HIV Protease
Os inibidores da protease do HIV são uma classe de medicamentos antirretrovirais que têm como alvo específico a enzima protease do vírus da imunodeficiência humana (HIV). Ao inibir esta enzima, esses compostos impedem o vírus de processar suas poliproteínas em proteínas maduras e funcionais, bloqueando assim a produção de novos virions infecciosos. Os inibidores da protease do HIV são um pilar da terapia antirretroviral altamente ativa (HAART) utilizada para o tratamento do HIV/AIDS. Na CymitQuimica, oferecemos uma variedade de inibidores da protease do HIV para apoiar sua pesquisa em tratamento do HIV, resistência a medicamentos e virologia.
Foram encontrados 507 produtos de "HIV Protease"
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Bz-RS-ISer(3-Ph)-Ome
CAS:<p>Bz-RS-ISer(3-Ph)-Ome (Methyl (2R,3S)-3-(benzoylamino)-2-hydroxy-3-phenylpropanoate) is a paclitaxel derivative that inhibits the HSV replication cycle.</p>Fórmula:C17H17NO4Pureza:99.36% - 99.89%Cor e Forma:White CrystalPeso molecular:299.32Saquinavir
CAS:<p>Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS.</p>Fórmula:C38H50N6O5Pureza:99.50% - >99.99%Cor e Forma:SolidPeso molecular:670.84LDC4297 hydrochloride
CAS:LDC4297 hydrochloride is a selective and potent CDK7 inhibitor with broad-spectrum antiviral activity, useful for research on viral infections.Fórmula:C23H29ClN8OCor e Forma:SolidPeso molecular:468.982,4-Dihydroxypyridine
CAS:2,4-Dihydroxypyridine: a pyridine derivative, chelates metals, assesses ion levels, measures enzymatic reactions, and quantifies biomolecules.Fórmula:C5H5NO2Pureza:97.79%Cor e Forma:White To Yellow-Beige Crystals OrPeso molecular:111.1Raltegravir potassium
CAS:Raltegravir potassium (MK 0518 potassium salt) salt(MK0518 potassium salt) is a potent integrase (IN) inhibitor, used to treat HIV infection.Fórmula:C20H20FN6O5·KPureza:98% - 99.55%Cor e Forma:Off-White SolidPeso molecular:482.51Dexelvucitabine
CAS:Dexelvucitabine (RVT), a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.Fórmula:C9H10FN3O3Pureza:98.25%Cor e Forma:SolidPeso molecular:227.19Rolipram
CAS:Rolipram (SB 95952) is a phosphodiesterase 4 inhibitor with antidepressant properties.Fórmula:C16H21NO3Pureza:99.22% - >99.99%Cor e Forma:SolidPeso molecular:275.34Dimercaprol
CAS:Dimercaprol (Dicaptol) is an anti-gas warfare agent that is effective against Lewisite (dichloro(2-chlorovinyl)arsine) and formerly known as British Anti-Fórmula:C3H8OS2Pureza:98.91% - 99.64%Cor e Forma:Viscous Oily LiquidPeso molecular:124.22Didanosine
CAS:Didanosine (ddI) is a nucleoside reverse transcriptase inhibitor analog of adenosine (IC50: 0.49 μM).Fórmula:C10H12N4O3Pureza:99.64%Cor e Forma:White Crystalline PowderPeso molecular:236.23Rilpivirine
CAS:Rilpivirine (R278474) is a diarylpyrimidine derivative and reverse transcriptase inhibitor with antiviral activity against HIV-1 that is used in the treatmentFórmula:C22H18N6Pureza:97.22% - 98.83%Cor e Forma:SolidPeso molecular:366.42RN-18
CAS:RN-18 is an inhibitor of HIV-1 viral infectivity factor (IC50: 6 μM in nonpermissive H9 cells).Fórmula:C20H16N2O4SPureza:97.21% - 98.39%Cor e Forma:SolidPeso molecular:380.42Fostemsavir
CAS:Fostemsavir (BMS-663068) is an HIV-1 attachment inhibitor in development for the treatment of HIV-1 infection.Fórmula:C25H26N7O8PPureza:98.95%Cor e Forma:SolidPeso molecular:583.49Obefazimod
CAS:<p>Obefazimod (ABX-464) is a potent anti-HIV agent. ABX464 inhibits HIV-1 replication in stimulated peripheral blood mononuclear cells (PBMCs).</p>Fórmula:C16H10ClF3N2OPureza:99.86%Cor e Forma:SolidPeso molecular:338.71Bictegravir
CAS:Bictegravir (GS-9883) is a potent inhibitor of HIV-1 integrase (IC50: 7.5 nM).Fórmula:C21H18F3N3O5Pureza:97.6% - 99.51%Cor e Forma:SolidPeso molecular:449.38IMB-301
CAS:IMB-301 is a small molecular inhibitor via virtual screening according to the hA3G model.Fórmula:C19H17Cl2FN2OPureza:99.72%Cor e Forma:SolidPeso molecular:379.26PMEDAP
CAS:PMEDAP is a potent inhibitor of Moloney murine sarcoma virus (MSV)-induced tumor formation and associated mortality and an inhibitor of human immunodeficiencyFórmula:C8H13N6O4PPureza:99.77%Cor e Forma:SolidPeso molecular:288.2Filgotinib
CAS:Filgotinib (GLPG0634) is a selective JAK1 inhibitor. The IC50 values against JAK1, JAK2, JAK3, and TYK2 are 10 nM, 28 nM, 810 nM, and 116 nM, respectively.Fórmula:C21H23N5O3SPureza:98.03% - ≥95%Cor e Forma:SolidPeso molecular:425.5Dolutegravir sodium
CAS:<p>Dolutegravir sodium (GSK-1349572A) salt(DTG; GSK1349572) is an HIV integrase inhibitor(IC50: 2.7 nM), modest activity against raltegravir-resistant signature</p>Fórmula:C20H18F2N3NaO5Pureza:98% - 99.46%Cor e Forma:SolidPeso molecular:441.36Filgotinib maleate
CAS:Filgotinib maleate, a selective oral JAK1 inhibitor, treats RA and Crohn's. IC50s: JAK1-10nM, JAK2-28nM, JAK3-810nM, TYK2-116nM.Fórmula:C25H27N5O7SCor e Forma:SolidPeso molecular:541.58Des(benzylpyridyl) Atazanavi
CAS:The N-dealkylated metabolite (M1) of Atazanavir, a HIV protease inhibitor.Fórmula:C26H43N5O7Pureza:98% - 99.75%Cor e Forma:SolidPeso molecular:537.65
