Sarafotoxin 6c

Ref. 3D-FS73598

Product Information

• Name: Sarafotoxin 6c
• Brand: Biosynth
• Description: Sarafotoxin 6c is a potent, selective, and noncompetitive endothelin-1 receptor antagonist. Sarafotoxin 6c binds to the extracellular domain of the endothelin-1 receptor and prevents endothelin-1 from binding, thereby inhibiting its activity. Sarafotoxin 6c has been shown to inhibit the production of intracellular Ca2+ in mesenteric artery cells. Sarafotoxin 6c also inhibits the enzymatic inactivation of endothelin-1 by carboxypeptidases and calpains. Sarafotoxin 6c has been shown to be effective against a number of infectious diseases including myocardial infarction.

Chemical properties

• Molecular weight: 2,515.76 g/mol
• Formula: C₁₀₃H₁₄₇N₂₇O₃₇S₅
• Purity: Min. 95%