Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 298 produtos de "Receptor opioide"
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Porcine dynorphin A(1-13) acetate
<p>Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like NMDA.</p>Fórmula:C77H130N24O17Pureza:99.14%Cor e Forma:SolidPeso molecular:1664Dynorphin B (1-13) acetate(83335-41-5 free base)
<p>Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.</p>Fórmula:C76H119N21O19Pureza:99.72%Cor e Forma:SolidPeso molecular:1630.89CTAP(TFA) (103429-32-9 free base)
<p>CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM.</p>Fórmula:C53H70F3N13O13S2Pureza:99.62%Cor e Forma:SolidPeso molecular:1218.33Nociceptin (1-13) amide TFA
<p>Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).</p>Fórmula:C63H101F3N22O17Pureza:97.64%Cor e Forma:SolidPeso molecular:1495.61Ac-RYYRIK-NH2 acetate
<p>Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.</p>Fórmula:C46H74N14O11Pureza:99.84%Cor e Forma:SolidPeso molecular:999.17[Met5]-Enkephalin, amide TFA
<p>[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.</p>Fórmula:C29H37F3N6O8SPureza:99.81%Cor e Forma:SolidPeso molecular:686.7Leuphasyl TFA
CAS:<p>Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.</p>Fórmula:C31H40F3N5O9Pureza:98.79%Cor e Forma:SolidPeso molecular:683.67Orphanin FQ(1-11) acetate(178249-41-7 free base)
<p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>Fórmula:C51H79N15O16Pureza:95.54%Cor e Forma:SolidPeso molecular:1158.26N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Fórmula:C30H39N5O8Pureza:>99.99%Cor e Forma:SolidPeso molecular:597.66b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Fórmula:C25H31N3O7Pureza:98.99%Cor e Forma:SolidPeso molecular:485.53Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Fórmula:C51H73N15O11Pureza:98.59%Cor e Forma:SolidPeso molecular:1072.22Hemorphin-7 acetate(152685-85-3 free base)
<p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>Fórmula:C51H68N12O13Pureza:99.66%Cor e Forma:SolidPeso molecular:1057.16Dynorphin A 1-10 acetate(79994-24-4 free base)
<p>Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.</p>Fórmula:C59H95N19O14Pureza:99.88%Cor e Forma:SolidPeso molecular:1294.53[Leu5]-Enkephalin, amide acetate
<p>[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.</p>Fórmula:C30H42N6O8Pureza:99.36%Cor e Forma:SolidPeso molecular:614.69Nociceptin (1-7) acetate
Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.Fórmula:C31H41N7O9Pureza:98.92%Cor e Forma:SoildPeso molecular:655.7AR-M 1000390 hydrochloride
CAS:<p>ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.</p>Fórmula:C23H29ClN2OPureza:98.66%Cor e Forma:SolidPeso molecular:384.94Bisacodyl
CAS:<p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>Fórmula:C22H19NO4Pureza:99.45% - 99.78%Cor e Forma:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderPeso molecular:361.39BRL 52537 hydrochloride
CAS:<p>BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.</p>Fórmula:C18H25Cl3N2OPureza:99.04%Cor e Forma:SolidPeso molecular:391.76Aticaprant
CAS:<p>Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.</p>Fórmula:C26H27FN2O2Pureza:99.53% - 99.93%Cor e Forma:SolidPeso molecular:418.5Deltorphin 2
CAS:<p>Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.</p>Fórmula:C38H54N8O10Pureza:>99.99%Cor e Forma:SolidPeso molecular:782.88
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