Ritanserin

CAS: 87051-43-2

Ref. TM-T16759

Product Information

• Name: Ritanserin
• Synonyms: R 55667, 5H-Thiazolo(3,2-a)pyrimidin-5-one, 6-(2-(4-bis(4-fluorophenyl)methylene)-1-piperidinyl)ethyl)-7-methyl-, 6-(2-(4-(Bis(p-fluorophenyl)methylene)-piperidino)ethyl)-7-methyl-5H-thiazolo-(3,2-a)pyrimidin-5-one, 6-(2-{4-[bis(4-fluorophenyl)methylidene]piperidin-1-yl}ethyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one, 6-[2-[4-[Bis(4-fluorophenyl)methylene]-1-piperidinyl]ethyl]-7-methyl-5H-thiazolo[3,2-a]pyrimidin-5-one, R 55,667, Ritanserin [USAN:INN:BAN], Ritanserina, Ritanserina [Spanish], Ritanserine, Ritanserine [French], Ritanserinum, Ritanserinum [Latin], Tiserton, Unii-145Tfv465S, Zinc 00538314
• CAS: 87051-43-2

Description

Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.

• Brand: Targetmol

Chemical properties

• Molecular weight: 477.57
• Formula: C₂₇H₂₅F₂N₃OS
• Purity: 99.89%
• Color/Form: Solid
• InChI: InChI=1S/C27H25F2N3OS/c1-18-24(26(33)32-16-17-34-27(32)30-18)12-15-31-13-10-21(11-14-31)25(19-2-6-22(28)7-3-19)20-4-8-23(29)9-5-20/h2-9,16-17H,10-15H2,1H3
• InChI key: InChIKey=JUQLTPCYUFPYKE-UHFFFAOYSA-N
• SMILES: Cc1nc2sccn2c(=O)c1CCN1CCC(=C(c2ccc(F)cc2)c2ccc(F)cc2)CC1