DDR1-IN-5

CAS: 2416022-90-5

Ref. TM-T40062

Product Information

• Name: DDR1-IN-5
• Brand: Targetmol
• Description: DDR1-IN-5 is a potent and selective inhibitor of the Discoidin Domain Receptor family, member 1 (DDR1). It effectively inhibits the phosphorylation of DDR1b (Y513) with an IC 50 value of 4.1 nM. Furthermore, DDR1-IN-5 demonstrates remarkable anti-cancer activity. Its inhibitory potency against DDR1 (IC 50 = 7.36 nM) makes it a promising compound for targeted therapy in cancer treatment.

Chemical properties

• Molecular weight: 434.382
• Formula: C₂₂H₁₃F₃N₆O
• Color/Form: Solid