LE135
CAS: 155877-83-1
Ref. TM-T22920
| 1mg | 46.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 133.00 € | ||
| 25mg | 213.00 € | ||
| 50mg | 318.00 € | ||
| 100mg | 462.00 € | ||
| 1ml*10 (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 21 May 2024
Product Information
Name:
LE135
Synonyms:
- LE 135
- Le 135
- 4-(7,8,9,10-Tetrahydro-5,7,7,10,10-pentamethyl-(5H)-benzo[e]naphtho[2.3-b][1.4]diazepine-13-yl)benzoicacid
- 4-(5,7,7,10,10-pentamethyl-7,8,9,10-tetrahydro-5H-benzo[e]naphtho[2,3-b][1,4]diazepin-13-yl)benzoic acid
CAS:
Description:
LE135 is a potent RAR antagonist that binds selectively to RARα (Ki of 1.4 μM) and RARβ (Ki of 220 nM), and has a higher affinity to RARβ. LE135 is highly selective over RARγ, RXRα, RXRβ and RXRγ. LE135 is also a potent TRPV1 and TRPA1 receptors activator with EC50s of 2.5 μM and 20 μM, respectively.
Brand:
Targetmol
Long term storage:
Notes:
Chemical properties
Molecular weight:
438.56
Formula:
C29H30N2O2
Purity:
98.33%
Color/Form:
Solid
MDL:
Melting point:
Boiling point:
Flash point:
Density:
Concentration:
EINECS:
Merck:
HS code:
Technical inquiry about: TM-T22920 LE135
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