
Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 298 produtos de "Receptor opioide"
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BMS986188
CAS:<p>BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.</p>Fórmula:C30H31BrO4Pureza:98.76%Cor e Forma:SolidPeso molecular:535.47BW-180C
CAS:<p>BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.</p>Fórmula:C29H39N5O7Pureza:>99.99%Cor e Forma:SolidPeso molecular:569.65DAMGO TFA (78123-71-4(Free base))
<p>DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and quality-assured.</p>Fórmula:C28H36F3N5O8Pureza:98.67% - 99.76%Cor e Forma:SolidPeso molecular:627.6Asimadoline hydrochloride
CAS:<p>Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.</p>Fórmula:C27H31ClN2O2Pureza:98.94% - 99.32%Cor e Forma:SolidPeso molecular:451.01Endomorphin 1
CAS:Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).Fórmula:C34H38N6O5Pureza:95.92%Cor e Forma:Solid (Solid Powder )Peso molecular:610.7Salvinorin A
CAS:<p>Salvinorin A is a non-nitrogenous κ-opioid selective agonist.</p>Fórmula:C23H28O8Pureza:99.06%Cor e Forma:SolidPeso molecular:432.46GRT2932Q
CAS:<p>GRT2932Q is a nonpeptidic agonist of the opioid receptor-like 1 (ORL1) [1].</p>Fórmula:C25H26ClN3OCor e Forma:SolidPeso molecular:419.95BMS-986124
CAS:<p>BMS-986124 is an allosteric modulator of the μ-Opioid Receptor.</p>Fórmula:C16H15BrClNO3S2Cor e Forma:SolidPeso molecular:448.78DDD028
CAS:<p>DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.</p>Fórmula:C20H20N2Pureza:98%Cor e Forma:SolidPeso molecular:288.39GSK1521498
CAS:<p>GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).</p>Fórmula:C24H23F2N4O4PPureza:98%Cor e Forma:SolidPeso molecular:500.43LY 281217
CAS:<p>LY 281217, an organic opioid agonist, can produce analgesic effects in mice.</p>Fórmula:C32H42N4O6Pureza:98%Cor e Forma:SolidPeso molecular:578.7SR8993
CAS:<p>SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.</p>Fórmula:C25H37FN4Pureza:98%Cor e Forma:SolidPeso molecular:412.59ADL-5859 HCl
CAS:<p>ADL-5859 is a delta-opioid receptor agonist.</p>Fórmula:C24H28N2O3Pureza:98%Cor e Forma:SolidPeso molecular:392.49LY 164929
CAS:<p>LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.</p>Fórmula:C28H41N5O4Cor e Forma:SolidPeso molecular:511.66GSK1521498 free base
CAS:<p>GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.</p>Fórmula:C24H20F2N4Pureza:99.85%Cor e Forma:SolidPeso molecular:402.44ML 190
CAS:ML 190 is a potent and selective κ opioid receptor (KOR) antagonist (Ki=129 nM), exhibiting an IC50=150 nM in β-arrestin assays, drug addiction.Fórmula:C27H32N6O3Pureza:99.88%Cor e Forma:SolidPeso molecular:488.58BW 373U86
CAS:<p>BW373U86 (SNC86), a δ-opioid receptor agonist, demonstrates potent activity with an IC50 value of 1.49 nM and has shown to exhibit antidepressant-like effects [</p>Fórmula:C27H37N3O2Cor e Forma:SolidPeso molecular:435.6GSK1521498 free base (hydrochloride)
CAS:GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).Fórmula:C24H21ClF2N4Pureza:98%Cor e Forma:SolidPeso molecular:438.9Endomorphin 1 acetate
CAS:<p>Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.</p>Fórmula:C36H42N6O7Cor e Forma:SolidPeso molecular:670.75CP-866087
CAS:<p>CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.</p>Fórmula:C24H28N2O2Pureza:99.56% - >99.99%Cor e Forma:SoildPeso molecular:376.49
