare:201.693Azvudine
CAS:<p>Azvudine (FNC) is a powerful NRTI effective against HIV, HBV, HCV, and resistant strains.</p>Formula:C9H11FN6O4Purezza:99.76% - >99.99%Colore e forma:SolidPeso molecolare:286.223-Feruloyl-4-caffeoylquinic acid
CAS:<p>3-Feruloyl-4-caffeoylquinic acid: a chlorogenic acid isomer, key in coffee quality, flavor, and health benefits.</p>Formula:C26H26O12Purezza:99.06% - 99.89%Colore e forma:SolidPeso molecolare:530.48Propargyl-PEG12-bromide
CAS:<p>Propargyl-PEG12-bromide is a PEG-based PROTAC linker used to synthesize PROTACs.</p>Formula:C29H55BrO13Purezza:≥98%Colore e forma:SolidPeso molecolare:691.64EI1
CAS:<p>EI1 (Ezh2 inhibitor) is a potent and selective EZH2 inhibitor with IC50 of 15 nM and 13 nM for EZH2 (WT) and EZH2 (Y641F), respectively.</p>Formula:C23H26N4O2Purezza:99.93%Colore e forma:SolidPeso molecolare:390.48CPI-455
CAS:<p>CPI-455 is a specific KDM5 inhibitor.</p>Formula:C16H14N4OPurezza:97.87% - 99.03%Colore e forma:SolidPeso molecolare:278.31Thymine
CAS:<p>Thymine: Derived from DNA hydrolysis or methylcyanoacetylurea, found in DNA (not RNA), binds adenine, used in biochemical research.</p>Formula:C5H6N2O2Purezza:99.77% - 99.97%Colore e forma:SolidPeso molecolare:126.11PRT4165
CAS:<p>PRT4165 (NSC600157) is a potent PRC1-mediated H2A ubiquitylation inhibitor.</p>Formula:C15H9NO2Purezza:98.91% - 99.6%Colore e forma:SolidPeso molecolare:235.24VU0155041
CAS:<p>VU0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, at human/rat).</p>Formula:C14H15Cl2NO3Purezza:99.52% - 99.56%Colore e forma:SolidPeso molecolare:316.18Azido-PEG2-azide
CAS:<p>Azido-PEG2-azide is a PEG-based PROTAC linker that can be used in PROTAC synthesis.</p>Formula:C6H12N6O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:200.2PD 128042
CAS:<p>PD 128042 (CI 976) is a potent orally active and selective ACAT inhibitor(IC50: 73 nM) and a potent lysophospholipid acyltransferase(LPAT) inhibitor.</p>Formula:C23H39NO4Purezza:99.79%Colore e forma:SolidPeso molecolare:393.56GANT 61
CAS:<p>GANT 61 (GANT61) is an inhibitor for Gli1 and Gli2.</p>Formula:C27H35N5Purezza:97.59% - >99.99%Colore e forma:SolidPeso molecolare:429.6FDI-6
CAS:<p>FDI-6 is an effective and selective inhibitor of FOXM1 that blocks DNA binding. FDI-6 binds to the FOXM1 protein and downregulates FOXM1-activated genes.</p>Formula:C19H11F4N3OS2Purezza:98.92% - >99.99%Colore e forma:SolidPeso molecolare:437.43Flavopiridol hydrochloride
CAS:<p>Flavopiridol hydrochloride (MDL 107826A), an inhibitor of cyclin-dependent kinase, is a synthetic N-methylpiperidinyl chlorophenyl flavone compound.</p>Formula:C21H21Cl2NO5Purezza:98.87% - 99.88%Colore e forma:SolidPeso molecolare:438.3ABT-737
CAS:<p>ABT-737 is a BH3 mimetic and an inhibitor of Bcl-2, Bcl-xL, and Bcl-w. ABT-737 exhibits antitumor activity and anti-aging activity. Cost-effective and quality-assured.</p>Formula:C42H45ClN6O5S2Purezza:98.15% - >99.99%Colore e forma:SolidPeso molecolare:813.43Dimethyl fumarate
CAS:<p>Dimethyl fumarate (DMF) is an orally Nrf2 activator. Dimethyl fumarate has antimicrobial and anti-inflammatory activities. Cost-effective and quality-assured.</p>Formula:C6H8O4Purezza:90.51% - >99.99%Colore e forma:White To Off-White Powder White Crystalline PowderPeso molecolare:144.132-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1λ*6*-BENZO[D]ISOTHIAZOL-3-ONE
CAS:<p>2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE targets the Neutrophil elastase (human).</p>Formula:C8H6ClNO3SPurezza:97.28%Colore e forma:SolidPeso molecolare:231.66YM-201636
CAS:<p>YM201636 (IC50=33 nM), a specific PIKfyve inhibitor, is less effective to p110α and insensitive to Fabl, which is yeast orthologue.</p>Formula:C25H21N7O3Purezza:93.28% - 98.3%Colore e forma:SolidPeso molecolare:467.48Pyruvic acid
CAS:<p>Pyruvic acid, key in metabolizing carbs, proteins, and fats, builds up in tissue, notably nerves, if thiamine is deficient.</p>Formula:C3H4O3Purezza:95.31%Colore e forma:LiquidPeso molecolare:88.06Chemerin-9 (149-157) acetate
<p>Chemerin-9 (149-157) acetate, a nonapeptide C-terminal fragment of chemerin, retains full protein's activity as chemerinR agonist.</p>Formula:C56H70N10O15Purezza:99.93%Colore e forma:SolidPeso molecolare:1123.23γ-Linolenic acid
CAS:<p>gamma-Linolenic acid (gamolenic acid), is an unsaturated fatty acid synthesized from linoleic acid (LA) by the enzyme delta-6-desaturase.</p>Formula:C18H30O2Purezza:95% - 98.5%Colore e forma:SolidPeso molecolare:278.43Liensinine diperchlorate
CAS:<p>Liensinine Diperchlorate is an isoquinoline alkaloid extracted from the embryonic seeds of the sacred lotus.</p>Formula:C37H44Cl2N2O14Purezza:99.8% - ≥95%Colore e forma:SolidPeso molecolare:811.67Remibrutinib
CAS:<p>Remibrutinib inhibits BTK activity with an IC50 value of 0.023 μM in blood.</p>Formula:C27H27F2N5O3Purezza:99.5% - 99.81%Colore e forma:SolidPeso molecolare:507.536-O-Methyl Guanosine
CAS:<p>6-O-Methyl Guanosine inhibit colony-forming ability in a malignant xeroderma pigmentosum cell line.</p>Formula:C11H15N5O5Purezza:97.5%Colore e forma:SolidPeso molecolare:297.27[Sar9] Substance P acetate(77128-75-7 free base)
<p>[Sar9]-Substance P acetate, an NK-1 receptor agonist, mimics SP's effect on progesterone metabolism.</p>Formula:C66H104N18O15SPurezza:96.67%Colore e forma:SolidPeso molecolare:1421.71Navitoclax dihydrochloride
CAS:<p>Navitoclax dihydrochloride is a synthetic Bcl-2 antagonist with potential cancer-fighting properties.</p>Formula:C47H57Cl3F3N5O6S3Colore e forma:SolidPeso molecolare:1047.54[Leu5]-Enkephalin acetate(58822-25-6 free base)
<p>Endogenous [Leu5]-Enkephalin acetate is a δ- and μ-opioid receptor agonist involved in pain; Ki: δ=4.0 nM, μ=3.4 nM.</p>Formula:C30H41N5O9Purezza:99.28%Colore e forma:SolidPeso molecolare:615.68ML239
CAS:<p>ML239 (CID-49843203) is a potent and selective inhibitor of breast cancer stem cells, with an IC50 of 1.16 μM.</p>Formula:C13H10Cl3N3O2Purezza:99.13%Colore e forma:SolidPeso molecolare:346.6LOX-IN-3 dihydrochloride monohydrate
CAS:<p>LOX-IN-3 dihydrochloride monohydrate is an oral lysyl oxidase inhibitor for research in fibrosis, cancer, and angiogenesis.</p>Formula:C13H17Cl2FN2O3SColore e forma:SolidPeso molecolare:371.25Ramosetron
CAS:<p>Ramosetron 是一种血清素 5-HT3 受体拮抗剂,用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。</p>Formula:C17H17N3OPurezza:98.84%Colore e forma:SolidPeso molecolare:279.34Articaine
CAS:<p>Articaine (Hoe-045 free base), an amide anesthetic featuring an ester group, effectively relieves pain by reversibly binding to the α-subunit of the voltage-</p>Formula:C13H20N2O3SColore e forma:SolidPeso molecolare:284.37Stearic acid
CAS:<p>Stearic acid reduces tumor load, cuts visceral fat, gels foods/pharma, boosts insulin signaling, and ups milk yield without weight impact.</p>Formula:C18H36O2Purezza:99.40% - 99.81%Colore e forma:White Solid LeafletsPeso molecolare:284.48NBI-31772 hydrate
<p>NBI-31772 hydrate blocks IGF and IGFBPs binding, freeing IGF-I with Ki 1-24 nM; it has anxiolytic and antidepressant effects.</p>Formula:C17H13NO8Colore e forma:SolidPeso molecolare:372.82

