Product Information
Name:HDGFRP2/PSIP1-IN-1
Synonyms:
- 4-(4-Bromo-1H-pyrazol-5-yl)pyridine
Brand:Targetmol
Description:Compound BPP (HDGFRP2/PSIP1-IN-1) is a dual inhibitor targeting the PWWP domains of Hepatoma-derived Growth Factor Related Protein 2 (HDGFRP2) and its homologue PSIP1. This compound effectively hinders the occurrence and progression of Diffuse Intrinsic Pontine Glioma (DIPG). It demonstrates binding affinity with a Kd value of 7 μM for HDGFRP2, indicative of its efficient ligand efficacy at 0.47. Additionally, Compound BPP exhibits a Kd value of 27 μM when binding to the PSIP1 PWWP domain, and a Kd value of 14 μM against HDGFRP3, confirming its potency as an inhibitor within the HDGFRP2 PWWP subfamily.
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Chemical properties
Molecular weight:224.06
Formula:C8H6BrN3
Color/Form:Solid
Technical inquiry about: HDGFRP2/PSIP1-IN-1
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