2-Epi-darunavir

CAS: 850141-19-4

Ref. 3D-AJB14119

Product Information

• Name: 2-Epi-darunavir
• Brand: Biosynth
• Description: 2-Epi-darunavir is a peptide that acts as an activator of the HIV-1 protease. It has been shown to be a potent inhibitor of HIV-1 protease, with IC50 values in the low nanomolar range. The 2-Epi-darunavir peptide binds to the active site of HIV-1 protease, blocking access by other molecules and preventing cleavage at the P1' position on the substrate. This results in a conformational change that prevents its interaction with the binding site on HIV-1 gp41. The 2-Epi darunavir peptide also inhibits protein interactions with ion channels and receptor proteins, which may inhibit cellular processes such as cell proliferation and apoptosis.

Chemical properties

• Molecular weight: 547.7 g/mol
• Formula: C₂₇H₃₇N₃O₇S
• Purity: Min. 95%