Keap1-IN-1
Ref. TM-T204622
Product Information
Name:Keap1-IN-1
Brand:Targetmol
Description:Keap1-IN-1 (Compound 27) is an inhibitor of Keap1, functioning by covalently modifying the Cys151 residue on the BTB domain of KEAP1, thereby disrupting the interaction between Keap and Nrf. It enhances the mRNA expression of the antioxidant response element (ARE) dependent gene NQO1, with an EC50 of 160 nM, and exhibits cytotoxicity in U2OS cells, with an EC50 of 527 nM.
Notice:Our products are intended for lab use only. For any other use, please contact us.
Chemical properties
Molecular weight:531.434
Formula:C17H21Cl2N2O5PS3
Color/Form:Solid
Technical inquiry about: Keap1-IN-1
Please use instead the cart to request a quotation or an order
If you want to request a quotation or place an order, please instead add the desired products to your cart and then request a quotation or order from the cart. It is faster, cheaper, and you will be able to benefit from the available discounts and other advantages.