Product Information
Name:trans-Loperamide N-Oxide
Controlled Product
Synonyms:
- Arestal
- Loperamide oxide
- R 58425,Loperamide Oxide
- Loperamide Hydrochloride Imp. F (EP)
- trans-4-(4-chlorophenyl)-4-hydroxy-N,N-dimethyl-α,α-diphenyl-1-piperidinebutanamide 1-oxide
Brand:TRC
Description:Stability HygroscopicApplications Loperamide oxide (LOPOX) is a prodrug of Loperamide (LOP). It is concluded that Loperamide oxide administered intraluminally is reduced to Loperamide and has the same antisecretory potency as Loperamide in jejunum and colon. Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the packageReferences Lavrijsen, K., et al.: Drug Metab. Dispos., 23, 354 (1995), Hesselink, D., et al.: Clin. Pharmacol. Ther., 74, 245 (2003), Hooijberg, J., et al.: Biochem. Pharmacol., 67, 1541 (2004),
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Chemical properties
Molecular weight:493.04
Formula:C29H33ClN2O3
Color/Form:Off-White
InChI:InChI=1S/C29H33ClN2O3/c1-31(2)27(33)29(24-9-5-3-6-10-24,25-11-7-4-8-12-25)19-22-32(35)20-17-28(34,18-21-32)23-13-15-26(30)16-14-23/h3-16,34H,17-22H2,1-2H3/t28-,32-
InChI key:InChIKey=KXVSBTJVTUVNPM-UHFFFAOYSA-N
SMILES:CN(C)C(=O)C(CC[N+]1([O-])CCC(O)(c2ccc(Cl)cc2)CC1)(c1ccccc1)c1ccccc1
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