
Receptor de Androgénio
O receptor de andrógenos (AR) é um receptor hormonal nuclear que é ativado pela ligação a andrógenos, como a testosterona e a diidrotestosterona. Este receptor desempenha um papel crucial no desenvolvimento e na manutenção das características masculinas, bem como na regulação de vários processos fisiológicos, incluindo o crescimento muscular, a libido e a densidade óssea. Inibidores do receptor de andrógenos são amplamente estudados no contexto do câncer de próstata, onde a sinalização do AR é frequentemente aumentada. Na CymitQuimica, oferecemos uma gama de moduladores do receptor de andrógenos de alta qualidade para apoiar sua pesquisa em endocrinologia, biologia do câncer e regulação hormonal.
Foram encontrados 229 produtos de "Receptor de Androgénio"
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Inocoterone acetate
CAS:Inocoterone acetate is a nonsteroidal antiandrogen that binds to the androgen receptor and possesses antiandrogenic activity in animal models.Fórmula:C18H26O3Cor e Forma:SolidPeso molecular:290.40Linuron
CAS:Linuron herbicide disrupts photosynthesis and acts as an androgen receptor antagonist.Fórmula:C9H10Cl2N2O2Pureza:99.08%Cor e Forma:White Crystalline Solid Linuron Is A Colorless Crystals Non Corrosive Used As An HerbicidePeso molecular:249.09Enzalutamide-d3
CAS:Enzalutamide D3 is a deuterium labeled Enzalutamide . Enzalutamide is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cells.Fórmula:C21H16F4N4O2SCor e Forma:SolidPeso molecular:467.45Anti-Androgen receptor Antibody (8R912)
Anti-Androgen receptor Antibody (8R912) is a Mouse antibody targeting Androgen receptor. Anti-Androgen receptor Antibody (8R912) can be used in ICC/IF.Cor e Forma:Odour LiquidAnti-Androgen receptor Antibody (7Q574)
Anti-Androgen receptor Antibody (7Q574) is an antibody targeting Androgen receptor. Anti-Androgen receptor Antibody (7Q574) can be used in ELISA, WB, IHC.Cor e Forma:Odour LiquidMK-0773
CAS:MK-0773 (PF-05314882) is a selective androgen receptor modulator that binds to AR (IC50: 6.6 nM) for the study of diseases caused by endocrine abnormalities.Fórmula:C27H34FN5O2Pureza:98.38% - 99.14%Cor e Forma:SolidPeso molecular:479.59Anti-Androgen receptor Antibody (8H883)
Anti-Androgen receptor Antibody (8H883) is an antibody targeting Androgen receptor. Anti-Androgen receptor Antibody (8H883) can be used in ELISA, IHC.Cor e Forma:Odour LiquidARD-1676
CAS:<p>ARD-1676 is an orally administered androgen receptor (AR) PROTAC degrader that combines an AR ligand with a cereblon ligand.</p>Fórmula:C44H46ClN7O5Pureza:98%Cor e Forma:SolidPeso molecular:788.33Alternariol (Standard)
CAS:Alternariol (Standard) is the standard substance of Alternariol, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Alternariol (AOH), a mycotoxin synthesized by Alternaria species, displays numerous therapeutic and biological effects, including phytotoxic, cytotoxic, anti-HIV, anti-cancer, and anti-microbial properties. It functions by inhibiting the catalytic activity of topoisomerase I and II enzymes.Fórmula:C14H10O5Peso molecular:258.23Estradiol valerate
CAS:β-estradiol 17-valerate (EV) is a synthetic estrogen. In hormone replacement therapy drugs, it is widely used in combination with other steroid hormones.Fórmula:C23H32O3Pureza:99.11% - 99.9%Cor e Forma:NaPeso molecular:356.51Tricaprin (Standard)
CAS:Tricaprin (Standard) is the standard substance of Tricaprin, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Glycerol Tridecanoate is an orally active precursor (DA precursor) of caprylic acid that can be hydrolyzed to caprylic acid. It is a major component of medium chain triglycerides (MCT) and has antiandrogenic and antihyperglycemic properties. It can be used as an additive in food, pharmaceuticals and cosmetics.Fórmula:C33H62O6Cor e Forma:SolidPeso molecular:554.84Dehydroepiandrosterone-d2
CAS:Dehydroepiandrosterone-d2 is a deuterated compound of Dehydroepiandrosterone.Fórmula:C19H26D2O2Cor e Forma:SolidPeso molecular:290.44Rezvilutamide
CAS:Rezvilutamide (SHR3680) is an orally available androgen receptor inhibitor that crosses the blood-brain barrier and has antitumor activity.Fórmula:C22H20F3N3O4SPureza:99.96% - 99.97%Cor e Forma:SolidPeso molecular:479.47D4-abiraterone
CAS:D4-abiraterone is the active metabolite of abiraterone.Δ4-Abiraterone is a inhibitor of CYP17A1, 3β-HSD and SRD5A, and an antagonist of the androgen receptor.Fórmula:C24H29NOPureza:99.75% - 99.8%Cor e Forma:SolidPeso molecular:347.49Leelamine hydrochloride
CAS:Leelamine hydrochloride, a pine bark extract, inhibits androgen receptor and CB1, reducing lipid synthesis in prostate cancer.Fórmula:C20H32ClNPureza:98%Cor e Forma:SolidPeso molecular:321.93(Rac)-PF-998425
CAS:(Rac)-PF-998425: nonsteroidal AR antagonist, potent & selective, IC50: 26 nM (binding), 90 nM (cellular), potential for androgenetic alopecia study.Fórmula:C14H14F3NOCor e Forma:SolidPeso molecular:269.267Apalutamide-13C-d3
Apalutamide-13C-d3 is a 13C and 2H labeled Apalutamide. Apalutamide is an androgen receptor (AR) antagonist, used in research on prostate diseases.Fórmula:CC20H12F4N5O2SD3Cor e Forma:SolidPeso molecular:481.45Fenarimol
CAS:Fenarimol, a pyrimidine-type fungicide, exhibits potent inhibitory activity against BR biosynthesis.Fórmula:C17H12Cl2N2OCor e Forma:SolidPeso molecular:331.2Darolutamide
CAS:Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).Fórmula:C19H19ClN6O2Pureza:97.36% - >99.99%Cor e Forma:SolidPeso molecular:398.853-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
CAS:3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.Fórmula:C18H14N4OPureza:98.41%Cor e Forma:SolidPeso molecular:302.33

