Tetranor-pgdm

CAS: 70803-91-7

Ref. 3D-VCA80391

Product Information

• Name: Tetranor-pgdm
• Brand: Biosynth
• Description: Tetranor-pgdm is a peptide that binds to the G protein-coupled chemokine receptor CXCR1, which may inhibit the binding of chemokines to CXCR1. Tetranor-pgdm has been shown to inhibit the activity of ion channels and ligand-gated ion channels, such as nicotinic acetylcholine receptors and voltage-gated potassium channels. Tetranor-pgdm is a potent inhibitor of the β2 subunit of the calcium channel, which is an important target for antihypertensive drugs. Tetranor-pgdm also inhibits the production of inflammatory cytokines in vitro and decreases blood pressure in vivo.

Chemical properties

• Molecular weight: 328.36 g/mol
• Formula: C₁₆H₂₄O₇
• Purity: Min. 95%