rac Bopindolol

CAS: 62658-63-3

Ref. TR-B675400

Product Information

• Name: rac Bopindolol
• Synonyms: 2-Propanol, 1-[(1,1-dimethylethyl)amino]-3-[(2-methyl-1H-indol-4-yl)oxy]-, 2-benzoate, 2-Propanol, 1-[(1,1-dimethylethyl)amino]-3-[(2-methyl-1H-indol-4-yl)oxy]-, benzoate (ester) (9CI), 2-Propanol, 1-[(1,1-dimethylethyl)amino]-3-[(2-methyl-1H-indol-4-yl)oxy]-, benzoate (ester), (±)-, (±)-Bopindolol, Bopindolol, (±)-1-(tert-Butylamino)-3-[(2-methylindol-4-yl)oxy]-2-propanol Benzoate (Ester), (±)1-[(1,1-Dimethylethyl)amino]-3-[(2-methyl-1H-indol-4-yl)oxy]-2-propanol Benzoate Ester, 1-(tert-Butylamino)-3-[(2-methyl-1H-indol-4-yl)oxy]propan-2-yl benzoate, 2-(tert-butylamino)-1-{[(2-methyl-1H-indol-4-yl)oxy]methyl}ethyl benzoate, 2-Propanol, 1-[(1,1-dimethylethyl)amino]-3-[(2-methyl-1H-indol-4-yl)oxy]-, 2-benzoate, 2-[(1,1-dimethylethyl)amino]-1-{[(2-methyl-1H-indol-4-yl)oxy]methyl}ethyl benzoate, 2-propanol, 1-[(1,1-dimethylethyl)amino]-3-[(2-methyl-1H-indol-4-yl)oxy]-, benzoate (ester), 82857-38-3, Sandonorm, Wandonorm

Description

Applications Bopindolol is an ester prodrug of Pindolol (P468000). Bopindolol is a long acting β-adrenoceptor blocking agent. Bopindolol displays antispasmogenic activity mediated by α1-adrenoceptors and 5-HT2 receptors.
References Turner, D.R. et al.: Br. J. Clin. Pharmacol., 17, 295 (1984); Brodde, O.E. et al.: J. Cardio. Pharmacol., 8, S70 91986); Doggrell, S.A.: Med, Sci. Res., 17, 681 (1989);

• Brand: TRC

Chemical properties

• Molecular weight: 380.48
• Formula: C₂₃H₂₈N₂O₃
• Color/Form: Neat
• InChI: InChI=1S/C23H28N2O3/c1-16-13-19-20(25-16)11-8-12-21(19)27-15-18(14-24-23(2,3)4)28-22(26)17-9-6-5-7-10-17/h5-13,18,24-25H,14-15H2,1-4H3
• InChI key: InChIKey=UUOJIACWOAYWEZ-UHFFFAOYSA-N
• SMILES: Cc1cc2c(OCC(CNC(C)(C)C)OC(=O)c3ccccc3)cccc2[nH]1