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Receptor Glucagon

Receptor Glucagon

Os receptores de glucagon são GPCRs que mediam os efeitos do glucagon, um hormônio envolvido na regulação da homeostase da glicose, promovendo a quebra de glicogênio e a liberação de glicose pelo fígado. Esses receptores são críticos na gestão dos níveis de açúcar no sangue e são de particular interesse no estudo do diabetes e distúrbios metabólicos. Antagonistas dos receptores de glucagon estão sendo explorados como potenciais tratamentos para hiperglicemia no diabetes tipo 2. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores de glucagon de alta qualidade para apoiar sua pesquisa em endocrinologia, diabetes e regulação metabólica.

Foram encontrados 191 produtos de "Receptor Glucagon"

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produtos por página.
  • Retatrutide

    CAS:
    Retatrutide (LY3437943) is a triple agonist of GCGR, GIPR and GLP-1R that can be used to study obesity.
    Fórmula:C221H342N46O68
    Pureza:98.31%
    Cor e Forma:Solid
    Peso molecular:4732.09

    Ref: TM-T76279

    1mg
    222,00€
    5mg
    560,00€
    10mg
    898,00€
    25mg
    1.324,00€
    50mg
    1.791,00€
    100mg
    2.422,00€
  • Orforglipron

    CAS:
    Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1
    Fórmula:C48H48F2N10O5
    Pureza:99.47% - 99.8%
    Cor e Forma:Solid
    Peso molecular:882.96

    Ref: TM-T11408

    1mg
    54,00€
    5mg
    114,00€
    10mg
    177,00€
    25mg
    334,00€
    50mg
    467,00€
    100mg
    655,00€
    1mL*10mM (DMSO)
    44,00€
  • Avexitide acetate

    CAS:
    Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.
    Fórmula:C155H246N40O53S
    Pureza:96.64% - 98.65%
    Cor e Forma:Solid
    Peso molecular:3549.91

    Ref: TM-TP2100L

    1mg
    158,00€
    5mg
    444,00€
    10mg
    622,00€
    25mg
    964,00€
    50mg
    1.305,00€
    100mg
    1.755,00€
  • Glucagon (1-29), bovine, human, porcine hydrochloride

    CAS:
    Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. Glucagon increases HNF4α phosphorylation.
    Fórmula:C153H225N43O49S·ClH
    Pureza:95.65% - 98.03%
    Cor e Forma:Solid
    Peso molecular:3519.21

    Ref: TM-T15389L

    1mg
    66,00€
    5mg
    173,00€
    10mg
    260,00€
    25mg
    449,00€
    50mg
    657,00€
    100mg
    887,00€
    200mg
    1.198,00€
    250mg
    1.368,00€
  • PF-06882961

    CAS:
    PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
    Fórmula:C31H30FN5O4
    Pureza:97.19% - 99.56%
    Cor e Forma:Solid
    Peso molecular:555.6

    Ref: TM-T12431

    1mg
    47,00€
    5mg
    94,00€
    10mg
    147,00€
    25mg
    187,00€
    50mg
    240,00€
    100mg
    411,00€
    1mL*10mM (DMSO)
    103,00€
  • Retatrutide sodium salt


    Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.
    Pureza:99.97%
    Cor e Forma:Soild

    Ref: TM-T76279L1

    1mg
    235,00€
    5mg
    590,00€
    10mg
    948,00€
    25mg
    1.396,00€
    50mg
    1.890,00€
    100mg
    2.555,00€
  • Tirzepatide monosodium salt


    Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective activity and can be used to treat obesity.
    Fórmula:C225H347N48O68Na
    Pureza:99.69%
    Cor e Forma:Soild
    Peso molecular:4835.51

    Ref: TM-TP1111L1

    1mg
    236,00€
    5mg
    620,00€
    10mg
    1.018,00€
    25mg
    1.521,00€
    50mg
    2.088,00€
    100mg
    2.817,00€
  • VU0453379

    CAS:
    VU0453379 is a highly selective and central nervous system penetrant positive allosteric modulator of glucagon-like peptide-1R (EC50: 1.3 μM).
    Fórmula:C26H34N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:434.57

    Ref: TM-T17242

    2mg
    231,00€
  • GLP-1 receptor agonist 4

    CAS:
    GLP-1 receptor agonist 4 targets GLP-1R, EC50 64.5 nM, potential diabetes treatment research.
    Fórmula:C51H44Cl2N4O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:879.82

    Ref: TM-T11405

    100mg
    A consultar
    500mg
    A consultar
  • Glucagon-like peptide 1 (1-37), human

    CAS:
    Human GLP-1 (1-37) is a potent GLP-1 receptor agonist without impact on rat food intake or insulin secretion.
    Fórmula:C186H275N51O59
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:4169.48

    Ref: TM-TP1148

    1mg
    1.773,00€
  • GLP-1R Antagonist 1

    CAS:
    GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).
    Fórmula:C16H11ClF6N4O2
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:440.73

    Ref: TM-T15387

    1mg
    43,00€
    5mg
    93,00€
    10mg
    137,00€
    25mg
    259,00€
    50mg
    409,00€
    1mL*10mM (DMSO)
    90,00€
  • HAEGTFTSD

    CAS:
    HAEGTFTSD is GLP-1's initial segment; GLP-1 (7-36) amide, tied to food intake, stems from preproglucagon in L-cells.
    Fórmula:C40H57N11O17
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:963.94

    Ref: TM-TP1452

    1mg
    131,00€
    5mg
    394,00€
    10mg
    630,00€
  • Tirzepatide

    CAS:
    Tirzepatide (LY-3298176) is a dual glucose-dependent polypeptide (GIP) (EC50=0.042 nM) and glucagon-like peptide-1 (GLP-1) (EC50=0.086 nM) receptor agonist.
    Fórmula:C225H348N48O68
    Pureza:99.52% - 99.99%
    Cor e Forma:Solid
    Peso molecular:4813.45

    Ref: TM-TP1111

    1mg
    240,00€
    5mg
    628,00€
    10mg
    893,00€
    25mg
    1.324,00€
  • Cinnamtannin A2

    CAS:

    Cinnamtannin A2, a tetrameric procyanidin, boosts GLP-1, insulin, CRH expression, and has antioxidant, anti-diabetic, nephroprotective properties.

    Fórmula:C60H50O24
    Cor e Forma:Solid
    Peso molecular:1155.02

    Ref: TM-T40977

    1mg
    175,00€
    5mg
    449,00€
  • (S, R)-LSN 3318839

    CAS:
    (S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.
    Fórmula:C26H23Cl2N3O2
    Pureza:99.41%
    Cor e Forma:Soild
    Peso molecular:480.39

    Ref: TM-T63166L

    1mg
    175,00€
    5mg
    388,00€
    10mg
    572,00€
    25mg
    888,00€
    50mg
    1.224,00€
    100mg
    1.648,00€
  • Tirzepatide hydrochloride


    Tirzepatide HCl is a dual GIP and GLP-1 receptor agonist.
    Fórmula:C225H349N48O68Cl
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:4849.91

    Ref: TM-TP1110

    1mg
    240,00€
    5mg
    628,00€
  • GLP-1 moiety from Dulaglutide


    GLP-1 moiety from Dulaglutide is a 31-amino acid fragment of Dulaglutide which is a glucagon-like peptide 1 receptor (GLP-1) agonist.
    Fórmula:C149H221N37O49
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3314.62

    Ref: TM-TP1316

    1mg
    311,00€
    5mg
    989,00€
  • GLP-1 (9-36) amide

    CAS:
    GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.
    Fórmula:C140H214N36O43
    Pureza:97%
    Cor e Forma:Solid
    Peso molecular:3089.41

    Ref: TM-TP2252

    1mg
    84,00€
    5mg
    230,00€
    10mg
    340,00€
    25mg
    563,00€
    50mg
    795,00€
    100mg
    1.071,00€
  • V-0219 hydrochloride


    V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.

    Fórmula:C20H26ClF3N4O2
    Pureza:99.97%
    Cor e Forma:Soild
    Peso molecular:446.89

    Ref: TM-T60047L

    1mg
    38,00€
    5mg
    84,00€
    10mg
    128,00€
    25mg
    235,00€
    50mg
    350,00€
    100mg
    500,00€
    200mg
    672,00€
  • GLP-1 receptor agonist 13


    Compound (S)-9, a GLP-1 receptor agonist, exhibits an EC50 of 76 nM for the glucagon GLP-1 receptor [1].
    Fórmula:C25H23ClF2N6O
    Cor e Forma:Solid
    Peso molecular:496.94

    Ref: TM-T79348

    5mg
    A consultar
    50mg
    A consultar