Ospemifene

CAS: 128607-22-7

Ref. 3D-FC57468

Product Information

• Name: Ospemifene
• Synonyms: (deaminohydroxy)toremifene2-[4-[(1Z)-4-Chloro-1,2-diphenyl-1-buten-1-yl]phenoxy]ethanol, 2-[4-[(1Z)-4-Chloro-1,2-diphenyl-1-buten-1-yl]phenoxy]ethanol, 2-[4-[4-Chloro-1,2-diphenyl-1(Z)-butenyl]phenoxy]ethanol, 2-{4-[(1Z)-4-chloro-1,2-diphenylbut-1-en-1-yl]phenoxy}ethanol, Ethanol, 2-[4-(4-chloro-1,2-diphenyl-1-butenyl)phenoxy]-, (Z)-, Ethanol, 2-[4-[(1Z)-4-chloro-1,2-diphenyl-1-buten-1-yl]phenoxy]-, Ethanol, 2-[4-[(1Z)-4-chloro-1,2-diphenyl-1-butenyl]phenoxy]-, FC-1271a, Fc 1271, Osphena, Senshio

Description

2-[4-[(1Z)-4-Chloro-1,2-diphenyl-1-buten-1-yl]phenoxy]ethanol is a selective estrogen receptor modulator that has been shown to inhibit the growth of breast cancer cells in mice. It binds to the estrogen receptor (ER) and inhibits its transcriptional activity by competing with estradiol for binding. 2-[4-[(1Z)-4-Chloro-1,2-diphenyl-1-buten-1-yl]phenoxy]ethanol can be used as a postmenopausal hormonal therapy in women who are at an increased risk for breast cancer. This drug has been shown to have genotoxic activity and may cause dyspareunia and carcinogenic potential.

• Brand: Biosynth

Chemical properties

• Molecular weight: 378.89 g/mol
• Formula: C₂₄H₂₃ClO₂
• Purity: Min. 95%
• Color/Form: Powder
• InChI: InChI=1S/C24H23ClO2/c25-16-15-23(19-7-3-1-4-8-19)24(20-9-5-2-6-10-20)21-11-13-22(14-12-21)27-18-17-26/h1-14,26H,15-18H2/b24-23-
• InChI key: InChIKey=LUMKNAVTFCDUIE-VHXPQNKSSA-N
• SMILES: OCCOc1ccc(/C(=C(/CCCl)c2ccccc2)c2ccccc2)cc1