Menin-KMT2A-IN-1
Ref. TM-T205488
Product Information
Name:Menin-KMT2A-IN-1
Brand:Targetmol
Description:Menin–KMT2A-IN-1 (Compound 20) is an inhibitor of menin–KMT2A, binding to menin with an IC50 of 8 nM, and disrupting the interaction between menin and lysine methyltransferase 2A (KMT2A). It inhibits hERG channels with an IC50 of 65 μM and suppresses MV4-11 cells with an IC50 of 74 nM. Furthermore, Menin–KMT2A-IN-1 exhibits favorable pharmacokinetic properties in CD-1 mice, with an oral bioavailability of 74%.
Notice:Our products are intended for lab use only. For any other use, please contact us.
Chemical properties
Molecular weight:522.61
Formula:C28H35FN6O3
Color/Form:Solid
Technical inquiry about: Menin-KMT2A-IN-1
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