Product Information
Name:GNE-0439
Brand:Biosynth
Description:GNE-0439 is a small molecule that inhibits the activity of the sodium channel. It binds to the extracellular domain of the alpha subunit and blocks voltage-gated sodium channels, which are necessary for action potential propagation. GNE-0439 is a potent inhibitor of neuronal and cardiomyocyte Na(+) current, with an IC50of 2 nM in rat neurons and 1 μM in human atrial myocytes. In addition, GNE-0439 inhibits voltage-gated potassium channels (IC50 = 200 nM) and glutamate receptors (IC50 = 2 μM).GNE-0439 is a high purity compound that has been synthesized according to Good Manufacturing Practices (GMP). It is >98% pure as determined by HPLC analysis.
Notice:Our products are intended for lab use only. For any other use, please contact us.
Chemical properties
Molecular weight:345.5 g/mol
Formula:C21H31NO3
Purity:Min. 95%
Technical inquiry about: GNE-0439
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