CGP 77675

CAS: 234772-64-6

Ref. 3D-JJA77264

Product Information

• Name: CGP 77675
• CAS: 234772-64-6

Description

CGP 77675 is a voltage-dependent calcium channel inhibitor that has shown to be an effective chemotherapeutic agent in prostate cancer cells. It has been shown to inhibit the activity of MMP-9, which is an enzyme involved in the degradation of the extracellular matrix and tumor growth. CGP 77675 also inhibits the activity of growth factor-β1, which is a protein that regulates cell proliferation and differentiation. In addition, it inhibits dna binding activity and chemical inhibitors in prostate cancer cells. The drug has significant cytotoxicity on carcinoma cell lines and basic fibroblast cells. CGP 77675 selectively binds to kinases with basic amino acid residues near the ATP binding site (e.g., epidermal growth factor receptor).

• Brand: Biosynth

Chemical properties

• Molecular weight: 443.54 g/mol
• Formula: C₂₆H₂₉N₅O₂
• Purity: Min. 95%