Receptor de Androgénio
O receptor de andrógenos (AR) é um receptor hormonal nuclear que é ativado pela ligação a andrógenos, como a testosterona e a diidrotestosterona. Este receptor desempenha um papel crucial no desenvolvimento e na manutenção das características masculinas, bem como na regulação de vários processos fisiológicos, incluindo o crescimento muscular, a libido e a densidade óssea. Inibidores do receptor de andrógenos são amplamente estudados no contexto do câncer de próstata, onde a sinalização do AR é frequentemente aumentada. Na CymitQuimica, oferecemos uma gama de moduladores do receptor de andrógenos de alta qualidade para apoiar sua pesquisa em endocrinologia, biologia do câncer e regulação hormonal.
Foram encontrados 207 produtos de "Receptor de Androgénio"
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Adrenosterone
CAS:<p>Adrenosterone (11-ketoandrostenedione) is a steroid hormone isolated from the adrenal cortex.</p>Fórmula:C19H24O3Pureza:98.13% - 98.29%Cor e Forma:SolidPeso molecular:300.39UT-155
CAS:<p>UT-155 is a selective and potent antagonist of the androgen receptor (AR) (Ki: 267 nM for UT-155 binding to AR-LBD).</p>Fórmula:C20H15F4N3O2Pureza:98.94%Cor e Forma:SolidPeso molecular:405.352,2,5,7,8-Pentamethyl-6-Chromanol
CAS:<p>2,2,5,7,8-Pentamethyl-6-Chromanol (PMC) is the anti-oxidant moiety of vitamin E (α-tocopherol), which has potent androgen receptor (AR) signaling modulation and</p>Fórmula:C14H20O2Pureza:98.72%Cor e Forma:SolidPeso molecular:220.31Allylestrenol
CAS:<p>Allylestrenol (Gestanin) is a synthetic steroid with progestational activity.</p>Fórmula:C21H32OPureza:>99.99%Cor e Forma:White Crystalline PowderPeso molecular:300.48UT-34
CAS:<p>UT-34 is a selective and orally active antagonist of second-generation pan-androgen receptor (AR) and degrader(IC50s of 211.7 nM, 262.4 nM and 215.7 nM for wild</p>Fórmula:C15H12F4N4O2Pureza:98.12%Cor e Forma:SolidPeso molecular:356.27Bicalutamide
CAS:<p>Bicalutamide (ICI-176334), a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, thereby inhibiting the</p>Fórmula:C18H14F4N2O4SPureza:98% - 99.87%Cor e Forma:Off-White Crystalline SolidPeso molecular:430.37Luxdegalutamide
CAS:<p>Luxdegalutamide (ARV-766) is an orally available and effective protein degrader of protein hydrolysis-targeted chimeras (PROTAC).Luxdegalutamide degrades the</p>Fórmula:C45H54FN7O6Pureza:99.95%Cor e Forma:SolidPeso molecular:807.95Topilutamide
CAS:<p>Topilutamide (Fluridil) is a topical nonsteroidal antiandrogen.</p>Fórmula:C13H11F6N3O5Pureza:98.77% - 99.24%Cor e Forma:SolidPeso molecular:403.23Medroxyprogesterone Acetate
CAS:<p>Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. Farlutin is a long-acting contraceptive.</p>Fórmula:C24H34O4Pureza:99.05% - 99.44%Cor e Forma:White PowderPeso molecular:386.52Zanoterone
CAS:<p>Zanoterone is an AR antagonist (androgen receptor).Zanoterone has antitumor activity for the treatment of genitourinary disorders and oncological disorders and</p>Fórmula:C23H32N2O3SPureza:99.03% - 99.92%Cor e Forma:SoildPeso molecular:416.58AR antagonist 1
CAS:<p>AR antagonist 1 is a potent antagonist of the androgen receptor.</p>Fórmula:C15H19ClN2OPureza:99.07%Cor e Forma:SolidPeso molecular:278.78SK33
CAS:<p>SK33 is a potent and tissue selective anti-androgen agent. SK33 reduces androgen receptor (AR) transcriptional activity.</p>Fórmula:C20H13F9N2O3Pureza:99.55%Cor e Forma:SolidPeso molecular:500.31Octinoxate
CAS:<p>Octinoxate (Octyl 4-methoxycinnamate) is an organic compound that is used is in sunscreens and other cosmetics to absorb UV-B rays from the sun.</p>Fórmula:C18H26O3Pureza:99.93%Cor e Forma:Less To Pale Yellow Viscous Liquid (Ntp 1992) Physical Description Colorless To Pale Yellow Viscous Liquid (Ntp 1992)Peso molecular:290.40Adrenocorticotropic hormone TFA
<p>Adrenocorticotropic hormone TFA is an adrenocorticotropic hormone involved in neurohormonal regulation of the body.</p>Pureza:99.71%Cor e Forma:Odour SolidORM-15341
CAS:<p>ORM-15341 is a potent and full antagonist for human AR (hAR)( with IC50 values of 38 nM as shown by transactivation assays in AR-HEK293 cells)</p>Fórmula:C19H17ClN6O2Pureza:98.01%Cor e Forma:SolidPeso molecular:396.83Flutamide
CAS:<p>Flutamide (SCH 13521) is an antiandrogen with about the same potency as cyproterone in rodent and canine species.</p>Fórmula:C11H11F3N2O3Pureza:99.6% - 99.96%Cor e Forma:SolidPeso molecular:276.21Cyproterone acetate
CAS:<p>Cyproterone acetate (Cyproterone 17-O-acetate) binds the androgen receptor (AR), thereby preventing androgen-induced receptor activation in target tissues and</p>Fórmula:C24H29ClO4Pureza:98.43% - 99.83%Cor e Forma:Crystals From Diisopropyl Ether OdourPeso molecular:416.943,3'-Diindolylmethane
CAS:<p>3,3'-Diindolylmethane (DIM), a small molecule compound, is a proposed Y preventive agent.</p>Fórmula:C17H14N2Pureza:99.09%Cor e Forma:SolidPeso molecular:246.31Spironolactone
CAS:<p>Spironolactone (SC9420) is an Aldosterone Antagonist. The mechanism of action of spironolactone is as an Aldosterone Antagonist.</p>Fórmula:C24H32O4SPureza:99.87%Cor e Forma:White PowderPeso molecular:416.57Nilutamide
CAS:<p>Nilutamide, a nonsteroidal anti-androgen, treats prostate cancer by blocking androgen receptors, not affecting other hormone receptors.</p>Fórmula:C12H10F3N3O4Pureza:98.67% - 99.78%Cor e Forma:Crystalline SolidPeso molecular:317.22
