Derivados de Aminoácidos

Z-LLY-a-keto aldehyde (peptidyl glyoxal), previously shown to be an excellent inhibitor of the serine and …

Leu-OMe (LME) causes lysosomal disruption and death of human monocytes (M phi). In addition, LME …

Muramyl dipeptide (MDP) inhibits HIV replication in CD4+ H9 lymphocytes..

pTH (1-31) amide appears so far to be the smallest of the potently osteogenic pTH …

a-Melanotropin, also known as a-melanocyte-stimulating hormone (a-MSH), is a 13-amino acid peptide originally characterized as …

The major regulator of adrenal cortex function. ACTH stimulates the synthesis of steroidal hormones.

Bachem ID: 4101678.

The presence of halogen substituents at the fluorescent group improves membrane permeability of the YVAD-derived …

The prolyl oligopeptidase (POP) substrate Z-AP-pNA was used in combination with Z-GP-pNA and Z-AA-pNA for …

Exendin (9-39) is a potent glucagon-like peptide 1 (GLP-1) receptor antagonist. It has also been …

CALP-3, VKFGVGFK, acts as a calmodulin agonist. The octapeptide interacts with the calmodulin EF-hand motif, …

o-Conotoxin MVIIA, originally isolated from the venom of the fish-hunting cone snail Conus magus, is …

Caloxin 2A1 is a selective extracellular inhibitor of the plasma membrane Ca2+-pump.

a-Methyl-proline restores normal levels of bone collagen type I synthesis in ovariectomized rats, used as …

Short-term administration of deslorelin stimulates the formation of LH and FSH, which induce an increase …

Fragment of human leptin, an adipose tissue-derived protein encoded by the obese gene. Leptin has …

Substrate for leucine aminopeptidase.

This NPY analog is a highly potent and selective ligand for Y1 receptors in different …

Specific Y1 receptor agonist.

The sequence RRPYIL is essential for neurotensin-NT receptor interaction.

AFP-pNA, substrate for prolyl tripeptidyl aminopeptidases from the periodontal pathogens Porphyromonas gingivalis and Prevotella nigrescens.

N-terminal sequence of dynorphin A and the neoendorphins.

Substrate for dipeptidyl aminopeptidase I (cathepsin C).

Apelin-17 is an endogenous ligand of the human orphan G protein-coupled receptor APJ, reported to …

Former CAS-number 26469-81-8.

Bachem ID: 4089772.

Nafarelin is a synthetic decapeptide agonist of the luteinizing hormone-releasing hormone (LHRH) which is approximately …

a-Conotoxin MI has been isolated from the venom of the sea snail Conus imperialis. The …

Bachem ID: 4097932.

VSV-8, RGYVYQGL, corresponds to positions 52 to 59 of vesicular stomatitis virus (VSV) nucleoprotein which …

Fluorophore-labeled phalloidin used for visualizing the actin cytoskeleton.

Potential impurity of exenatide.

Substrate for human plasma carboxypeptidase N and membrane-bound carboxypeptidase D.

This biotinylated LHRH derivative has been used in a functional analysis of the LHRH receptor …

Main degradation product of NPY in serum and Y2/Y5 receptor agonist.

In contrast to the encephalitogenic rat homolog, myelin oligodendrocyte glycoprotein (35-55) (human) does not appear …

pTHrP (7-34) amide is a potent antagonist of the effects of pTH-related protein (1-34) in …

In vitro, this compound competitively inhibited sweetalmond b-glucosidase (Ki = 17 uM).

Suc-AAPL-pNA, a sensitive substrate for human and especially porcine pancreatic elastases. Substrate for leucine endopeptidase …

Suc-YVAD-pNA, a chromogenic caspase-1 substrate.

GLP-2 administration to mice or rats promotes stimulation of crypt cell proliferation and inhibition of …

Bachem ID: 4011662.

Tetraproline. PPPP was used as an internal standard in the quantitative determination of the antihypertensive …

Iberiotoxin (IbTx), from the venom of the scorpion Buthus tamulus, shows 68% sequence homology with …

Bachem ID: 4031199.

u-Conotoxin GIIIA from the Conus geographus L. venom blocks with very high selectivity the muscle …

Thymopentin (TP5), an active fragment of thymopoietin (TP), reduces endocrine and behavioral responses to experimental …

This GIP fragment has potent insulinotropic activity in the isolated, perfused rat pancreas but greatly …

Bachem ID: 4044101.

Sensitive fluorogenic substrate for dipeptidyl aminopeptidase I (DPP I, cathepsin C).

Tertiapin (TPN), a potent inhibitor of the inward-rectifier K+ channels, blocked a G-protein-gated channel (GIRK1/4) …

The pentapeptide TRSAW, a highly conserved sequence within the pTH-related protein, is a potent inhibitor …

Deltorphin B, a selective d-opioid receptor agonist isolated from the skin of Phyllomedusa bicolor.

A ghrelin receptor antagonist. Asakawa et al. found that peripherally administered (D-Lys3)-GHRP-6 (HwkWfK-amide) decreased food …

Substrate for aminopeptidase B (arginine aminopeptidase) and cathepsin H.

Bachem ID: 4001907.

NLS, cell-penetrating peptide containing 7 amino acids homologous to the SV40 T antigen, was capable …

The lipopeptide FSL-1, synthesized on the basis of the N-terminal structure of a M. salivarium …

Z-VEID-AFC, fluorogenic substrate for caspase-6 (Mch2).

Bachem ID: 4096177.

Bachem ID: 4012218.

Bachem ID: 4015469.

Bachem ID: 4014443.

CCK-8 exhibits various gastrointestinal effects as contraction of the gallbladder and stimulation of pancreatic secretion …

Bachem ID: 4012160.

Calcitonin is a peptide hormone involved in calcium and phosphorus homeostasis. Its inhibitory effect on …

Bachem ID: 4096190.

A good substrate for carboxypeptidase Y. Educt for the synthesis of fluorinated a-keto carboxylic inhibitors …

GRF antagonist.

KALA amphipathic peptide, a low-molecular weight cationic amphipathic peptide was able to bind to DNA, …

Degradation product of oxytocin.

GLP-1 (7-36) amide is secreted from the lower small intestine and shows a strong insulinotropic …

Potential degradation product of exenatide resulting from aspartimide formation and cleavage.

Fmoc-D-AzF can be incorporated in peptides as precursor of p-aminophenylalanine. Levinson et al. reduced the …