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Caspase

Caspase

Os inibidores de caspases são compostos que bloqueiam a atividade das caspases, uma família de proteases que são executores centrais da apoptose. As caspases clivam substratos específicos dentro da célula para desencadear o processo apoptótico, levando à morte celular programada. Os inibidores de caspases são usados para estudar os mecanismos da apoptose, bem como para prevenir a morte celular indesejada em vários modelos de pesquisa. Esses inibidores também são explorados em contextos terapêuticos para proteger as células da apoptose em doenças como a neurodegeneração. Na CymitQuimica, oferecemos uma ampla gama de inibidores de caspases de alta qualidade para apoiar sua pesquisa em apoptose, morte celular e áreas relacionadas.

Foram encontrados 144 produtos de "Caspase"

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produtos por página.
  • Crustecdysone

    CAS:
    <p>Crustecdysone (Hydroxyecdysone) is a steroid hormone that regulates the processes of molting or ecdysis in insects.</p>
    Fórmula:C27H44O7
    Pureza:99.06% - 99.67%
    Cor e Forma:Canary Yellow Fine Powder
    Peso molecular:480.63

    Ref: TM-T2881

    5mg
    38,00€
    10mg
    50,00€
    25mg
    73,00€
    50mg
    94,00€
    100mg
    136,00€
    500mg
    323,00€
  • ML-9

    CAS:
    ML-9 suppresses MLCK, PKA, and PKC activity with Ki values of 4, 32, and 54 μM, respectively.
    Fórmula:C15H18Cl2N2O2S
    Pureza:99.69%
    Cor e Forma:Crystalline Solid
    Peso molecular:361.29

    Ref: TM-T16104

    5mg
    40,00€
    10mg
    57,00€
    25mg
    96,00€
    50mg
    140,00€
    100mg
    202,00€
    200mg
    330,00€
    1mL*10mM (DMSO)
    44,00€
  • Diclofenac diethylamine

    CAS:
    Diclofenac Diethylamine, a non-selective COX inhibitor, is utilized as a nonsteroidal anti-inflammatory drug (NSAID).
    Fórmula:C18H22Cl2N2O2
    Pureza:99.81% - 99.87%
    Cor e Forma:Solid
    Peso molecular:369.29

    Ref: TM-T0432

    50mg
    34,00€
    1mL*10mM (DMSO)
    55,00€
  • Q-VD-OPH

    CAS:
    Q-VD-OPh is an irreversible caspase inhibitor with an IC50 value of 48 nM against caspase-7 and between 25 and 400 nM against caspase-1, 3, 8, 9, 10, 12.
    Fórmula:C26H25F2N3O6
    Pureza:97.8% - 98.95%
    Cor e Forma:Solid
    Peso molecular:513.5

    Ref: TM-T0282

    1mg
    51,00€
    5mg
    95,00€
    10mg
    144,00€
    25mg
    225,00€
    50mg
    349,00€
    100mg
    520,00€
    1mL*10mM (DMSO)
    97,00€
  • Fenbufen

    CAS:
    Fenbufen (Lederfen) is a non-steroidal anti-inflammatory drug used primarily to treat inflammation in osteoarthritis, ankylosing spondylitis, and tendinitis.
    Fórmula:C16H14O3
    Pureza:98.35% - 98.46%
    Cor e Forma:White Solid
    Peso molecular:254.28

    Ref: TM-T0859

    1g
    57,00€
    200mg
    35,00€
    500mg
    48,00€
  • Oxidopamine hydrobromide

    CAS:
    Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.
    Fórmula:C8H12BrNO3
    Pureza:98.22% - 99.88%
    Cor e Forma:Beige To Brown Fine Crystalline Powder
    Peso molecular:250.09

    Ref: TM-T12352L

    50mg
    35,00€
    100mg
    52,00€
    500mg
    157,00€
  • Ac-FLTD-CMK

    CAS:
    <p>Ac-FLTD-CMK, an abscisicin D derivative, selectively inhibits inflammatory caspases-1, -4, and -11 (IC50: 46.7 nM, 1.49 μM, 329 nM) but not caspase-3.</p>
    Fórmula:C26H37ClN4O8
    Pureza:95.17%
    Cor e Forma:Solid
    Peso molecular:569.05

    Ref: TM-T36819

    1mg
    283,00€
    5mg
    692,00€
    10mg
    938,00€
    25mg
    1.454,00€
    50mg
    1.882,00€
    100mg
    2.642,00€
  • Ac-YVAD-CMK

    CAS:
    <p>Ac-YVAD-CMK: Irreversible Caspase-1 inhibitor; halts pyroptosis, IL-1β/IL-18; neuroprotective and anti-inflammatory.</p>
    Fórmula:C24H33ClN4O8
    Pureza:97.08% - 99.909%
    Cor e Forma:Solid
    Peso molecular:540.99

    Ref: TM-T36347

    1mg
    70,00€
    5mg
    216,00€
    10mg
    354,00€
    25mg
    582,00€
    50mg
    825,00€
  • Lacidipine

    CAS:
    Lacidipine (SN-305) is a slow-acting, long-duration lipophilic dihydropyridine calcium blocker that prevents reflex tachycardia and lowers blood pressure.
    Fórmula:C26H33NO6
    Pureza:99.98%
    Cor e Forma:White-To-Off-White Crystalline Solid
    Peso molecular:455.54

    Ref: TM-T1439

    25mg
    39,00€
    50mg
    59,00€
    100mg
    96,00€
    500mg
    234,00€
    1mL*10mM (DMSO)
    34,00€
  • Inclisiran sodium

    CAS:
    Inclisiran (ALN-PCSsc) possesses antihypertensive activity, inhibiting the transcription of PCSK9, and can be used to research cardiovascular diseases.
    Pureza:99.29%
    Cor e Forma:Odour Solid

    Ref: TM-T39122

    1mg
    306,00€
    5mg
    792,00€
    10mg
    1.094,00€
    25mg
    1.610,00€
    50mg
    2.127,00€
    100mg
    2.872,00€
  • Aspirin

    CAS:
    Aspirin (Acetylsalicylic Acid) is a COX inhibitor. Aspirin has anti-inflammatory, antipyretic and analgesic activities. Cost-effective and quality-assured.
    Fórmula:C9H8O4
    Pureza:99.78% - 99.91%
    Cor e Forma:White Solid Crystalline
    Peso molecular:180.16

    Ref: TM-T0005

    1g
    58,00€
    5g
    95,00€
    200mg
    37,00€
    500mg
    50,00€
    1mL*10mM (DMSO)
    55,00€
  • Diclofenac sodium

    CAS:
    <p>Diclofenac sodium (GP 45840) is a non-steroidal anti-inflammatory agent (NSAID) with antipyretic and analgesic actions.</p>
    Fórmula:C14H10Cl2NNaO2
    Pureza:98.21% - 99.73%
    Cor e Forma:White Or Off-White Powder
    Peso molecular:318.13

    Ref: TM-T1555

    500mg
    49,00€
  • Diclofenac

    CAS:
    Diclofenac: a nonsteroidal compound inhibiting COX-1 and COX-2, reducing pro-inflammatory prostaglandins.
    Fórmula:C14H11Cl2NO2
    Pureza:99.69% - 99.97%
    Cor e Forma:Crystals From Ether-Petroleum Ether Solid
    Peso molecular:296.15

    Ref: TM-T0196

    5g
    56,00€
    10g
    90,00€
    500mg
    49,00€
    1mL*10mM (DMSO)
    50,00€
  • Dehydrocorydaline chloride

    CAS:
    Dehydrocorydaline chloride (13-Methylpalmatine chloride) is an alkaloid with anti-inflammatory and anti-cancer activity. Can improve the activation of p38 MAPK.
    Fórmula:C22H24ClNO4
    Pureza:99.53%
    Cor e Forma:Solid
    Peso molecular:401.88

    Ref: TM-T10990

    1mg
    58,00€
    5mg
    111,00€
    10mg
    160,00€
    25mg
    264,00€
    50mg
    396,00€
    100mg
    563,00€
    1mL*10mM (DMSO)
    124,00€
  • Terfenadine

    CAS:
    Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.
    Fórmula:C32H41NO2
    Pureza:98.76% - 99.75%
    Cor e Forma:Solid
    Peso molecular:471.67

    Ref: TM-T1266

    50mg
    43,00€
    100mg
    55,00€
    200mg
    82,00€
    1mL*10mM (DMSO)
    55,00€
  • Oxidopamine hydrochloride

    CAS:
    Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride) is an neurotransmitter dopamine antagonist.
    Fórmula:C8H12ClNO3
    Pureza:98.34% - 99.85%
    Cor e Forma:Physical Description Beige Solid (Ntp 1992)
    Peso molecular:205.64

    Ref: TM-T12352

    5mg
    47,00€
    10mg
    65,00€
    25mg
    103,00€
    50mg
    170,00€
    100mg
    259,00€
  • Thiabendazole

    CAS:
    Thiabendazole (2-(4-Thiazolyl)benzimidazole) is a benzimidazole derivative with anthelminthic property.
    Fórmula:C10H7N3S
    Pureza:99.14%
    Cor e Forma:Light Yellow Powder
    Peso molecular:201.25

    Ref: TM-T0938

    1g
    34,00€
    5g
    48,00€
    1mL*10mM (DMSO)
    34,00€
  • Ac-Trp-Glu-His-Asp-Aldehyde

    CAS:
    Ac-Trp-Glu-His-Asp-Aldehyde is a powerful and selective inhibitor of caspase-1, demonstrating a K_i value of 56 pM [1] [2].
    Fórmula:C28H33N7O9
    Cor e Forma:Solid
    Peso molecular:611.6

    Ref: TM-T76600

    5mg
    A consultar
    50mg
    A consultar
  • TNF-α-IN-11


    TNF-α-IN-11 (Compound 10) is a TNF-α inhibitor exhibiting a dissociation constant (K D) of 12.06 μM.
    Fórmula:C24H26N2O5
    Cor e Forma:Solid
    Peso molecular:422.47

    Ref: TM-T78730

    5mg
    A consultar
    50mg
    A consultar
  • IRF1-IN-2

    CAS:
    IRF1-IN-2 is a small molecule IRF1 inhibitor that suppresses pyroptosis, protecting against radiation-induced skin damage.
    Fórmula:C18H20N2O4S
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:360.43

    Ref: TM-T203076

    25mg
    43,00€
    50mg
    60,00€
    100mg
    88,00€
    1mL*10mM (DMSO)
    34,00€