
Receptor de Androgénio
O receptor de andrógenos (AR) é um receptor hormonal nuclear que é ativado pela ligação a andrógenos, como a testosterona e a diidrotestosterona. Este receptor desempenha um papel crucial no desenvolvimento e na manutenção das características masculinas, bem como na regulação de vários processos fisiológicos, incluindo o crescimento muscular, a libido e a densidade óssea. Inibidores do receptor de andrógenos são amplamente estudados no contexto do câncer de próstata, onde a sinalização do AR é frequentemente aumentada. Na CymitQuimica, oferecemos uma gama de moduladores do receptor de andrógenos de alta qualidade para apoiar sua pesquisa em endocrinologia, biologia do câncer e regulação hormonal.
Foram encontrados 229 produtos de "Receptor de Androgénio"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Darolutamide
CAS:Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).Fórmula:C19H19ClN6O2Pureza:97.36% - >99.99%Cor e Forma:SolidPeso molecular:398.85Dimethylcurcumin
CAS:Dimethylcurcumin (ASC-J9) (ASC-J9) is an androgen receptor degradation enhancer.Fórmula:C23H24O6Pureza:97.36% - 98.96%Cor e Forma:SolidPeso molecular:396.43Testosterone acetate
CAS:Testosterone acetate (NSC-523836) is a hormone with in vitro antitumor activity.Fórmula:C21H30O3Pureza:99.6%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:330.46GSK-2881078
CAS:GSK-2881078 is a selective androgen receptor modulato (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting.Fórmula:C14H13F3N2O2SPureza:98.16% - 98.81%Cor e Forma:SolidPeso molecular:330.33MI-136
CAS:MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.Fórmula:C23H21F3N6SPureza:98.63% - 99.12%Cor e Forma:SolidPeso molecular:470.51Nandrolone phenylpropionate
CAS:Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosisFórmula:C27H34O3Pureza:99.2% - 99.46%Cor e Forma:White Or Milky Crystalline PowderPeso molecular:406.56YK11
CAS:YK11 is an androgen receptor partial agonist that activates androgen receptor transcriptional activity in HEK293 cells overexpressing androgen receptors when used at a concentration of 0.1 μM, with osteogenic activity.Fórmula:C25H34O6Pureza:98.91%Cor e Forma:SoildPeso molecular:430.533-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
CAS:3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.Fórmula:C18H14N4OPureza:98.41%Cor e Forma:SolidPeso molecular:302.332-hydroxy Flutamide
CAS:2-hydroxy Flutamide is competitive inhibition of androgen receptor (AR) for the treatment of prostate cancerFórmula:C11H11F3N2O4Pureza:99.45% - 99.82%Cor e Forma:SolidPeso molecular:292.21Testosterone undecanoate
CAS:Testosterone undecanoate is a metabolite of Testosterone, which is a promising androgen for male hormonal contraception.Fórmula:C30H48O3Pureza:99.45% - 99.788%Cor e Forma:White Crystalline PowderPeso molecular:456.7Apalutamide
CAS:<p>Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.</p>Fórmula:C21H15F4N5O2SPureza:99.03% - 99.91%Cor e Forma:SolidPeso molecular:477.43AH-3960
CAS:AH-3960 是一种甲状腺激素受体 1 (PTHR1) 激动剂。Fórmula:C13H22N4O3Pureza:98.44%Cor e Forma:SolidPeso molecular:282.34VPC-13163
CAS:VPC-13566 inhibits growth in LNCaP, Enzalutamide-resistant MR49F, lowers AR gene, PSA, TMPRSS2 expression, but not in AR-independent PC3 cells.Fórmula:C16H14N2Pureza:98.02%Cor e Forma:SolidPeso molecular:234.3S-23
CAS:S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (Fórmula:C18H13ClF4N2O3Pureza:99.55%Cor e Forma:SolidPeso molecular:416.75Iprodione
CAS:Iprodione is a fungicide. Iprodione is also used in cannabis testing kits as a component of pesticide mixes.Fórmula:C13H13Cl2N3O3Pureza:98.82%Cor e Forma:Colorless Crystals Cream To Colorless Odorless PowderPeso molecular:330.17Bavdegalutamide
CAS:Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR).Fórmula:C41H43ClFN9O6Pureza:97.17% - 99.04%Cor e Forma:SolidPeso molecular:812.29N-desmethyl Enzalutamide
CAS:N-desmethyl Enzalutamide (N-desmethyl MDV 3100) is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide.Fórmula:C20H14F4N4O2SPureza:99.74%Cor e Forma:SolidPeso molecular:450.41Enzalutamide carboxylic acid
CAS:<p>Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .</p>Fórmula:C20H13F4N3O3SPureza:97.88%Cor e Forma:SolidPeso molecular:451.39Lupeol
CAS:Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.Fórmula:C30H50OPureza:98% - 99.96%Cor e Forma:Needles From Alcohol Acetone White PowderPeso molecular:426.72VPC-13566
CAS:<p>VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the</p>Fórmula:C18H14N2Pureza:99.55%Cor e Forma:SolidPeso molecular:258.32
