Endocrinologia/Hormónios
Os inibidores de endocrinologia/hormônios são compostos que bloqueiam a ação dos hormônios ou interferem nas vias de sinalização hormonal. Esses inibidores são essenciais para estudar a regulação dos sistemas endócrinos e para desenvolver tratamentos para doenças relacionadas aos hormônios, como diabetes, distúrbios da tireoide e cânceres dependentes de hormônios. Ao modular a atividade hormonal, esses inibidores podem ajudar a elucidar as complexas interações dentro do sistema endócrino. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para endocrinologia/hormônios para apoiar sua pesquisa em endocrinologia, farmacologia e ciências médicas.
Subcategorias de "Endocrinologia/Hormónios"
- Receptor de Androgénio(229 produtos)
- Anexina A(16 produtos)
- Aromatase(22 produtos)
- Receptor de estrogénio/progestagénio(64 produtos)
- GPR(1 produtos)
- Receptor de glicocorticoides(165 produtos)
- LHRH(2 produtos)
- Receptor opioide(325 produtos)
- Receptor de Prostaglandina(122 produtos)
- RAAS(86 produtos)
- Redutase(51 produtos)
- Somatostatina(57 produtos)
- Receptor de hormónio tireoidiano (THR)(33 produtos)
- Receptor de Vasopressina(48 produtos)
Exibir 6 mais subcategorias
Foram encontrados 3369 produtos de "Endocrinologia/Hormónios"
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22-Hydroxy mifepristone
CAS:22-Hydroxy Mifepristone (RU 42698) is an orally active hydroxylated alcohol metabolite that exhibits both anti-progestational and anti-glucocorticoid activities. This compound contains an alkyne group and is capable of undergoing copper-catalyzed azide-alkyne cycloaddition (CuAAC) with azide-containing molecules. Furthermore, 22-Hydroxy Mifepristone demonstrates a relative binding affinity of 48% to the human glucocorticoid receptor.Fórmula:C29H35NO3Cor e Forma:SolidPeso molecular:445.59THR-β agonist 4
CAS:THR-β agonist 4 is a potent agonist of THR-β.Fórmula:C16H11Cl2F2N5O6SCor e Forma:SolidPeso molecular:510.26LXT34
CAS:LXT34 (Example 2) is a GPR120 agonist with anti-inflammatory properties. This compound enhances GLP-1 formation in the gastrointestinal tract and improves insulin resistance in macrophages and pancreatic cells. LXT34 is applicable in studies related to inflammatory conditions, such as type 2 diabetes, obesity, and non-alcoholic fatty liver disease.Fórmula:C18H21NO3SCor e Forma:SolidPeso molecular:331.43Phenethyl 4-ANPP
CAS:Phenethyl 4-ANPP is a MOR (μ-opioid receptor) agonist with a structure similar to known opioids.Fórmula:C27H32N2Cor e Forma:SolidPeso molecular:384.56Novokinin
CAS:Angiotensin AT2 receptor agonistFórmula:C39H61N11O7Pureza:98%Cor e Forma:SolidPeso molecular:795.97ErSO-DFP
ErSO-DFP activates a-UPR, targets ERα+ cancer cells with high selectivity, and effectively reduces MCF-7 tumours.Fórmula:C20H17F5N2O2Cor e Forma:SolidPeso molecular:412.355′-Guanidinonaltrindole
CAS:5′-Guanidinonaltrindole (GNTI) is a selective antagonist of the kappa opioid receptor.Fórmula:C27H29N5O3Cor e Forma:SolidPeso molecular:471.551BMS-248360
CAS:BMS-248360: Oral dual hAT1/hETA antagonist with Kis of 10nM & 1.9nM, respectively; treats hypertension.Fórmula:C36H45N5O5SPureza:98%Cor e Forma:SolidPeso molecular:659.84GDC-0927 Racemate
CAS:GDC-0927 Racemate is a degrader of estrogen receptor, is used in the research of ER-related diseases, potently inhibits ER-α activity, with an IC50 of 0.2 nM.Fórmula:C28H28FNO4Pureza:98%Cor e Forma:SolidPeso molecular:461.52BNTX
CAS:BNTX (7-Benzylidenenaltrexone) is a selective δ1-opioid receptor antagonist. It competitively counteracts the antisecretory effects of DPDPE, Deltorphin 2, and DAMGO. BNTX is applicable in research focused on antinociceptive effects.Fórmula:C27H27NO4Cor e Forma:SolidPeso molecular:429.508AKR1C3-IN-7
AKR1C3-IN-7 (Compound 13) is an effective and selective AKR1C3 inhibitor (IC50=0.19 μM). AKR1C3-IN-7 has antitumor activity.Fórmula:C24H20N2O4Cor e Forma:SolidPeso molecular:400.43AR ligand-44
CAS:AR ligand-44 is an androgen receptor (androgen receptor) ligand that can be utilized in the synthesis of PROTACs such as [ARD-2051].Fórmula:C23H24ClN3O2Cor e Forma:SolidPeso molecular:409.91(S)-MCOPPB
CAS:(S)-MCOPPB is the S-enantiomer of MCOPPB, an orally active selective agonist for the Nociceptin/Orphanin FQ-Receptor. It inhibits signal transduction in mouse brain NOP receptors and is utilized in anxiety disorder research.Fórmula:C26H40N4Cor e Forma:SolidPeso molecular:408.623BMS-986118
CAS:BMS-986118 is a GPR40 full agonist targeting type II diabetes, prompting insulin release without hypoglycemia risk.Fórmula:C25H28ClF3N4O4Pureza:98%Cor e Forma:SolidPeso molecular:540.96(±)-J 113397
CAS:(±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM).Fórmula:C24H37N3O2Cor e Forma:SolidPeso molecular:399.57Win 45164
CAS:Win 45164 is an orally active ligand for the glucocorticoid receptor (Glucocorticoid Receptor), exhibiting activity that inhibits the pituitary-adrenal axis. It enhances liver glycogen deposition and thymolysis in adrenalectomized male rats. Additionally, Win 45164 possesses anti-inflammatory properties and is applicable in research related to inflammation and neurological disorders.Fórmula:C26H27FN2O2Peso molecular:418.503NOP agonist-1
CAS:NOP agonist-1 (compound 4) is a nociceptin opioid receptor (NOP) partial agonist that attenuates Parkinsonian disabilities in 6-OHDA hemilesioned rats [1].Fórmula:C22H34N2Peso molecular:326.52TD-0212
CAS:TD-0212: Oral dual antagonist for AT1 (pKi 8.9) & NEP inhibitor (pIC50 9.2).Fórmula:C28H34FN3O4SPureza:98%Cor e Forma:SolidPeso molecular:527.65TD-0212 TFA
CAS:TD-0212 TFA is an oral AT1 receptor antagonist & NEP inhibitor with pKi 8.9 & pIC50 9.2.Fórmula:C30H35F4N3O6SPureza:98%Cor e Forma:SolidPeso molecular:641.67Saprisartan potassium
CAS:Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.Fórmula:C25H21BrF3KN4O4SCor e Forma:SolidPeso molecular:649.52
