![[D-Ala2,Met5]-Enkephalinamide](https://static.cymitquimica.com/products/3D/img/PEK-4117.png "Click to enlarge")
Product Information
- Tyr-D-Ala-Gly-Phe-Met-NH2 • AcOH • H2O
- (D-Ala2,D-Met5)-Enkephalin
- H-Tyr-D-Ala-Gly-Phe-D-Met-OH
D-Ala2,Met5]-Enkephalinamide is a potent endogenous opioid peptide that binds to opioid receptors and has been shown to have both antinociceptive and depressant effects. It has been shown to be effective in a model system of pain, acting on the descending antinociceptive pathway from the rostral ventromedial medulla (RVM) to the spinal cord. D-Ala2,Met5]-Enkephalinamide has also been observed to inhibit locomotor activity in CD1 mice at sub-effective doses. D-Ala2,Met5]-Enkephalinamide has been shown to act through activation of both G protein-coupled mu opioids receptors and G protein-coupled delta opioid receptors.
Chemical properties
Technical inquiry about: 3D-PEK-4117 [D-Ala2,Met5]-Enkephalinamide
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