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PDGFR

PDGFR

Os inibidores do receptor do fator de crescimento derivado de plaquetas (PDGFR) são compostos que bloqueiam a sinalização do PDGFR, um receptor envolvido no crescimento celular, proliferação e angiogênese. O PDGFR desempenha um papel significativo no desenvolvimento dos vasos sanguíneos que alimentam os tumores. Inibir o PDGFR pode, portanto, impedir a angiogênese, tornando esses inibidores valiosos na terapia contra o câncer. Na CymitQuimica, oferecemos uma seleção de inibidores de PDGFR de alta qualidade para apoiar sua pesquisa em oncologia, biologia vascular e angiogênese.

Foram encontrados 127 produtos de "PDGFR"

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produtos por página.
  • TCS 359

    CAS:
    Fórmula:C18H20N2O4S
    Pureza:>98.0%(HPLC)
    Cor e Forma:Light yellow to Brown powder to crystal
    Peso molecular:360.43

    Ref: 3B-D5275

    25mg
    109,00€
    100mg
    328,00€
  • Sorafenib Tosylate

    CAS:
    Fórmula:C21H16ClF3N4O3·C7H8O3S
    Pureza:>98.0%(T)(HPLC)
    Cor e Forma:White to Light yellow powder to crystal
    Peso molecular:637.03

    Ref: 3B-N1229

    1g
    72,00€
  • Regorafenib

    CAS:
    Fórmula:C21H15ClF4N4O3
    Pureza:>98.0%(HPLC)
    Cor e Forma:White to Light yellow to Light orange powder to crystal
    Peso molecular:482.82

    Ref: 3B-R0142

    25mg
    81,00€
    100mg
    212,00€
  • Imatinib

    CAS:
    Fórmula:C29H31N7O
    Pureza:>98.0%(HPLC)
    Cor e Forma:White to Light yellow to Light orange powder to crystal
    Peso molecular:493.62

    Ref: 3B-I0906

    1g
    287,00€
    100mg
    54,00€
  • GW 2580

    CAS:
    Fórmula:C20H22N4O3
    Pureza:>98.0%(HPLC)
    Cor e Forma:White to Light yellow to Light orange powder to crystal
    Peso molecular:366.42

    Ref: 3B-G0504

    50mg
    82,00€
    250mg
    296,00€
  • Imatinib Mesylate

    CAS:
    Fórmula:C29H31N7O·CH4O3S
    Pureza:>98.0%(HPLC)
    Cor e Forma:White to Light yellow powder to crystal
    Peso molecular:589.72

    Ref: 3B-I0936

    1g
    213,00€
    100mg
    44,00€
  • Dasatinib

    CAS:
    Fórmula:C22H26ClN7O2S
    Pureza:>95.0%(T)(HPLC)
    Cor e Forma:White to Light yellow powder to crystal
    Peso molecular:488.01

    Ref: 3B-D5949

    1g
    84,00€
    5g
    238,00€
  • Sunitinib Malate

    CAS:
    Sunitinib Malate (Sunitinib) is an indolinone-based tyrosine kinase inhibitor.
    Fórmula:C26H33FN4O7
    Pureza:98% - 99.26%
    Cor e Forma:Solid
    Peso molecular:532.56

    Ref: TM-T0374

    1g
    105,00€
    25mg
    34,00€
    50mg
    42,00€
    100mg
    52,00€
    500mg
    82,00€
    1mL*10mM (DMSO)
    52,00€
  • AG 1295

    CAS:
    AG 1295 is a selective PDGFR tyrosine-kinase inhibitor; it blocks PDGFR autophosphorylation without affecting EGF receptor.
    Fórmula:C16H14N2
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:234.3

    Ref: TM-T14137

    5mg
    49,00€
    10mg
    84,00€
    25mg
    136,00€
    50mg
    222,00€
    100mg
    334,00€
    1mL*10mM (DMSO)
    54,00€
  • Olaratumab

    CAS:

    Olaratumab(IMC-3G3) is a human monoclonal IgG1 antibody against platelet-derived growth factor receptor alpha (PDGFRα), which has antitumor effects and can be

    Pureza:SDS-PAGE:95% SEC-HPLC:98.70%
    Cor e Forma:Liquid
    Peso molecular:147.12 kDa

    Ref: TM-T76761

    1mg
    235,00€
    5mg
    612,00€
    10mg
    938,00€
    25mg
    1.454,00€
    50mg
    1.882,00€
    100mg
    2.650,00€
  • N-Desmethyl imatinib

    CAS:
    N-Desmethyl imatinib (Imatinib metabolite N-Desmethyl imatinib) is a metabolite of Imatinib, which is a multi-target inhibitor of c-Kit, v-Abl, and PDGFR.
    Fórmula:C28H29N7O
    Pureza:98.60%
    Cor e Forma:Off-White To Pale-Yellow Solid
    Peso molecular:479.58

    Ref: TM-T11641

    1mg
    87,00€
    5mg
    166,00€
    10mg
    303,00€
    25mg
    512,00€
    50mg
    737,00€
    100mg
    1.018,00€
    1mL*10mM (DMSO)
    170,00€
  • Imatinib Mesylate

    CAS:

    Imatinib Mesylate (STI-571) is a tyrosine kinase receptor inhibitor with antineoplastic activity (IC50s: 0.6 μM, 0.1 μM and 0.1 μM for v-Abl, c-Kit and PDGFR,

    Fórmula:C29H31N7O·CH4SO3
    Pureza:98% - >99.99%
    Cor e Forma:White Crystalline Powder
    Peso molecular:589.71

    Ref: TM-T1621

    1u
    163,20€
    200mg
    59,00€
    500mg
    89,00€
  • Trapidil

    CAS:
    Trapidil (Avantrin) is a coronary vasodilator agent.
    Fórmula:C10H15N5
    Pureza:99.42%
    Cor e Forma:Solid
    Peso molecular:205.26

    Ref: TM-T0080

    25mg
    58,00€
    50mg
    96,00€
    100mg
    141,00€
    200mg
    200,00€
    1mL*10mM (DMSO)
    34,00€
  • Tyrphostin RG 13022

    CAS:
    Fórmula:C16H14N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:266.2946

    Ref: IN-DA009ATR

    10mg
    110,00€
    25mg
    155,00€
    100mg
    635,00€
    250mg
    A consultar
  • Sunitinib

    CAS:
    Sunitinib (SU 11248) is a multi-targeted receptor tyrosine kinase (RTK) inhibitor that inhibits VEGFR2 and PDGFRβ (IC50=80/2 nM).
    Fórmula:C22H27FN4O2
    Pureza:98% - 99.67%
    Cor e Forma:Yellow Solid
    Peso molecular:398.47

    Ref: TM-T0374L

    1g
    130,00€
    25mg
    34,00€
    50mg
    44,00€
    100mg
    55,00€
    500mg
    89,00€
    1mL*10mM (DMSO)
    44,00€
  • Ref: IN-DA00350H

    1g
    25,00€
    5g
    33,00€
    10g
    56,00€
    1kg
    506,00€
    25g
    61,00€
    5kg
    A consultar
    100g
    164,00€
    10kg
    A consultar
    500g
    687,00€
  • GW2580

    CAS:
    Fórmula:C20H22N4O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:366.4137

    Ref: IN-DA0036CW

    1g
    547,00€
    10mg
    61,00€
    25mg
    100,00€
    50mg
    120,00€
    100mg
    138,00€
    250mg
    177,00€
  • 2-(3,4-Dimethoxyphenylcarbamoyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide

    CAS:
    Fórmula:C18H20N2O4S
    Pureza:95%
    Cor e Forma:Solid
    Peso molecular:360.4274

    Ref: IN-DA003UHX

    10mg
    129,00€
    25mg
    135,00€
    100mg
    164,00€
    250mg
    200,00€
  • Regorafénib N-oxyde (M2)

    CAS:

    Regorafénib N-oxyde M2 is an active metabolite of Regorafenib.

    Fórmula:C21H15ClF4N4O4
    Pureza:98.03% - 98.26%
    Cor e Forma:Solid
    Peso molecular:498.81

    Ref: TM-T10157

    1mg
    44,00€
    2mg
    56,00€
    5mg
    80,00€
    10mg
    103,00€
    25mg
    180,00€
    50mg
    324,00€
    100mg
    472,00€
  • JNJ-10198409

    CAS:
    JNJ-10198409: selective ATP competitive PDGF-RTK inhibitor; IC50: PDGFR-β 4.2 nM, PDGFR-α 45 nM; antiangiogenic & antiproliferative.
    Fórmula:C18H16FN3O2
    Pureza:98.51%
    Cor e Forma:Solid
    Peso molecular:325.34

    Ref: TM-T15616

    1mg
    33,00€
    5mg
    92,00€
    10mg
    122,00€
    25mg
    198,00€
    50mg
    294,00€
    100mg
    419,00€
    200mg
    587,00€
    1mL*10mM (DMSO)
    92,00€