1-Epi-darunavir

CAS: 1546918-95-9

Ref. 3D-WLC91895

Product Information

• Name: 1-Epi-darunavir
• Brand: Biosynth
• Description: 1-Epi-darunavir is a potent HIV protease inhibitor that blocks the cleavage of polyproteins that are necessary for the assembly and release of new viruses. It is an epimer of darunavir and has been shown to be more potent than its parent compound. 1-Epi-darunavir binds to the active site of HIV protease and prevents the formation of a complex between the enzyme and its substrate, leading to inhibition of HIV replication. This drug also inhibits ion channels, including calcium channels, potassium channels, sodium channels, and chloride channels. 1-Epi-darunavir has been shown to inhibit ligand binding to receptors in cell culture, such as peptides or antibodies.

Chemical properties

• Molecular weight: 547.7 g/mol
• Formula: C₂₇H₃₇N₃O₇S
• Purity: Min. 95%