
Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 298 produtos de "Receptor opioide"
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Viminol
CAS:<p>Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.</p>Fórmula:C21H31ClN2OPureza:98%Cor e Forma:SolidPeso molecular:362.94PF-4455242 HCl
CAS:<p>PF-4455242 HCl is a selective and orally available κ-opioid receptor antagonist that exhibiting antidepressant effects.</p>Fórmula:C21H29ClN2O2SPureza:99.59%Cor e Forma:SolidPeso molecular:408.99Opioid receptor modulator 1
CAS:<p>Opioid receptor modulator 1 is a modulator of opioid receptor.</p>Fórmula:C18H23NO2Pureza:98%Cor e Forma:SolidPeso molecular:285.38LY2444296
CAS:<p>LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 nM).</p>Fórmula:C24H22F2N2O2Pureza:99.18%Cor e Forma:SolidPeso molecular:408.44LY2048978
CAS:<p>LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.</p>Fórmula:C19H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:312.41μ opioid receptor agonist 2
CAS:μ opioid receptor agonist 2 (Compound H-3)is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases.Fórmula:C25H34N4OCor e Forma:SolidPeso molecular:406.56SCH 221510
CAS:<p>SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.</p>Fórmula:C28H31NOPureza:99.54%Cor e Forma:SolidPeso molecular:397.55JTC-801 free base
CAS:<p>JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).</p>Fórmula:C26H25N3O2Pureza:98%Cor e Forma:SolidPeso molecular:411.5TIPP
CAS:<p>TIPP is an agent of delta opioid antagonist.</p>Fórmula:C37H38N4O6Pureza:98%Cor e Forma:SolidPeso molecular:634.72ICI 154,129
CAS:<p>Selective δ opioid antagonist</p>Fórmula:C34H46N4O6SPureza:98%Cor e Forma:SolidPeso molecular:638.82AT-076
CAS:<p>AT-076: κ-opioid (Ki=1.14 nM) & nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) & δ-opioid (Ki=19.6 nM) competitive antagonist.</p>Fórmula:C26H35N3O3Cor e Forma:SolidPeso molecular:437.57AZD7268
CAS:<p>AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.</p>Fórmula:C29H30N4O2SCor e Forma:SolidPeso molecular:498.64ORL1 antagonist 1
CAS:<p>ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).</p>Fórmula:C20H22ClN5Pureza:98.92%Cor e Forma:SolidPeso molecular:367.88Norbinaltorphimine
CAS:<p>nor-Binaltorphimine dihydrochloride is a long-acting potent and highly selective kappa opioid receptor antagonist.</p>Fórmula:C40H43N3O6Cor e Forma:SolidPeso molecular:661.79Dup 747
CAS:<p>Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.</p>Fórmula:C24H28Cl2N2O2Pureza:98%Cor e Forma:SolidPeso molecular:447.4CR-665 Acetate
CAS:<p>CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.</p>Fórmula:C38H53N9O6Cor e Forma:SolidPeso molecular:731.899Loperamide oxide
CAS:<p>Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.</p>Fórmula:C29H33ClN2O3Cor e Forma:SolidPeso molecular:493.04Diallyl G
CAS:<p>Diallyl G is a delta-opioid receptor antagonist agent.</p>Fórmula:C38H53N5O8Cor e Forma:SolidPeso molecular:707.86DIPPA hydrochloride
CAS:<p>κ receptor antagonist</p>Fórmula:C22H24Cl3N3OSPureza:98%Cor e Forma:SolidPeso molecular:484.87σ1 Receptor/μ Opioid receptor modulator 1
CAS:<p>σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM).</p>Fórmula:C24H31FN2O2Cor e Forma:SolidPeso molecular:398.51
