
Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 298 produtos de "Receptor opioide"
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ML138
CAS:<p>ML138 is a probe for MLPCN, an agonist of the κ opioid receptor.</p>Fórmula:C19H14Cl2N4OSCor e Forma:SolidPeso molecular:417.31Axomadol
CAS:<p>Axomadol (EN3324) is a centrally active analgesic compound. It has opioid agonistic properties and inhibitory effects on the reuptake of monoamines.</p>Fórmula:C16H25NO3Pureza:98%Cor e Forma:SolidPeso molecular:279.37Ici 174865
CAS:<p>Ici 174865 is a delta opioid receptor antagonist agent.</p>Fórmula:C38H53N5O7Cor e Forma:SolidPeso molecular:691.86Trimebutine CTB salt
CAS:<p>Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.</p>Fórmula:C29H36N2O8S2Pureza:99.85% - >99.99%Cor e Forma:SolidPeso molecular:604.74AT-121
CAS:<p>AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively).</p>Fórmula:C24H38N4O3SPureza:98.49% - 99.73%Cor e Forma:SolidPeso molecular:462.65ADL-5747
CAS:<p>ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletal</p>Fórmula:C24H28N2O3Pureza:98.94% - 99.74%Cor e Forma:SolidPeso molecular:392.49ICI 199,441 hydrochloride
CAS:<p>ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.</p>Fórmula:C21H25Cl3N2OPureza:99.57%Cor e Forma:SolidPeso molecular:427.8JNJ-20788560
CAS:<p>JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).</p>Fórmula:C25H28N2O2Pureza:98.02%Cor e Forma:SolidPeso molecular:388.5GR 89696 fumarate
CAS:<p>GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.</p>Fórmula:C23H29Cl2N3O7Pureza:99.84%Cor e Forma:SolidPeso molecular:530.4IPAG
CAS:<p>IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.</p>Fórmula:C17H22IN3Pureza:99.65%Cor e Forma:SolidPeso molecular:395.28ML-335
CAS:<p>ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief properties.</p>Fórmula:C25H32N2O3Pureza:98.52%Cor e Forma:SolidPeso molecular:408.53ICI 204,448
CAS:<p>ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.</p>Fórmula:C23H27Cl3N2O4Pureza:>99.99%Cor e Forma:SolidPeso molecular:501.83SCH-486757
CAS:<p>SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used in the study of cough.</p>Fórmula:C24H23Cl2N3OPureza:99.53% - >99.99%Cor e Forma:SolidPeso molecular:440.37NNC 63-0532
CAS:<p>NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.</p>Fórmula:C27H29N3O3Pureza:99.53%Cor e Forma:SolidPeso molecular:443.54Bevenopran
CAS:<p>Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies about the treatment of opioid-induced bowel dysfunction.</p>Fórmula:C20H26N4O4Pureza:98.69% - 98.9%Cor e Forma:SolidPeso molecular:386.44Naloxonazine dihydrochloride
CAS:<p>μ1 receptor antagonist</p>Fórmula:C38H43ClN4O6Pureza:98%Cor e Forma:SolidPeso molecular:687.22Prodilidine hydrochloride
CAS:Prodilidine hydrochloride is an opioid analgesic.Fórmula:C15H22ClNO2Cor e Forma:SolidPeso molecular:283.79μ opioid receptor agonist 1
CAS:<p>μ opioid receptor agonist 1 (Compound H-1a) is an optically pure oxyheterocyclic substituted pyrroloxypyrazole derivative and an MOR receptor agonist that can</p>Fórmula:C26H38N4OCor e Forma:SolidPeso molecular:422.61SNC 162
CAS:<p>SNC 162 is a potent and selective delta-opioid receptor (δ-opioid) agonist with analgesic, antidepressant and antiarrhythmic effects.</p>Fórmula:C27H37N3OPureza:98%Cor e Forma:SolidPeso molecular:419.6DPI-3290
CAS:<p>DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent</p>Fórmula:C30H34FN3O2Pureza:98%Cor e Forma:SolidPeso molecular:487.61
