Product Information
Cuspidiol is a natural product that has been identified as a novel inhibitor of the enzyme phosphatase 1B (PTP1B). It is a potent and selective inhibitor of PTP1B, with an IC50 value of 0.27 μM. Cuspidiol may function by binding to the active site of the PTP1B enzyme, blocking access to its ATP substrate, and inhibiting its activity. Cuspidiol has also been shown to inhibit transcriptional activation of genes in human cells by suppressing the expression of c-Fos protein. This inhibition is specific for PTP1B and does not affect other phosphatases. The mechanism by which cuspidiol inhibits PTP1B is currently unknown but may involve binding at the active site or interference with substrate binding.
Chemical properties
Technical inquiry about: 3D-BCA59396 Cuspidiol
If you want to request a quotation or place an order, please instead add the desired products to your cart and then request a quotation or order from the cart. It is faster, cheaper, and you will be able to benefit from the available discounts and other advantages.
