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Receptor adrenérgico

Receptor adrenérgico

Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.

Subcategorias de "Receptor adrenérgico"

Foram encontrados 645 produtos de "Receptor adrenérgico"

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  • Heptaminol hydrochloride

    CAS:
    <p>Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.</p>
    Fórmula:C8H20ClNO
    Pureza:98.61%
    Cor e Forma:White Crystalline Powder
    Peso molecular:181.71
  • Nicergoline

    CAS:
    <p>Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.</p>
    Fórmula:C24H26BrN3O3
    Pureza:98% - 99.80%
    Cor e Forma:Solid
    Peso molecular:484.39
  • Norepinephrine bitartrate monohydrate

    CAS:
    <p>Norepinephrine bitartrate monohydrate (Levophed) is a direct alpha-adrenergic receptors stimulator.</p>
    Fórmula:C8H11NO3·C4H6O6·H2O
    Pureza:97.88% - ≥95%
    Cor e Forma:Solid
    Peso molecular:337.28
  • DL-Norepinephrine hydrochloride

    CAS:
    <p>DL-Norepinephrine hydrochloride (DL-lysine) is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400</p>
    Fórmula:C8H12ClNO3
    Pureza:98.45% - 98.82%
    Cor e Forma:Solid
    Peso molecular:205.639
  • Terazosin hydrochloride

    CAS:
    <p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>
    Fórmula:C19H26ClN5O4
    Pureza:99.69% - 99.91%
    Cor e Forma:Solid
    Peso molecular:423.89
  • Mirtazapine

    CAS:
    <p>Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.</p>
    Fórmula:C17H19N3
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:265.35
  • Methoxamine hydrochloride

    CAS:
    <p>Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.</p>
    Fórmula:C11H18ClNO3
    Pureza:99.84% - >99.99%
    Cor e Forma:Colorless Or White Plate-Like Crystals Or White Crystalline Powder Solid
    Peso molecular:247.719
  • Iobenguane sulfate

    CAS:
    <p>Iobenguane sulfate is used in radioiodinated form to diagnose and treat adrenergic tumors.</p>
    Fórmula:C8H10IN3H2O4S
    Pureza:99.04%
    Cor e Forma:Solid
    Peso molecular:324.12
  • Talipexole dihydrochloride

    CAS:
    <p>Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and</p>
    Fórmula:C10H17Cl2N3S
    Pureza:99.89%
    Cor e Forma:Light Yellow Solid
    Peso molecular:282.23
  • PF-610355 HCl


    <p>PF-610355 HCl is a selective and potent β2-adrenergic receptor agonist, a bronchodilator, and for asthma and chronic obstructive pulmonary disease.</p>
    Fórmula:C19H22ClN7O6
    Pureza:97.97%
    Cor e Forma:Solid
    Peso molecular:479.87
  • Isoxsuprine hydrochloride

    CAS:
    <p>Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.</p>
    Fórmula:C18H24ClNO3
    Pureza:99.38%
    Cor e Forma:Crystals From Water Solid
    Peso molecular:337.84
  • Blonanserin

    CAS:
    <p>Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.</p>
    Fórmula:C23H30FN3
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:367.5
  • Carbazochrome sodium sulfonate

    CAS:
    <p>Carbazochrome sodium sulfonate (AC-17) (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.</p>
    Fórmula:C10H11N4NaO5S
    Pureza:99.63%
    Cor e Forma:Orange Yellow Crystalline Powder
    Peso molecular:322.03
  • Amitriptyline hydrochloride

    CAS:
    <p>Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive</p>
    Fórmula:C20H24ClN
    Pureza:97% - 99.94%
    Cor e Forma:Crystals White To Off-White Powder
    Peso molecular:313.86
  • Metaproterenol hemisulfate

    CAS:
    <p>Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.</p>
    Fórmula:C11H17NO3·5H2O4S
    Pureza:98.53% - 99.74%
    Cor e Forma:Solid
    Peso molecular:260.3
  • Octopamine hydrochloride

    CAS:
    <p>Octopamine hydrochloride is akin to noradrenaline and acts as a neurohormone, neurotransmitter, and neuromodulator in invertebrates.</p>
    Fórmula:C8H12ClNO2
    Pureza:98.87% - 99.85%
    Cor e Forma:White Or Off-White Solid
    Peso molecular:189.64
  • Efloxate

    CAS:
    <p>Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency.</p>
    Fórmula:C19H16O5
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:324.33
  • Moxonidine

    CAS:
    <p>Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug.</p>
    Fórmula:C9H12ClN5O
    Pureza:99.81% - 99.94%
    Cor e Forma:Crystal
    Peso molecular:241.68
  • Nebivolol hydrochloride

    CAS:
    <p>Nebivolol hydrochloride is a beta-1 blocker and vasodilator treating hypertension and heart failure in the elderly.</p>
    Fórmula:C22H25F2NO4·HCl
    Pureza:99.77% - >99.99%
    Cor e Forma:White To Off-White Powder
    Peso molecular:441.90
  • 2-(1-Piperazinyl)pyrimidine

    CAS:
    <p>2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.</p>
    Fórmula:C8H12N4
    Pureza:98.46%
    Cor e Forma:Liquid - Crystal - Lump
    Peso molecular:164.21
  • Brefonalol HCl


    <p>Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.</p>
    Fórmula:C22H29ClN2O2
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:388.93
  • Terbutaline Sulfate

    CAS:
    <p>Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.</p>
    Fórmula:C12H19NO3H2SO4
    Pureza:99.47% - 99.94%
    Cor e Forma:Crystalline Powder
    Peso molecular:274.32
  • Fenoterol

    CAS:
    <p>Fenoterol is an agonist of β2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication.</p>
    Fórmula:C17H21NO4
    Pureza:98.29%
    Cor e Forma:Solid
    Peso molecular:303.35
  • Dopexamine hydrochloride

    CAS:
    <p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>
    Fórmula:C22H34Cl2N2O2
    Pureza:98.55%
    Cor e Forma:Solid
    Peso molecular:429.42
  • Olodaterol

    CAS:
    <p>Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptors</p>
    Fórmula:C21H26N2O5
    Pureza:98.9%
    Cor e Forma:Solid
    Peso molecular:386.45
  • Noradrenaline bitartrate

    CAS:
    <p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>
    Fórmula:C12H19NO10
    Pureza:99.53% - >99.99%
    Cor e Forma:Solid
    Peso molecular:337.28
  • Mirabegron

    CAS:
    <p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>
    Fórmula:C21H24N4O2S
    Pureza:99.64%
    Cor e Forma:Light Yellow To Yellow Solid
    Peso molecular:396.51
  • Labetalol

    CAS:
    <p>Labetalol: mixed alpha/beta blocker for hypertension, oral or IV; affected by CYP2C19 genetics.</p>
    Fórmula:C19H24N2O3
    Pureza:99.87% - 99.89%
    Cor e Forma:Solid
    Peso molecular:328.41
  • Midodrine hydrochloride

    CAS:
    <p>Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a prodrug in hydrochloride form.</p>
    Fórmula:C12H19ClN2O4
    Pureza:99.79% - >99.99%
    Cor e Forma:Crystalline Solid
    Peso molecular:290.74
  • Ritodrine hydrochloride

    CAS:
    <p>Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing calcium in myometrial cells.</p>
    Fórmula:C17H21NO3·HCl
    Pureza:99% - 99.52%
    Cor e Forma:Solid
    Peso molecular:323.82
  • Dronedarone hydrochloride

    CAS:
    <p>Dronedarone hydrochloride (SR33589) is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.</p>
    Fórmula:C31H44N2O5S·HCl
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:593.22
  • Olanzapine

    CAS:
    <p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>
    Fórmula:C17H20N4S
    Pureza:99.86% - ≥95%
    Cor e Forma:Yellowish Crystalline Powder
    Peso molecular:312.43
  • Hydrocortisone 17-butyrate

    CAS:
    <p>Hydrocortisone 17-butyrate (Cortisol 17-butyrate) is a glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects.</p>
    Fórmula:C25H36O6
    Pureza:98% - 99.57%
    Cor e Forma:Solid
    Peso molecular:432.55
  • Atomoxetine hydrochloride

    CAS:
    <p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>
    Fórmula:C17H22ClNO
    Pureza:99.86%
    Cor e Forma:White Solid
    Peso molecular:291.82
  • Methyldopa

    CAS:
    <p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>
    Fórmula:C10H13NO4
    Pureza:98.95% - 99.86%
    Cor e Forma:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Peso molecular:211.21
  • Labetalol hydrochloride

    CAS:
    <p>Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.</p>
    Fórmula:C19H25ClN2O3
    Pureza:99.54% - 99.85%
    Cor e Forma:Solid
    Peso molecular:364.87
  • Clonidine hydrochloride

    CAS:
    <p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>
    Fórmula:C9H10Cl3N3
    Pureza:99.16% - 99.86%
    Cor e Forma:Solid
    Peso molecular:266.55
  • Isoprenaline hydrochloride

    CAS:
    <p>Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.</p>
    Fórmula:C11H18ClNO3
    Pureza:98% - 99.65%
    Cor e Forma:Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)
    Peso molecular:247.719
  • Indacaterol maleate

    CAS:
    <p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>
    Fórmula:C28H32N2O7
    Pureza:99.03% - 99.67%
    Cor e Forma:Solid
    Peso molecular:508.56
  • Xylometazoline hydrochloride

    CAS:
    <p>Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.</p>
    Fórmula:C16H24N2·HCl
    Pureza:99.77% - 99.87%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:280.84
  • Perphenazine

    CAS:
    <p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>
    Fórmula:C21H26ClN3OS
    Pureza:99.3% - 99.99%
    Cor e Forma:Solid
    Peso molecular:403.97
  • Terbutaline

    CAS:
    <p>Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterol</p>
    Fórmula:C12H19NO3
    Pureza:99.12%
    Cor e Forma:Solid
    Peso molecular:225.3
  • Ifenprodil

    CAS:
    <p>Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 &amp; GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.</p>
    Fórmula:C21H27NO2
    Pureza:99.58%
    Cor e Forma:White Crystalline Powder
    Peso molecular:325.44
  • Dabuzalgron

    CAS:
    <p>Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence.</p>
    Fórmula:C12H16ClN3O3S
    Pureza:98.35%
    Cor e Forma:Solid
    Peso molecular:317.79
  • Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Fórmula:C10H11ClFNO2
    Pureza:99.98%
    Cor e Forma:Soild
    Peso molecular:231.65
  • Gemfibrozil

    CAS:
    <p>Gemfibrozil, a fibric acid derivative, stimulates PPARalpha, boosts fatty acid oxidation, LPL, lowers VLDL-C, apoC-III, and raises HDL-C.</p>
    Fórmula:C15H22O3
    Pureza:99.53% - 99.88%
    Cor e Forma:Crystals From Hexane Solid
    Peso molecular:250.33
  • Metoprolol tartrate

    CAS:
    <p>Metoprolol Tartrate is a blocker of the cardioselective β-adrenergic receptor.</p>
    Fórmula:C15H25NO3C4H6O6
    Pureza:99.72% - 99.93%
    Cor e Forma:White To Off-White / Powder
    Peso molecular:684.81
  • Nylidrin hydrochloride

    CAS:
    <p>Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells &amp; human basophils.</p>
    Fórmula:C19H26ClNO2
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:335.87
  • Clorprenaline hydrochloride

    CAS:
    <p>Clorprenaline hydrochloride (Clorprenaline HCl) is a beta-2 adrenergic agonist with bronchodilator activity.</p>
    Fórmula:C11H17Cl2NO
    Pureza:99.59% - >99.99%
    Cor e Forma:Solid
    Peso molecular:250.16
  • Trifluoperazine dihydrochloride

    CAS:
    <p>Trifluoperazine dihydrochloride (SKF5019) is a potent dopamine D2 receptor inhibitor used as an antipsychotic and an antiemetic.</p>
    Fórmula:C21H26Cl2F3N3S
    Pureza:99.57% - 99.96%
    Cor e Forma:Cream Fine Powder
    Peso molecular:480.43
  • Tolazoline hydrochloride

    CAS:
    <p>Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary</p>
    Fórmula:C10H13ClN2
    Pureza:99.67%
    Cor e Forma:Pale Yellow Crystalline Solid
    Peso molecular:196.68
  • DSP-4 hydrochloride

    CAS:
    <p>DSP-4 hydrochloride is a neurotoxin that degrades noradrenergic neurons in rats and crosses the blood-brain barrier.</p>
    Fórmula:C11H16BrCl2N
    Pureza:99.9%
    Cor e Forma:Solid
    Peso molecular:313.06
  • Bisoprolol hemifumarate

    CAS:
    <p>Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart,</p>
    Fórmula:C20H33NO6
    Pureza:98.69% - 99.84%
    Cor e Forma:White To Offf-White Powder
    Peso molecular:383.49
  • Fenspiride hydrochloride

    CAS:
    <p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>
    Fórmula:C15H20N2O2·HCl
    Pureza:99.64% - 99.92%
    Cor e Forma:Solid
    Peso molecular:296.79
  • Salmeterol

    CAS:
    <p>Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.</p>
    Fórmula:C25H37NO4
    Pureza:99.2% - 99.9%
    Cor e Forma:Solid
    Peso molecular:415.57
  • Bucumolol

    CAS:
    <p>Bucumolol (Bucumarol) is a β-adrenergic blocking agent and a local anesthetic with antihypertensive activity and can be used to study myocardial infarction.</p>
    Fórmula:C17H23NO4
    Pureza:99.66%
    Cor e Forma:Soild
    Peso molecular:305.37
  • Acebutolol hydrochloride

    CAS:
    <p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension &amp; ventricular arrhythmias.</p>
    Fórmula:C18H29ClN2O4
    Pureza:99.92% - >99.99%
    Cor e Forma:White Or Slightly Off-White Crystalline Powder Solid
    Peso molecular:372.89
  • Synephrine

    CAS:
    <p>Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.</p>
    Fórmula:C9H13NO2
    Pureza:99.274% - >99.99%
    Cor e Forma:Solid
    Peso molecular:167.21
  • Phenoxybenzamine hydrochloride

    CAS:
    <p>Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.</p>
    Fórmula:C18H23Cl2NO
    Pureza:98.04% - >99.99%
    Cor e Forma:Antihypertensive Drug
    Peso molecular:340.3
  • Tolamolol

    CAS:
    <p>Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of the S-T segment and can be used in the</p>
    Fórmula:C19H24N2O4
    Pureza:98.59%
    Cor e Forma:Solid
    Peso molecular:344.4
  • Tizanidine hydrochloride

    CAS:
    <p>Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.</p>
    Fórmula:C9H9Cl2N5S
    Pureza:99.96%
    Cor e Forma:Solid White
    Peso molecular:290.17
  • Delequamine

    CAS:
    <p>Delequamine (RS 15385-197) is a TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study mental retardation.</p>
    Fórmula:C18H26N2O3S
    Pureza:99.39%
    Cor e Forma:Solid
    Peso molecular:350.48
  • Phenylephrine hydrochloride

    CAS:
    <p>Phenylephrine hydrochloride (NCI-c55641) is a selective agonist of the α1-adrenergic receptor.</p>
    Fórmula:C9H14ClNO2
    Pureza:99.51% - 99.97%
    Cor e Forma:Physical Description Odorless White Microcrystalline Powder Bitter Taste Ph (1%
    Peso molecular:203.67
  • Moxisylyte hydrochloride

    CAS:
    <p>Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.</p>
    Fórmula:C16H26ClNO3
    Pureza:99.93% - ≥95%
    Cor e Forma:Solid
    Peso molecular:315.84
  • Isoferulic acid

    CAS:
    <p>Isoferulic acid (Hesperetate) exhibits hypoglycemic properties.</p>
    Fórmula:C10H10O4
    Pureza:99.36% - 99.49%
    Cor e Forma:Solid
    Peso molecular:194.18
  • Carvedilol phosphate hemihydrate

    CAS:
    <p>Carvedilol phosphate hemihydrate (BM 14190 phosphate hemihydrate) is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent.</p>
    Fórmula:C24H26N2O4·5H2O·H3O4P
    Pureza:99.24% - 99.98%
    Cor e Forma:Solid
    Peso molecular:513.49
  • CXCR7 antagonist-1

    CAS:
    <p>CXCR7 antagonist-1 is a specific antagonist of the binding of the SDF-1 chemokine or I-TAC to the chemokine receptor CXCR7.</p>
    Fórmula:C21H19FN6O
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:390.41
  • Tetrahydrozoline

    CAS:
    <p>Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.</p>
    Fórmula:C13H16N2
    Pureza:97.85% - 99.77%
    Cor e Forma:Solid
    Peso molecular:200.28
  • 2',5'-Dideoxyadenosine

    CAS:
    <p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>
    Fórmula:C10H13N5O2
    Pureza:99.55%
    Cor e Forma:White Solid
    Peso molecular:235.24
  • Centanafadine hydrochloride

    CAS:
    <p>Centanafadine HCl is a NE/DA reuptake inhibitor, also affects serotonin (IC50: NE 6 nM, DA 38 nM, serotonin 83 nM).</p>
    Fórmula:C15H16ClN
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:245.75
  • Ifenprodil Tartrate

    CAS:
    <p>Ifenprodil is a selective NMDA receptor (glutamate) antagonist.</p>
    Fórmula:C21H27NO2C4H6O6
    Pureza:99.02% - 99.55%
    Cor e Forma:Solid
    Peso molecular:400.49
  • Metaraminol tartrate

    CAS:
    <p>Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>
    Fórmula:C13H19NO8
    Pureza:99.68%
    Cor e Forma:White Powder
    Peso molecular:317.29
  • Silodosin

    CAS:
    <p>Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.</p>
    Fórmula:C25H32F3N3O4
    Pureza:99.282% - 99.76%
    Cor e Forma:Colorless To Pink Solid
    Peso molecular:495.53
  • Naphazoline hydrochloride

    CAS:
    <p>Naphazoline hydrochloride (Naphazoline HCl) is an adrenergic vasoconstrictor agent used as a decongestant.</p>
    Fórmula:C14H15ClN2
    Pureza:97.93%
    Cor e Forma:White Crystalline Powder White Crystalline Powder
    Peso molecular:246.74
  • Nardeterol HCl


    <p>Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4</p>
    Fórmula:C20H25ClFN3O2
    Pureza:97.72% - 98.65%
    Cor e Forma:Soild
    Peso molecular:393.88
  • Clozapine

    CAS:
    <p>Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.</p>
    Fórmula:C18H19ClN4
    Pureza:99.91% - 99.93%
    Cor e Forma:Yellow Crystals From Acetone-Petroleum Ether Solid
    Peso molecular:326.82
  • Carteolol hydrochloride

    CAS:
    <p>Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.</p>
    Fórmula:C16H24N2O3·HCl
    Pureza:99.84% - 99.91%
    Cor e Forma:Solid
    Peso molecular:328.83
  • Solabegron

    CAS:
    <p>Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR</p>
    Fórmula:C23H23ClN2O3
    Pureza:97.89%
    Cor e Forma:Solid
    Peso molecular:410.89
  • Buflomedil hydrochloride

    CAS:
    <p>Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.</p>
    Fórmula:C17H26ClNO4
    Pureza:99.7% - 99.91%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:343.85
  • Salbutamol

    CAS:
    <p>Salbutamol (Albuterol) 是短效的 β2 肾上腺素受体激动剂,用于哮喘和慢性阻塞性肺疾病(COPD) 引发的支气管痉挛的研究。</p>
    Fórmula:C13H21NO3
    Pureza:91.59% - 99.9%
    Cor e Forma:White To Off-White Crystalline Solid Solid
    Peso molecular:239.31
  • Alfuzosin hydrochloride

    CAS:
    <p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>
    Fórmula:C19H27N5O4·HCl
    Pureza:99.78%
    Cor e Forma:White To Off-White Solid
    Peso molecular:425.91
  • Propafenone

    CAS:
    <p>Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.</p>
    Fórmula:C21H27NO3
    Pureza:99.02%
    Cor e Forma:Solid
    Peso molecular:341.44
  • Bambuterol hydrochloride

    CAS:
    <p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>
    Fórmula:C18H30ClN3O5
    Pureza:99.53% - 99.61%
    Cor e Forma:White Solid
    Peso molecular:403.91
  • Phentolamine mesylate

    CAS:
    <p>Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.</p>
    Fórmula:C17H19N3O·CH4O3S
    Pureza:99.77% - >99.99%
    Cor e Forma:By The Metabolic Processes Of Bacillus Subtilis And Licheniformis
    Peso molecular:377.46
  • SR59230A

    CAS:
    <p>SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).</p>
    Fórmula:C23H29NO6
    Pureza:98.84%
    Cor e Forma:Solid
    Peso molecular:415.48
  • Betaxolol hydrochloride

    CAS:
    <p>Betaxolol HCl (SL 75212) is a cardioselective beta-blocker for hypertension without reported liver injury.</p>
    Fórmula:C18H30ClNO3
    Pureza:99.48% - 99.56%
    Cor e Forma:Solid
    Peso molecular:343.89
  • Adrenalone hydrochloride

    CAS:
    <p>Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.</p>
    Fórmula:C9H11NO3·HCl
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:217.65
  • JP1302 dihydrochloride

    CAS:
    <p>JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.</p>
    Fórmula:C24H26Cl2N4
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:441.4
  • Urapidil hydrochloride

    CAS:
    <p>Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.</p>
    Fórmula:C20H29N5O3·HCl
    Pureza:99.58%
    Cor e Forma:White Or Off-White Crystalline Powder
    Peso molecular:423.94
  • (S)-(-)-Atenolol

    CAS:
    <p>(S)-(-)-Atenolol has beta-adrenergic blocking effects.</p>
    Fórmula:C14H22N2O3
    Pureza:99.31% - 99.81%
    Cor e Forma:Solid
    Peso molecular:266.34
  • Naftopidil

    CAS:
    <p>Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-</p>
    Fórmula:C24H28N2O3
    Pureza:99.60% - 99.97%
    Cor e Forma:White Crystalline Powder
    Peso molecular:392.49
  • (3aR,9aR)-Fluparoxan

    CAS:
    <p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Fórmula:C10H10FNO2
    Pureza:97.82%
    Cor e Forma:Soild
    Peso molecular:195.19
  • Prazosin hydrochloride

    CAS:
    <p>Prazosin HCl, a synthetic antiadrenergic, treats hypertension, heart failure, and more by relaxing blood vessels with an unclear mechanism.</p>
    Fórmula:C19H22ClN5O4
    Pureza:99.88% - >99.99%
    Cor e Forma:White To Tan Powder Off-White To Yellow Powder
    Peso molecular:419.86
  • Tolnapersine TFA


    <p>Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.</p>
    Fórmula:C23H27F3N2O3
    Pureza:99.14%
    Cor e Forma:Soild
    Peso molecular:436.47
  • Doxazosin mesylate

    CAS:
    <p>Doxazosin mesylate (UK 33274 mesylate)(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.</p>
    Fórmula:C24H29N5O8S
    Pureza:99.92%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:547.58
  • RS 15385-198

    CAS:
    <p>RS 15385-198 is a less active isomer of Delequamine. Delequamine is a selective alpha2-adrenergic receptor antagonist.</p>
    Fórmula:C18H26N2O3S
    Pureza:>99.99%
    Cor e Forma:Soild
    Peso molecular:350.48
  • (R)-Terazosin

    CAS:
    <p>R-Terazosin is the active R-enantiomer and potent α1-adrenoceptor antagonist (Ki: α1a 6.51 nM, α1b 1.01 nM, α1d 1.97 nM).</p>
    Fórmula:C19H25N5O4
    Pureza:98.87% - 98.96%
    Cor e Forma:Solid
    Peso molecular:387.43
  • Tamsulosin hydrochloride

    CAS:
    <p>Tamsulosin hydrochloride (Flomax hydrochloride) is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 adrenergic antagonist activity.</p>
    Fórmula:C20H29ClN2O5S
    Pureza:95.45% - 99.95%
    Cor e Forma:White To Off-White Solid
    Peso molecular:444.97
  • Paliperidone

    CAS:
    <p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>
    Fórmula:C23H27FN4O3
    Pureza:95% - 99.08%
    Cor e Forma:Off White To Light Orange Coloured Solid
    Peso molecular:426.48
  • AA 497 HCl

    CAS:
    <p>AA 497, a beta-2 agonist, suppresses Ca spikes.</p>
    Fórmula:C14H22ClNO3
    Cor e Forma:Solid
    Peso molecular:287.78
  • Ivabradine-d3 hydrochloride

    CAS:
    <p>Ivabradine HCl: novel If blocker, IC50 2.9 μM, slows heart rate; D3 version is deuterium labeled.</p>
    Fórmula:C27H37ClN2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:508.07
  • Acrinor

    CAS:
    <p>Acrinor is a adrenergic beta receptor agonist.</p>
    Fórmula:C35H46Cl2N10O8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:805.72
  • Abediterol napadisylate

    CAS:
    <p>Abediterol napadisylate is a novel long-acting β2-agonist in persistent asthma that is efficacy, safe, and tolerable.</p>
    Fórmula:C60H68F4N4O14S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1209.32
  • Vilanterol

    CAS:
    <p>Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and asthma.</p>
    Fórmula:C24H33Cl2NO5
    Pureza:97.47% - 99.46%
    Cor e Forma:Solid
    Peso molecular:486.43
  • Methylhexanamine hydrochloride

    CAS:
    <p>Methylhexanamine hydrochloride is a fatty amine and vasoconstrictor that functions as a nasal decongestant when inhaled through the nasal mucosa.</p>
    Fórmula:C7H18ClN
    Cor e Forma:Solid
    Peso molecular:151.68
  • Saterinone

    CAS:
    <p>Saterinone: PDE III inhibitor, α-1-adrenoceptor antagonist, vasodilator, used for acute chronic heart failure, IC50 2.3x10^-5 M.</p>
    Fórmula:C27H30N4O4
    Pureza:98.23%
    Cor e Forma:Solid
    Peso molecular:474.55
  • Esmolol acid hydrochloride

    CAS:
    <p>Esmolol acid (ASL-8123) hydrochloride is a mild antagonist of β-adrenergic receptors. It inhibits the heart rate and diastolic pressure responses induced by Isoproterenol in a dose-dependent manner and is applicable for renal failure research.</p>
    Fórmula:C15H24ClNO4
    Cor e Forma:Solid
    Peso molecular:317.81
  • Prazobind

    CAS:
    <p>Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.</p>
    Fórmula:C23H27N5O3
    Cor e Forma:Solid
    Peso molecular:421.501
  • Tienoxolol FA


    <p>Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.</p>
    Fórmula:C22H30N2O7S
    Pureza:97.05% - 98.85%
    Cor e Forma:Soild
    Peso molecular:466.55
  • Metaraminol

    CAS:
    <p>Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>
    Fórmula:C9H13NO2
    Cor e Forma:Solid
    Peso molecular:167.21
  • CACPD2011a-0001278239

    CAS:
    <p>CACPD2011a-0001278239 is a β2AR hybrid agonist with high affinity binding to both the wild-type and T164I β2AR variants. It exhibits neither cytotoxicity nor mutagenicity, making it suitable for asthma research.</p>
    Fórmula:C21H22N4O4
    Cor e Forma:Solid
    Peso molecular:394.42
  • Detomidine carboxylic acid

    CAS:
    <p>Detomidine carboxylic acid, a urine metabolite of detomidine, is a synthetic α2-agonist, animal analgesic, with cardiac, respiratory, and diuretic effects.</p>
    Fórmula:C12H12N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:216.24
  • Benzquinamide

    CAS:
    <p>Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer</p>
    Fórmula:C22H32N2O5
    Pureza:94.86%
    Cor e Forma:Solid
    Peso molecular:404.5
  • SB-206606

    CAS:
    <p>SB-206606 is a novel, highly specific radioactive ligand for the β3-adrenergic receptor.</p>
    Fórmula:C19H22ClNO4
    Cor e Forma:Solid
    Peso molecular:363.83
  • (R)-(+)-Atenolol

    CAS:
    <p>(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.</p>
    Fórmula:C14H22N2O3
    Pureza:98.72%
    Cor e Forma:Solid
    Peso molecular:266.34
  • Azepexole hydrochloride

    CAS:
    <p>Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaesthetic</p>
    Fórmula:C9H16ClN3O
    Pureza:99.88% - 99.89%
    Cor e Forma:Soild
    Peso molecular:217.7
  • (±)5(6)-EET

    CAS:
    <p>5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.</p>
    Fórmula:C20H32O3
    Cor e Forma:Solid
    Peso molecular:320.473
  • N-Nitroso Atenolol

    CAS:
    <p>N-Nitroso Atenolol is a derivative of Atenolol. At concentrations ranging from 0.1 to 1 mM, it induces DNA fragmentation in rat hepatocytes.</p>
    Fórmula:C14H21N3O4
    Cor e Forma:Solid
    Peso molecular:295.33
  • Mapenterol hydrochloride

    CAS:
    <p>Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.</p>
    Fórmula:C14H21Cl2F3N2O
    Pureza:98.11% - 99.98%
    Cor e Forma:Solid
    Peso molecular:361.23
  • Sibenadet hydrochloride

    CAS:
    <p>Sibenadet, a D2/beta2-agonist, is potential useful for the treatment of symptoms of chronic obstructive pulmonary disease.</p>
    Fórmula:C22H29ClN2O5S2
    Cor e Forma:Solid
    Peso molecular:501.06
  • α1A-AR Degrader 9c

    CAS:
    <p>α1A-AR Degrader 9c is a potent, selective, and reversible PROTAC degrader targeting the α1A adrenergic receptor (α1A-AR) with a DC50 of 2.86 μM.</p>
    Fórmula:C38H43N11O11
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:829.82
  • Pafenolol

    CAS:
    <p>Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.</p>
    Fórmula:C18H31N3O3
    Pureza:98.33%
    Cor e Forma:Solid
    Peso molecular:337.46
  • AdTx1


    <p>Selective non-competitive α1A adrenoceptor antagonist with Ki of 0.35 nM; inactive on other GPCRs; affects phenylephrine actions.</p>
    Fórmula:C310H481N87O100S8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:7283.22
  • O-Desmethyl Mebeverine alcohol

    CAS:
    <p>Mebeverine metabolite O-desmethyl alcohol inhibits α1 receptors, relaxing the gut.</p>
    Fórmula:C15H25NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:251.36
  • Corynanthine

    CAS:
    <p>Corynanthe is a plant alkaloid. Corynanthe also has an alpha-2-adrenergic blocking activity.</p>
    Fórmula:C21H26N2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:354.44
  • Picumeterol FA


    <p>picumeterol FA is a potent and selective β2-adrenergic receptor agonist.</p>
    Fórmula:C22H31Cl2N3O4
    Pureza:99.8%
    Cor e Forma:Soild
    Peso molecular:472.4
  • Mabuterol free base

    CAS:
    <p>Mabuterol: selective β2 agonist, inhibits isoprenaline, affects rat uterus and rabbit jejunum, alters intestinal propulsion.</p>
    Fórmula:C13H18ClF3N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:310.74
  • Adrenergic Receptor-Targeted Compound Library


    <p>A unique collection of 193 bioactive compounds specifically targeting adrenergic receptors, effective tool for screening new drugs or new target identification;</p>
    Cor e Forma:Odour Solid
  • Mibenratide TFA


    <p>Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].</p>
    Pureza:98%
    Cor e Forma:Odour Solid
  • BM213 acetate


    <p>BM213 acetate is a selective C5aR1 agonist with antitumor activity that induces C5aR1-mediated calcium mobilization and pERK1/2 signaling.</p>
    Fórmula:C45H74N12O12
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:975.14
  • G-Protein antagonist peptide acetate


    <p>G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding.</p>
    Fórmula:C59H68N12O11S
    Pureza:98.06%
    Cor e Forma:Solid
    Peso molecular:1153.33
  • Conopeptide rho-TIA

    CAS:
    <p>Conopeptide rho-TIA, a peptide from Conus tulipa venom, acts as a selective, noncompetitive inhibitor at the human α1B-Adrenergic Receptor and as a competitive</p>
    Fórmula:C105H160N36O21S4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:2390.88
  • Isoprenaline

    CAS:
    <p>Isoprenaline is a non-selective and orally active β-adrenoceptor agonist.Isoproterenol is a potent peripheral vasodilator and bronchodilator.</p>
    Fórmula:C11H17NO3
    Pureza:99.31%
    Cor e Forma:Solid
    Peso molecular:211.26
  • Dipivefrin

    CAS:
    <p>Dipivefrin is a prodrug of epinephrine, and is used to treat open-angle glaucoma.</p>
    Fórmula:C19H29NO5
    Cor e Forma:Solid
    Peso molecular:351.44
  • Vatinoxan

    CAS:
    <p>Vatinoxan is a peripheral α2 adrenoreceptor antagonist.</p>
    Fórmula:C20H26N4O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:418.51
  • Agaridoxin

    CAS:
    <p>Agaridoxin is a mushroom metabolite.</p>
    Fórmula:C11H14N2O5
    Cor e Forma:Solid
    Peso molecular:254.242
  • L-770644 dihydrochloride

    CAS:
    <p>L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.</p>
    Fórmula:C30H38ClN7O4S
    Cor e Forma:Solid
    Peso molecular:628.19
  • Neurotransmitter Receptor Compound Library


    <p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>
    Cor e Forma:Odour Solid
  • Metipranolol

    CAS:
    <p>Metipranolol (Betamann) is a type of β- Adrenergic receptors( β- A potent antagonist of adrenergic receptor on guinea pig atria β 1- Adrenergic receptors and rat uterus β The 2-adrenergic receptor exhibited the beta blocking potentials (pA2) of 8.3 and 8.4, respectively. It is also a potent substituent in the 3H DHA binding assay, with a ligand concentration of 0.7 nM and a Ki of 39 ± 24 nM.</p>
    Fórmula:C17H27NO4
    Pureza:98.37%
    Cor e Forma:Solid
    Peso molecular:309.4
  • Metaterol

    CAS:
    <p>Metaterol is a bioactive chemical.</p>
    Fórmula:C11H17NO2
    Cor e Forma:Solid
    Peso molecular:195.2582
  • Bamosiran

    CAS:
    <p>Bamosiran, a small interfering RNA (siRNA), specifically targets the β-adrenergic receptor 2 to reduce intraocular pressure.</p>
    Cor e Forma:Solid
  • L-770644

    CAS:
    <p>L-770644 is an agonist of B3 adrenergic receptor.</p>
    Fórmula:C30H37N7O4S
    Cor e Forma:Solid
    Peso molecular:591.72
  • Ethylnorepinephrine hydrochloride

    CAS:
    <p>Ethylnorepinephrine hydrochloride is a unique bronchodilator.</p>
    Fórmula:C10H16ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:233.69
  • O-Desmethyl Mebeverine alcohol hydrochloride

    CAS:
    <p>O-Desmethyl Mebeverine alcohol HCl, a metabolite of Mebeverine, is a strong α1 inhibitor, relaxing the GI tract.</p>
    Fórmula:C15H26ClNO2
    Cor e Forma:Solid
    Peso molecular:287.83
  • Amitraz

    CAS:
    <p>Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine demodectic mange.</p>
    Fórmula:C19H23N3
    Pureza:99.88%
    Cor e Forma:White/Pale Yellow Crystalline Solid
    Peso molecular:293.41
  • Nolomirole

    CAS:
    <p>Nolomirole is a dopamine receptor agonist that reduces symptoms of congestive heart failure caused by monoclinine.</p>
    Fórmula:C19H27NO4
    Cor e Forma:Solid
    Peso molecular:333.42
  • Terazosin dimer impurity dihydrochloride

    CAS:
    <p>Terazosin dimer impurity dihydrochloride is a chemical byproduct of the α1-antagonist Terazosin, derived from quinazoline.</p>
    Fórmula:C24H30Cl2N8O4
    Cor e Forma:Solid
    Peso molecular:565.46
  • BMS-196085

    CAS:
    <p>BMS-196085 is an effective and selective human β( 3) All agonists of adrenergic receptors, in β( 1) Partial agonist activity was 45%.</p>
    Fórmula:C24H26F2N2O5S
    Cor e Forma:Solid
    Peso molecular:492.54
  • Phenylethanolamine A

    CAS:
    <p>Phenylethanolamine A is a β-adrenergic agonist and a byproduct of the Ractopamine synthesis process.</p>
    Fórmula:C19H24N2O4
    Cor e Forma:Solid
    Peso molecular:344.40
  • Bucindolol Formate


    <p>Bucindolol is a β1-adrenergic blocker with sympathomimetic activity, used in heart failure research.</p>
    Fórmula:C23H27N3O4
    Pureza:99.76% - 99.88%
    Cor e Forma:Solid
    Peso molecular:409.48
  • Phenoxybenzamine

    CAS:
    <p>Phenoxybenzamine blocks α-1 receptors, potentially reducing neuroinflammation post brain trauma.</p>
    Fórmula:C18H22ClNO
    Pureza:98%
    Cor e Forma:Crystals From Petroleum Ether Solid
    Peso molecular:303.83
  • Benzoquinamide hydrochloride

    CAS:
    <p>Benzoquinamide hydrochloride (3-carbamoyl-N,N-diethyl-1,3,4,6,7,11b-hexahydro-9,11-dimethoxy-2H-benzo[a]quinolizin-2-yl acetate hydrochloride) is an antiemetic</p>
    Fórmula:C22H33ClN2O5
    Pureza:97.13% - 99.56%
    Cor e Forma:Solid
    Peso molecular:440.96
  • allo-Yohimbine

    CAS:
    <p>allo-Yohimbine is a biochemical.</p>
    Fórmula:C21H26N2O3
    Cor e Forma:Solid
    Peso molecular:354.44
  • YM 09538

    CAS:
    <p>YM 09538 is a biochemical.</p>
    Fórmula:C18H25ClN2O5S
    Cor e Forma:Solid
    Peso molecular:416.92
  • 5-Bromoimidazo[1,2-A]Pyrazine

    CAS:
    <p>5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.</p>
    Fórmula:C6H4BrN3
    Pureza:97.04%
    Cor e Forma:Solid
    Peso molecular:198.02
  • Synephrine hemitartrate

    CAS:
    <p>Synephrine hemitartrate, an alkaloid from Citrus aurantium, is a sympathomimetic for weight loss, with α and β-adrenergic action.</p>
    Fórmula:C9H13NO2C4H6O6
    Cor e Forma:Solid
    Peso molecular:242.26
  • Yohimbine

    CAS:
    <p>Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)</p>
    Fórmula:C21H26N2O3
    Pureza:99.78% - 99.89%
    Cor e Forma:Solid
    Peso molecular:354.4
  • Propranolol hydrochloride

    CAS:
    <p>Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverse</p>
    Fórmula:C16H22ClNO2
    Pureza:99.94% - >99.99%
    Cor e Forma:White Or Almost White Powder White Powder
    Peso molecular:295.80
  • Oxaprotiline hydrochloride

    CAS:
    <p>Oxaprotiline hydrochloride is an antidepressant.</p>
    Fórmula:C20H24ClNO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:329.86
  • ARC 239 dihydrochloride

    CAS:
    <p>ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).</p>
    Fórmula:C24H31Cl2N3O3
    Pureza:99.72%
    Cor e Forma:Solid
    Peso molecular:480.43
  • Desglymidodrine

    CAS:
    <p>Desglymidodrine (ST 1059) is an α1-adrenoceptor agonist and vasoconstrictor, used in cardiovascular research and neurocardiogenic syncope studies.</p>
    Fórmula:C10H15NO3
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:197.23
  • Tamsolusin Hydrochloride

    CAS:
    <p>Tamsolusin Hydrochloride (YM 12617) is a highly selective alpha-1A adrenergic receptor antagonist used in the treatment of benign prostatic hypertrophy.</p>
    Fórmula:C20H29ClN2O5S
    Pureza:99.92%
    Cor e Forma:Soild
    Peso molecular:444.97
  • S(-)-Bisoprolol fumarate

    CAS:
    <p>S(-)-Bisoprolol fumarate is a selective β1-blocker for hypertension and heart research.</p>
    Fórmula:C18H31NO4·xC4H4O4
    Cor e Forma:Solid
    Peso molecular:441.521
  • (+)-ORM-10921

    CAS:
    <p>(+)-ORM-10921 is a conformation of ORM-10921 and can be used in chemical synthesis studies.</p>
    Fórmula:C18H23NO2
    Pureza:99.85%
    Cor e Forma:Soild
    Peso molecular:285.38
  • Formoterol O-β-D-Glucuronide

    CAS:
    <p>Formoterol O-β-D-glucuronide is a metabolite of formoterol .</p>
    Fórmula:C25H32N2O10
    Cor e Forma:Solid
    Peso molecular:520.535
  • YS-49 monohydrate


    <p>YS-49, a PI3K/Akt activator, curbs RhoA/PTEN; inhibits VSMC growth by inducing HO-1; an isoquinoline alkaloid that stimulates cardiac β-adrenoceptors.</p>
    Fórmula:C20H22BrNO3
    Cor e Forma:Solid
    Peso molecular:404.3
  • CTP-amiodarone


    <p>CTP-amiodarone, a cellular-penetrating conjugate of myocardial cell-targeting peptide and Amiodarone, exhibits anti-arrhythmic activity by blocking Na+, K+, and Ca2+ channels as well as β-adrenergic receptors.</p>
    Fórmula:C97H131F3I2N20O25S2
    Cor e Forma:Solid
    Peso molecular:2352.13
  • Nadolol

    CAS:
    <p>Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities.</p>
    Fórmula:C17H27NO4
    Pureza:99.87% - 99.92%
    Cor e Forma:White To Off-White Crystalline Powder Solid
    Peso molecular:309.40
  • D-Epinephrine

    CAS:
    <p>D-Epinephrine: a hormone and drug, boosts heart rate, muscle blood flow, pupil size, and sugar levels in stress responses.</p>
    Fórmula:C9H13NO3
    Cor e Forma:Solid
    Peso molecular:183.2
  • Carvedilol

    CAS:
    <p>Carvedilol (SKF 105517) Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intrinsic sympathomimetic activity. The S enantiomer of carvedilol nonselectively binds to and blocks beta-adrenergic receptors, thereby exerting negative inotropic and chronotropic effects, and leading to a reduction in cardiac output. In addition, both enantiomers of carvedilol bind to and block alpha 1-adrenergic receptors, thereby causing vasodilation and reducing peripheral vascular resistance.</p>
    Fórmula:C24H26N2O4
    Pureza:99.73% - 99.97%
    Cor e Forma:Colourless Crystalline Powder
    Peso molecular:406.47
  • Chir 2279

    CAS:
    <p>CHIR 2279, a peptoid trimer, binds alpha 1-adrenoceptors, blocking epinephrine effects in dogs (pseudo pA2 6.86).</p>
    Fórmula:C34H36N4O4
    Cor e Forma:Solid
    Peso molecular:564.67
  • 5-hydroxy Propranolol

    CAS:
    <p>5-hydroxy Propranolol, a propranolol metabolite, is formed in the liver via P450 2D6.</p>
    Fórmula:C16H21NO3
    Cor e Forma:Solid
    Peso molecular:275.348
  • Upidosin

    CAS:
    <p>Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.</p>
    Fórmula:C31H33N3O4
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:511.61
  • Apigenin 6,8-di-C-α-L-arabinopyranoside

    CAS:
    <p>Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.</p>
    Fórmula:C25H26O13
    Cor e Forma:Solid
    Peso molecular:534.47
  • Besipirdine hydrochloride

    CAS:
    <p>Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with cardiovascular activity that inhibits the uptake of biogenic amines.</p>
    Fórmula:C16H18ClN3
    Pureza:98.45%
    Cor e Forma:Soild
    Peso molecular:287.79
  • Tizanidine

    CAS:
    <p>Tizanidine, an α2-adrenergic receptor agonist, suppresses the release of neurotransmitters from central nervous system (CNS) noradrenergic neurons.</p>
    Fórmula:C9H8ClN5S
    Pureza:99.11%
    Cor e Forma:White Solid
    Peso molecular:253.71
  • Carazolol-d7

    CAS:
    <p>Carazolol-d7 is the deuterium-labeled isotope of Carazolol, commonly used in pharmacokinetic studies to investigate the metabolic pathways of Carazolol.</p>
    Fórmula:C18H22N2O2
    Cor e Forma:Solid
    Peso molecular:305.42
  • ACTH (1-14)

    CAS:
    <p>ACTH (1-14) is a pituitary hormone fragment that controls cortisol and androgen levels.</p>
    Fórmula:C77H109N21O20S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1680.88
  • Meluadrine tartrate

    CAS:
    <p>Meluadrine tartrate is an endogenous metabolite.</p>
    Fórmula:C16H24ClNO8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:393.82
  • Nafetolol

    CAS:
    <p>Nafetolol (K 5407) is a biochemical reagent that can be used to synthesize other compounds.</p>
    Fórmula:C19H29NO3
    Pureza:98.91%
    Cor e Forma:Solid
    Peso molecular:319.44
  • AG-825

    CAS:
    <p>AG-825(Tyrphostin C15) is a selective and competitive ErbB2 inhibitor that inhibits tyrosine phosphorylation with an IC50 value of 0.35 μM.AG-825 (Tyrphostin</p>
    Fórmula:C19H15N3O3S2
    Pureza:98.43%
    Cor e Forma:Yellow Solid
    Peso molecular:397.47
  • Esprolol

    CAS:
    <p>Esprolol (ACC-9369 free base) is a novel beta-adrenergic antagonist used to study exertional angina.</p>
    Fórmula:C17H27NO4
    Pureza:71.58% - 99.16%
    Cor e Forma:Soild
    Peso molecular:309.4
  • Bromchlorbuterol hydrochloride

    CAS:
    <p>Bromchlorbuterol HCl, a potent β-agonist, is used to study lung diseases like asthma.</p>
    Fórmula:C12H19BrCl2N2O
    Cor e Forma:Solid
    Peso molecular:358.1
  • MK-761 TFA


    <p>MK-761 TFA is an effective, orally active β2-adrenergic receptor blocker. It exhibits antihypertensive properties and positive inotropic effects, along with vasodilatory activity.</p>
    Fórmula:C15H20F3N3O4
    Cor e Forma:Solid
    Peso molecular:363.332
  • Vanilpyruvic acid

    CAS:
    <p>Vanillylpyruvic acid is a phenylpyruvic acid derivative applicable in biochemical experiments and drug synthesis research.</p>
    Fórmula:C10H10O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:210.18
  • 4-Hydroxypropranolol-d7 hydrochloride

    CAS:
    <p>Deuterium-labeled 4-Hydroxypropranolol HCl, a Propranolol metabolite that blocks β1/β2 receptors.</p>
    Fórmula:C16H22ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:318.85
  • Diacetolol D7

    CAS:
    <p>Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.</p>
    Fórmula:C16H24N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:315.42
  • Apraclonidine hydrochloride

    CAS:
    <p>Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.</p>
    Fórmula:C9H11Cl3N4
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:281.57
  • Benoxathian hydrochloride

    CAS:
    <p>Benoxathian hydrochloride is effective α 1 Adrenaline receptor antagonist. Benoxathian hydrochloride has value in the study of anorexia.</p>
    Fórmula:C19H24ClNO4S
    Cor e Forma:Solid
    Peso molecular:397.91
  • Nadolol-d9

    CAS:
    <p>Nadolol D9 is the deuterium labeled Nadolol is a blocker of non-selective beta.</p>
    Fórmula:C17H27NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:318.46
  • Clencyclohexerol-d10

    CAS:
    <p>Argipressin inhibits central corticotropin-releasing hormone. Argipressin acts as an inhibitory factor in the regulation of central CRH levels.</p>
    Fórmula:C14H20Cl2N2O2
    Cor e Forma:Solid
    Peso molecular:329.29
  • Zilpaterol-d7

    CAS:
    <p>Zilpaterol-d7 (trans-(±)-Zilpaterol-d7) is a deuterium-labeled version of Zilpaterol, a β-adrenergic receptor agonist.</p>
    Fórmula:C14H12D7N3O2
    Cor e Forma:Solid
    Peso molecular:268.36
  • Cimbuterol-d9

    CAS:
    <p>Cimbuterol-d9 is a deuterated compound of Cimbuterol.</p>
    Fórmula:C13H10D9N3O
    Pureza:99.22%
    Cor e Forma:Solid
    Peso molecular:242.37
  • 4-Hydroxyatomoxetine D3

    CAS:
    <p>4-Hydroxyatomoxetine D3, a deuterium variant, is Atomoxetine's active metabolite, metabolized by CYP2D6, an adrenergic reuptake blocker.</p>
    Fórmula:C17H21NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:274.37
  • Naphazoline nitrate

    CAS:
    <p>Naphazoline nitrate: α1-adrenergic agonist, induces autophagy, necrosis in cancer cells, inhibits differentiation, treats congestion and eye issues.</p>
    Fórmula:C14H15N3O3
    Pureza:98%
    Cor e Forma:White Crystalline Powder White Solid
    Peso molecular:273.29
  • Piribedil D8

    CAS:
    <p>Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.</p>
    Fórmula:C16H18N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:306.39
  • rac-Propranolol-d7

    CAS:
    <p>Rac-Propranolol-d7 is the deuterated form of Rac-Propranolol. Propranolol is a β-adrenergic receptor antagonist that inhibits β1AR.</p>
    Fórmula:C16H14D7NO2
    Cor e Forma:Solid
    Peso molecular:266.39
  • Ivabradine-d6 hydrochloride

    CAS:
    <p>Ivabradine HCl: novel If inhibitor, IC50 2.9 μM; lowers heart rate. Ivabradine D6 HCl is its deuterium variant.</p>
    Fórmula:C27H37ClN2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:511.08
  • (+)-Penbutolol

    CAS:
    <p>(+)-Penbutolol is an antagonist of β-adrenoceptor(IC50 of 0.74 μM). (+)-Penbutolol is an optical isomer of l-penbutolol with Na+ channel-blocking action.</p>
    Fórmula:C18H29NO2
    Cor e Forma:Solid
    Peso molecular:291.43
  • Brombuterol hydrochloride

    CAS:
    <p>Brombuterol is an agonist of the β2-adrenergic receptor (β2-AR).1It has been used as an illicit feed additive to increase the muscle-to-fat ratio of livestock.</p>
    Fórmula:C12H19Br2ClN2O
    Cor e Forma:Solid
    Peso molecular:402.56