Enzimas Inibidoras
Inibidores enzimáticos são compostos que diminuem ou interrompem a atividade das enzimas, ligando-se a elas de forma específica. Esses inibidores desempenham um papel crucial na regulação dos processos biológicos e são amplamente utilizados na pesquisa médica e no desenvolvimento de medicamentos. Ao bloquear a ação das enzimas, permitem o estudo da função enzimática e o desenvolvimento de tratamentos para diversas doenças. Na CymitQuimica, oferecemos uma ampla gama de inibidores enzimáticos de alta qualidade para apoiar suas pesquisas em biologia e farmacologia.
Foram encontrados 123 produtos de "Enzimas Inibidoras"
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Nafamostat
CAS:Fórmula:C19H17N5O2Pureza:≥ 98.0%Cor e Forma:White to off-white powderPeso molecular:347.37Vildagliptin
CAS:Fórmula:C17H25N3O2Pureza:≥ 98.0%Cor e Forma:White to off-white powderPeso molecular:303.40IU1
CAS:Fórmula:C18H21FN2OPureza:(TLC) ≥ 98%Cor e Forma:Off-white to pale brown solidPeso molecular:300.37Fumagillin
CAS:Fórmula:C26H34O7Pureza:≥ 95.0%Cor e Forma:White, off-white or pale yellow to tan powderPeso molecular:458.54Lactacystin
CAS:Fórmula:C15H24N2O7SPureza:≥ 95.0%Cor e Forma:White solid or powderPeso molecular:376.43Nα-Tosyl-L-lysine chloromethyl ketone hydrochloride
CAS:Fórmula:C14H21ClN2O3S·HClPureza:(HPLC) ≥ 98.0%Cor e Forma:White powderPeso molecular:369.31Bortezomib
CAS:Fórmula:C19H25BN4O4Pureza:≥ 98.0%Cor e Forma:White to off-white powder or solidPeso molecular:384.24E-64 protease inhibitor
CAS:Fórmula:C15H27N5O5Pureza:(HPLC) ≥ 98.0%Cor e Forma:White crystalline powderPeso molecular:357.40Bestatin hydrochloride
CAS:Fórmula:C16H24N2O4·HClPureza:≥ 98.0% (dried basis)Cor e Forma:White to almost white powderPeso molecular:344.87Argatroban
CAS:Fórmula:C23H38N6O6SPureza:(HPLC) ≥ 98%Cor e Forma:White to off-white powderPeso molecular:526.65AEBSF hydrochloride
CAS:Fórmula:C8H10FNO2S·HClPureza:≥ 98.0%Cor e Forma:White to off-white powder or solidPeso molecular:239.69N-p-Tosyl-L-phenylalanine chloromethyl ketone
CAS:Fórmula:C17H18ClNO3SPureza:(TLC) ≥ 98.0%Cor e Forma:White to off-white powderPeso molecular:351.85Z-VAD-FMK, cell permeable
CAS:Fórmula:C22H30FN3O7Pureza:≥ 95.0%Cor e Forma:White to off-white solidPeso molecular:467.5Elastatinal microbial
CAS:Fórmula:C21H36N8O7Pureza:~0.64μg/ml (IC50, pH8.8, 37°C)Cor e Forma:White to light-yellow or tan powderPeso molecular:512.60Pepstatin A
CAS:Fórmula:C34H63N5O9Pureza:≥ 98.0%Cor e Forma:White to off-white powderPeso molecular:685.90Suramin sodium salt
CAS:Fórmula:C51H34N6Na6O23S6Pureza:≥ 98%Cor e Forma:White to off-white powderPeso molecular:1429.16E-64d protease inhibitor
CAS:Fórmula:C17H30N2O5Pureza:≥ 95.0%Cor e Forma:White powderPeso molecular:342.43Carfilzomib
CAS:Fórmula:C40H57N5O7Pureza:(HPLC) ≥ 98.0%Cor e Forma:White to off-white crystalline powder or crystalsPeso molecular:719.91Phosphoramidon disodium salt
CAS:Fórmula:C23H32N3Na2O10PPureza:≥ 97.0%Cor e Forma:Colourless, transparent crystals or white to light yellow crystalline powderPeso molecular:587.47Nafamostat mesylate
CAS:Fórmula:C19H17N5O2Pureza:≥ 99.0%Cor e Forma:White to off-white or beige crystalline powderPeso molecular:347.37DAPT
CAS:Fórmula:C23H26F2N2O4Pureza:(NMR) ≥ 98.0%Cor e Forma:White to off-white solidPeso molecular:432.50Leupeptin hemisulfate
CAS:Fórmula:C20H38N6O4·5H2SO4Pureza:≥ 95%Cor e Forma:White to off-white powderPeso molecular:475.59Z-Leu-Leu-Leu-al
CAS:Fórmula:C26H41N3O5Pureza:≥ 97.0%Cor e Forma:White to off-white powder or solidPeso molecular:475.63CP-10447
CAS:<p>Applications CP-10447 is an inhibitor apolipoprotein B (apoB) and triglyceride secretion in human hepatoma cells (HepG2) by inhibiting MTP activity and stimulating the early ER degradation of apoB. It is useful tool for further study of the mechanisms of apoB secretion and triglyceride-rich lipoprotein assembly.<br>References Haghpassand, M. et al.: J. Lipid. Res., 37, 1468 (1996); Pan, M. et al.: J. Biol. chem., 275, 27399 (2000);<br></p>Fórmula:C16H13BrN2OCor e Forma:NeatPeso molecular:329.192-(Hydroxyamino)acetic Acid
CAS:Produto Controlado<p>Applications 2-(Hydroxyamino)acetic Acid is a novel lactase inhibitor.<br>References Hattori, M., et al.: J. Insect Physiol., 51, 1359 (2005); Murao, S., et al.: Biosci. Biotech. Biochem., 56, 987 (1992)<br></p>Fórmula:C2H5NO3Cor e Forma:NeatPeso molecular:91.07(3S,4S,3’S)-Ezetimibe
CAS:<p>Applications (3S,4S,3’S)-Ezetimbe is a 3-epimer impurity of Ezetimibe (E975000), a cholesterol absorption inhibitor.<br>References van Heek, M., at al.: J. Pharmacol. Exp. Ther., 283, 157 (1997), van Heek, M., at al.: Brit. J. Pharmacol., 129, 1748 (2000)<br></p>Fórmula:C24H21F2NO3Cor e Forma:Off-WhitePeso molecular:409.43LCZ696
CAS:<p>Applications LCZ696 is a novel dual-acting inhibitor of angiotensin II receptor and neprilysin, which can be used for blood pressure reduction.<br>References Ruilope, L.M.; et al.: Lancet, 375, 1255 (2010)<br></p>Fórmula:C24H28NO5·C24H27N5O3·3Na·x(H2O)Cor e Forma:MixturePeso molecular:479.48 + (433.47) + x(18.02)Abamine
CAS:Produto Controlado<p>Applications Abamine is an inhibitor of 9-Cis-Epoxycarotenoid dioxygenase (NCED), the key regulatory enzyme in the plant hormone abscisic acid (ABA) biosynthesis pathway.<br>References Kitahata, N., et al.: Bioorg. Med. Chem., 14, 5555 (2006); Han, S., et al.: Bioorg. Med. Chem. Lett., 14, 3033 (2004)<br></p>Fórmula:C21H24FNO4Cor e Forma:NeatPeso molecular:373.423'-Deoxyadenosine 5’-Diphosphate Triethylamine Salt (>90%)
CAS:<p>Stability Hygroscopic<br>Applications 3'-Deoxyadenosine 5’-Diphosphate Triethylamine Salt, is a nucleotide and was proposed to be a possible inhibitor of DNA synthesis.<br>References Frederiksen, Sune.: Biochimica et Biophysica Acta, 76(3), 366-71 (1963)<br></p>Fórmula:C10H15N5O9P2•xC6H15NPureza:>90%Cor e Forma:NeatPeso molecular:411.20 + x(101.19)Teneligliptin Hydrobromide (2:5)
CAS:Produto Controlado<p>Applications Teneligliptin Hydrobromide (2:5) is a dipeptidyl peptidase-4 (DPP-4) inhibitor that is used to treat type 2 diabetes. It is eliminated via excretion, and has a half-life of 24.2 hours in the human body.<br>References Goda, M. & Kadowaki, T.: Drugs Today, 49, 615 (2013); Kishimoto, M.: Diabetes Metab. Syndr. Obes., 6, 187 (2012)<br></p>Fórmula:C22H32·5Br2·5N6OSCor e Forma:NeatPeso molecular:628.86Daidzein Diglucuronide
CAS:Produto ControladoFórmula:C27H26O16Cor e Forma:White To Off-WhitePeso molecular:606.49(3S,5S)-Atorvastatin Calcium Salt
CAS:Produto Controlado<p>Impurity Atorvastatin Related Compound E<br>Applications Impuritiy of Atorvaststin (A791750), a selective, competitive HMG-CoA reductase inhibitor. Atorvastatin is the only drug in its class specfically indicated for lowering both elevated LDL-cholesterol and triglycerides in patients with hypercholesterolemia. Atorvastatin Related Compound E<br>References Kearney, A.S., et al.: Pharm. Res., 10, 1461 (1993), Heinonen, T.M., et al.: Clin. Ther., 18, 853 (1996), Whitfield, L.R., et al.: Eur. J. Drug Metab. Pharmacokinet., 25, 97 (2000),<br></p>Fórmula:C33H34FN2O5·CaCor e Forma:NeatPeso molecular:1155.34N-(2-Hydroxyethyl)-1-deoxy-L-idonojirimycin Hydrochloride
CAS:Produto Controlado<p>Stability Hygroscopic<br>Applications α-Glycosidase inhibitor.<br>References van de Water, F., et al.: Drug Metab. Rev., 37, 443 (2005), Koepsell, H., et al.: Pharm. Res., 24, 1227 (2007), Jappar, D., et al.: Pharm. Res., 26, 172 (2009),<br></p>Fórmula:C8H18ClNO5Cor e Forma:NeatPeso molecular:243.69N-(2-Hydroxyethyl)-1-deoxy-L-altronojirimycin Hydrochloride Salt
CAS:Produto Controlado<p>Stability Hygroscopic<br>Applications α-Glycosidase inhibitor.<br>References Jefferies, I., et al.: Bioorg. Med. Chem. Lett., 7, 1171 (1997), Hassan, A., et al.: Carbohydr. Res., 339, 1565 (2004),<br></p>Fórmula:C8H18ClNO5Cor e Forma:NeatPeso molecular:243.6852Aprotinin Hydrochloride
CAS:<p>Applications Aprotinin is used in cardiac surgery to minimize bleeding and reduce exposure to blood products.<br>References Mangano, D. et al.: New Eng. J. Med., 354, 353 (2006); Fergusson, D. et al.: New. Eng. J. Med., 358, 2319 (2008);<br></p>Fórmula:C284H432N84O79S7·x(ClH)Cor e Forma:White SolidPeso molecular:6511.51(free amine)Nitromifene Citrate (E/Z mixture)
CAS:Produto Controlado<p>Applications Nitromifene citrate is a non-steroidal estrogen antagonist. It is structurally similar to Tamoxifen (T006000) which is a selective estrogen response modifier (SERM).<br>References Rudick, C., et al.: Endorcrinol., 144, 179 (2003); Sutherland, R., et al.: Nature, 267, 434 (1977)<br></p>Fórmula:C33H36N2O11Cor e Forma:Yellow To OrangePeso molecular:636.65Galacto-PUGNAc (>90%)
CAS:Produto Controlado<p>Stability Moisture and Temperature Sensitive<br>Applications Galacto-PUGNAc is a highly selective inhibitor for β-hexosaminidases HEXA and HEXB is cell-permeable. Galacto-PUGNAc is able to modulate the activity of HEXA and HEXB in tissue culture, increasing ganglioside GM2 levels in neuroblastoma cells<br>References Stubbs, K.A. et al.: Angew. Chem. Int. Ed., 48, 1300 (2009);<br></p>Fórmula:C15H19N3O7Pureza:>90%Cor e Forma:NeatPeso molecular:353.332,5-Dideoxy-2,5-imino-D-mannitol
CAS:Produto Controlado<p>Stability Hygroscopic<br>Applications A glucosidase inhibitor.<br>References Fellows, L.E.: Pestic. Sci., 17, 602 (1986)<br></p>Fórmula:C6H13NO4Cor e Forma:Off White SolidPeso molecular:163.17Vitamin B12 e-Monocarboxylic Acid
CAS:<p>Stability Hygroscopic<br>Applications Vitamin B12 Monocarboxylic Acid is an impurity of Vitamin B12 (V676005) which is a water-soluble vitamin with a key role in the normal functioning of the brain and nervous system, and for the formation of blood.<br>References Rickes, et al.: Science, 107, 396 (1948); Kirschbaum, J., et al.: Anal. Profiles Drug Subs., 10, 183 (1981); Grasbeck, R., et al.: Clin. Biochem., 17, 99 (1984)<br></p>Fórmula:C63H87CoN13O15PCor e Forma:Dark Red SolidPeso molecular:1356.35tert-Butyl (2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]-2-[(1,3-thiazolidin-3-yl)carbonyl]pyrrolidine-1-carboxylate
CAS:Produto Controlado<p>Applications tert-Butyl (2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]-2-[(1,3-thiazolidin-3-yl)carbonyl]pyrrolidine-1-carboxylate is an orally anti-diabetic agent as a inhibitors of dipeptidylpeptidase IV (DPP-4).<br>References Yoshida, T., et al.: Bioorg. Med. Chem., 20, 5705-5719 (2012);<br></p>Fórmula:C27H38N6O3SCor e Forma:NeatPeso molecular:526.69
![tert-Butyl (2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]-2-[(1,3-thiazolidin-3-y…](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTR%2Fthumb-webp%2FB807705.webp&w=3840&q=75)