
AChR
Os inibidores do receptor de acetilcolina (AChR) são compostos que bloqueiam a atividade dos receptores de acetilcolina, essenciais para a neurotransmissão nos sistemas nervosos central e periférico. Os AChRs desempenham um papel vital na contração muscular, memória e funções cognitivas. Os inibidores de AChRs são usados para estudar condições como miastenia gravis, doença de Alzheimer e outros distúrbios neurológicos. Ao modular a atividade dos AChRs, esses inibidores podem ajudar a desvendar as complexidades da sinalização colinérgica no cérebro. Na CymitQuimica, oferecemos uma gama de inibidores de AChRs para apoiar sua pesquisa em neurociência, farmacologia e doenças neurodegenerativas.
Foram encontrados 575 produtos de "AChR"
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Solifenacin succinate
CAS:<p>Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.</p>Fórmula:C23H26N2O2·C4H6O4Pureza:99.85% - 99.98%Cor e Forma:SolidPeso molecular:480.56Diphenmanil methylsulfate
CAS:<p>Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.</p>Fórmula:C20H24N·CH3O4SPureza:98% - 99.27%Cor e Forma:SolidPeso molecular:389.51Pirenzepine dihydrochloride
CAS:<p>Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.</p>Fórmula:C19H21N5O2·2HClPureza:99.48% - 99.62%Cor e Forma:White PowderPeso molecular:424.32Temephos
CAS:<p>Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.</p>Fórmula:C16H20O6P2S3Pureza:≥95%Cor e Forma:White Crystalline Solid Or LiquidPeso molecular:466.47Carbetapentane citrate
CAS:<p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>Fórmula:C20H31NO3·C6H8O7Pureza:99.46%Cor e Forma:White To Off-White SolidPeso molecular:525.59Zelminemab
CAS:<p>Zelminemab (AMG-301) is a human monoclonal antibody designed to target and inhibit the PACAP type I (PAC1) receptor [1].</p>Pureza:98.8% (SDS-PAGE); 97% (SEC-HPLC) - 98.8% (SDS-PAGE); 97% (SEC-HPLC)Cor e Forma:LiquidRivastigmine tartrate
CAS:<p>Rivastigmine (SDZ-ENA 713), a CNS-selective carbamate, treats dementia in Alzheimer's and Parkinson's.</p>Fórmula:C14H22N2O2·C4H6O6Pureza:98% - 99.66%Cor e Forma:White To Off-White PowderPeso molecular:400.43Dequalinium chloride
CAS:<p>Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.</p>Fórmula:C30H40Cl2N4Pureza:99.79% - 99.9%Cor e Forma:SolidPeso molecular:527.59Cotinine
CAS:<p>Cotinine (NIH-10498) is an alkaloid found in tobacco and is also the predominant metabolite of nicotine.</p>Fórmula:C10H12N2OPureza:98% - 99.89%Cor e Forma:Viscous Oil SolidPeso molecular:176.22MK-7622
CAS:<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Fórmula:C25H25N3O2Pureza:99.77% - 99.8%Cor e Forma:SolidPeso molecular:399.48Dicyclomine hydrochloride
CAS:<p>Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.</p>Fórmula:C19H36ClNO2Pureza:99.81%Cor e Forma:SolidPeso molecular:345.95Benactyzine hydrochloride
CAS:<p>Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.</p>Fórmula:C20H26ClNO3Pureza:99.03% - 99.94%Cor e Forma:SolidPeso molecular:363.88Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Fórmula:C21H25NO·CH4SO3Pureza:98.41% - 99.96%Cor e Forma:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecular:403.53Procainamide hydrochloride
CAS:<p>Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog</p>Fórmula:C13H21N3O·HClPureza:99.83% - 99.97%Cor e Forma:White To Slightly Yellow PowderPeso molecular:271.79VU 0365114
CAS:<p>VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).</p>Fórmula:C22H14F3NO3Pureza:99.86%Cor e Forma:SolidPeso molecular:397.35Fipexide
CAS:<p>Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983.</p>Fórmula:C20H21ClN2O4Pureza:97.6% - 99.95%Cor e Forma:SolidPeso molecular:388.84(Rac)-ABT-202 dihydrochloride
CAS:<p>(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.</p>Fórmula:C9H15Cl2N3Pureza:97.4%Cor e Forma:SolidPeso molecular:236.142Lysipressin acetate(50-57-7(fb_acetate))
CAS:<p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.</p>Fórmula:C48H69N13O14S2Pureza:98.08%Cor e Forma:SolidPeso molecular:1116.28Nebracetam hydrochloride
CAS:<p>Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.</p>Fórmula:C12H17ClN2OPureza:99.23%Cor e Forma:SolidPeso molecular:240.729nAChR agonist 1
CAS:<p>nAChR agonist 1 (DUN71755) is a brain-permeable and orally efficacious positive allosteric α7 nicotinic acetylcholine receptor (α7 nAChR)modulator.</p>Fórmula:C20H18ClNO3S2Pureza:97.59%Cor e Forma:SolidPeso molecular:419.94

