Bisnortilidine

CAS: 53948-51-9

Ref. TR-B508850

Product Information

• Name: Bisnortilidine
• Synonyms: (1R,2S)-rel-2-Amino-1-phenyl-3-cyclohexene-1-carboxylic Acid Ethyl Ester, trans-(+/-)-2-Amino-1-phenyl-3-cyclohexene-1-carboxylic Acid Ethyl Ester, 3-Cyclohexene-1-carboxylic acid, 2-amino-1-phenyl-, ethyl ester, (1R,2S)-rel-, 3-Cyclohexene-1-carboxylic acid, 2-amino-1-phenyl-, ethyl ester, trans-(+-)-

Description

Applications A metabolite of Tilidine (T440300(M)), which is a controlled substance (opiate) and a analgesic. Tilidine is used in clinical trial in comparison with Nefopam. Tilidine is one of the most widely used narcotics in Germany and Belgium.
References Hengy, H., et al.: J. Pharm. Sci., 67, 1765 (1978); Cordonnier, J., et al.: J. Anal. Toxicol., 11, 144 (1987); Hajda, J., et al.: J. Clin. Pharmacol., 42, 1257 (2002); Vollmer, K.-O., et al.: Arzneim.-Forsch., 20, 990 (1970); Abeloos, J., et al.: Acta Anaesthesiol. Belg., 34, 283 (1983); Van Cauwenberge, H., et al.: Int. J. Clin. Pharmacol. Res., 12, 1 (1992)

• Brand: TRC

Chemical properties

• Molecular weight: 245.32
• Formula: C₁₅H₁₉NO₂
• Color/Form: Light Yellow
• InChI: InChI=1S/C15H19NO2/c1-2-18-14(17)15(11-7-6-10-13(15)16)12-8-4-3-5-9-12/h3-6,8-10,13H,2,7,11,16H2,1H3/t13-,15+/m0/s1
• InChI key: InChIKey=BTKAMSWFNMGLGM-DZGCQCFKSA-N
• SMILES: CCOC(=O)[C@@]1(c2ccccc2)CCC=C[C@@H]1N