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Gavestinel
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Gavestinel

CAS: 153436-38-5

Ref. 3D-DGA43638

1mg
138.00 €
2mg
194.00 €
5mg
310.00 €
10mg
436.00 €
25mg
801.00 €
Estimated delivery in United States, on Thursday 2 Jan 2025

Product Information

Name:
Gavestinel
Synonyms:
  • 1H-Indole-2-carboxylic acid, 4,6-dichloro-3-[(1E)-3-oxo-3-(phenylamino)-1-propen-1-yl]-, sodium salt (1:1)
  • 1H-Indole-2-carboxylic acid, 4,6-dichloro-3-[(1E)-3-oxo-3-(phenylamino)-1-propenyl]-, monosodium salt
  • 1H-Indole-2-carboxylic acid, 4,6-dichloro-3-[3-oxo-3-(phenylamino)-1-propenyl]-, monosodium salt, (E)-
  • 1H-Indole-2-carboxylicacid, 4,6-dichloro-3-[3-oxo-3-(phenylamino)-1-propenyl]-, monosodium salt,(E)-
  • Gv 150526A
Description:

Gavestinel is a novel anti-platelet agent that is undergoing clinical trials for the treatment of stroke. Gavestinel binds to and blocks the P2Y12 receptor in platelets, which inhibits platelet aggregation and prevents formation of blood clots. In addition to its anti-platelet effects, gavestinel also has been shown to protect neurons against ischemic brain damage. This protection is likely due to the inhibition of neuronal death by cation channels and protein transport, as well as an increase in the release of gamma-aminobutyric acid (GABA) from GABAergic neurons. Gavestinel also inhibits glutamate release from the presynaptic neuron, leading to less excitotoxicity at postsynaptic sites. The mechanism of action has been elucidated using kinetic data obtained from binding assays with recombinant proteins. Gavestinel is also an inhibitor of ATP channels that are found in many types of cells, including glial cells.

Notice:
Our products are intended for lab use only. For any other use, please contact us.
Brand:
Biosynth
Long term storage:
Notes:

Chemical properties

Molecular weight:
397.19 g/mol
Formula:
C18H11Cl2N2NaO3
Purity:
Min. 95%
MDL:
Melting point:
Boiling point:
Flash point:
Density:
Concentration:
EINECS:
Merck:
HS code:

Hazard Info

UN Number:
EQ:
Class:
H Statements:
P Statements:
Forbidden to fly:
Hazard Info:
Packing Group:
LQ:

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