N-Desmethyl eletriptan

Ref. 3D-DGA52555

Product Information

• Name: N-Desmethyl eletriptan
• Brand: Biosynth
• Description: N-Desmethyl eletriptan is a metabolite of eletriptan that has been shown to inhibit serotonin release. It has been tested in clinical trials and found to be effective in the treatment of migraine headaches. The pharmacokinetics of N-desmethyl eletriptan have been studied in humans and show that it rapidly penetrates the blood brain barrier, with plasma concentrations peaking at about 1 hour after ingestion. The drug also inhibits P-glycoprotein activity, which may increase its bioavailability by preventing it from being excreted through the kidneys. N-Desmethyl eletriptan is not approved for use in children or pregnant women, as there are no clinical data available on these populations.

Chemical properties

• Molecular weight: 368.5 g/mol
• Formula: C₂₁H₂₄N₂O₂S
• Purity: Min. 95%