
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.797 produtos)
- Apoptose(6.275 produtos)
- Ciclo celular/Ponto de verificação(4.805 produtos)
- Cromatina/Epigenética(2.462 produtos)
- Sinalização Citoesquelética(1.534 produtos)
- Dano de DNA/Reparo de DNA(2.959 produtos)
- Endocrinologia/Hormónios(3.708 produtos)
- Enzima(3.670 produtos)
- GPCR/Proteína-G(9.020 produtos)
- Imunologia e Inflamação(3.884 produtos)
- Vírus da Influenza(301 produtos)
- Sinalização JAK/STAT(414 produtos)
- Sinalização MAPK(1.249 produtos)
- Transportador de Membranas/Canal Iónico(3.050 produtos)
- Metabolismo(10.206 produtos)
- Microbiologia/Virologia(7.612 produtos)
- Neurociência(10.379 produtos)
- Outros inibidores(36.012 produtos)
- Oxidação-Redução(42 produtos)
- Sinalização PI3K/Akt/mTOR(1.442 produtos)
- Proteases/Proteassoma(1.724 produtos)
- Células - tronco e Derivados(819 produtos)
- Tirosina Quinase/Adaptador(2.035 produtos)
- Ubiquitinação(1.718 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66683 produtos de "Inibidores"
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Unesbulin
CAS:<p>Unesbulin (PTC596) is an orally active and selective inhibitor of B-cell-specific Moloney murine leukemia virus integration site 1 (BMI-1).</p>Fórmula:C19H13F5N6Pureza:98.71%Cor e Forma:SolidPeso molecular:420.34DSP-2230
CAS:<p>DSP-2230 is a selective blocker of Nav1.7/Nav1.8.</p>Fórmula:C20H20F3N5O2Pureza:97.14%Cor e Forma:SolidPeso molecular:419.4DNA2 inhibitor C5
CAS:DNA2 inhibitor C5 is a specific cancer sensitizer with an IC50 of 20 μM, targeting multiple DNA2 activities.Fórmula:C10H6N2O5Pureza:99.05%Cor e Forma:SolidPeso molecular:234.16Ref: TM-T15146
1mg60,00€2mg85,00€5mg119,00€10mg188,00€25mg432,00€50mg638,00€100mg908,00€500mg1.825,00€1mL*10mM (DMSO)118,00€L-Ascorbic acid
CAS:L-Ascorbic acid (Vitamin C) is a natural product that is a potent reducing agent and antioxidant.Fórmula:C6H8O6Pureza:99.85% - 99.89%Cor e Forma:Crystals (Usually Plates Sometimes Needles Mon°Clinic System) Taste Almost Odorless (Ntp 1992)Peso molecular:176.12PIT
CAS:PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with an IC50 of 0.14 μM for human P2Y1.Fórmula:C20H16N2O5SPureza:98.63%Cor e Forma:SolidPeso molecular:396.425,6-Dihydro-5-methyluracil
CAS:<p>5,6-Dihydro-5-methyluracil (Dihydrothymine) is an intermediate breakdown product of thymine.</p>Fórmula:C5H8N2O2Pureza:98.53%Cor e Forma:SolidPeso molecular:128.13Agaric acid
CAS:<p>Agaricic acid is an adenine nucleotide translocase antagonist.It is obtained from various plants of the fungous tribe, i.e.</p>Fórmula:C22H40O7Pureza:98.99% - ≥98%Cor e Forma:SolidPeso molecular:416.55Thiamphenicol
CAS:Thiamphenicol (Dextrosulphenidol) is a methylsulfonyl analog of chloramphenicol. It is an antibiotic and immunosuppressive agent.Fórmula:C12H15Cl2NO5SPureza:99.08% - 99.8%Cor e Forma:Off-White SolidPeso molecular:356.22Samidorphan HCl
CAS:<p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>Fórmula:C21H27ClN2O4Pureza:96.79% - 97.85%Cor e Forma:SoildPeso molecular:406.9Folinic Acid Calcium Salt Pentahydrate
CAS:<p>Folinic Acid Calcium Salt Pentahydrate (Leucovorin Calcium Pentahydrate), a reduced folic acid, is used in combination with other chemotherapeutics.</p>Fórmula:C20H21CaN7O7·5H2OPureza:99.17% - >99.99%Cor e Forma:Yellowish-White To Yellow PowderPeso molecular:601.58ST-193
CAS:ST-193 blocks various arenaviruses (Guanarito, Junin, Lassa, Machupo) with IC50s: 0.44-3.1 nM.Fórmula:C24H25N3OPureza:99.52%Cor e Forma:SolidPeso molecular:371.47Ref: TM-T13006
1mg40,00€5mg90,00€10mg123,00€25mg213,00€50mg298,00€100mg419,00€200mg563,00€1mL*10mM (DMSO)89,00€Ziprasidone hydrochloride
CAS:Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychoticFórmula:C21H22CL2N4OSPureza:97.97% - 99.82%Cor e Forma:SolidPeso molecular:449.48-Hydroxyquinoline
CAS:8-Hydroxyquinoline (8-Quinolinol) is a heterocyclic phenol and derivative of quinoline with antiseptic, disinfectant, and pesticide properties.Fórmula:C9H7NOPureza:99.23%Cor e Forma:Solid CrystallinePeso molecular:145.16STAT3-IN-1
CAS:STAT3-IN-1 selective and orally active inhibitor of STAT3(in HT29 and MDA-MB 231 cells, with IC50 values of 1.82 μM and 2.14 μM , respectively), induces tumorFórmula:C28H29NO6Pureza:95.89% - 95.89%Cor e Forma:SolidPeso molecular:475.53Ref: TM-T13009
1mg60,00€2mg88,00€5mg131,00€10mg192,00€25mg349,00€50mg523,00€100mg753,00€500mg1.549,00€1mL*10mM (DMSO)137,00€6-Methoxy-2-naphthoic acid
CAS:6-Methoxy-2-naphthoic acid (6-Methoxy-2-naphthalenecarboxylic acid) is an modulator of NMDAR.Fórmula:C12H10O3Pureza:99.25%Cor e Forma:White To Off-White Powder Crystals Crystalline Powder And/Or ChunksPeso molecular:202.21Gimeracil
CAS:Gimeracil (Gimestat) is a competitive, reversible inhibitor of dihydropyrimidine dehydrogenase.Fórmula:C5H4ClNO2Pureza:99.80%Cor e Forma:SolidPeso molecular:145.54N-Caffeoyl O-methyltyramine
CAS:N-Caffeoyl O-methyltyramine is isolated from Cuscuta reflexa with strong inhibitory activity against α-glucosidase with IC50 of 103.58 μM.Fórmula:C18H19NO4Pureza:97.01%Cor e Forma:SolidPeso molecular:313.35Ref: TM-T12142
1mg49,00€5mg104,00€10mg160,00€25mg329,00€50mg487,00€100mg707,00€200mg938,00€1mL*10mM (DMSO)87,00€MK-7622
CAS:<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Fórmula:C25H25N3O2Pureza:99.77% - 99.8%Cor e Forma:SolidPeso molecular:399.48Granisetron hydrochloride
CAS:Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapyFórmula:C18H25ClN4OPureza:99.88% - 99.93%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:348.87(R)-Terazosin
CAS:R-Terazosin is the active R-enantiomer and potent α1-adrenoceptor antagonist (Ki: α1a 6.51 nM, α1b 1.01 nM, α1d 1.97 nM).Fórmula:C19H25N5O4Pureza:98.96% - 99.79%Cor e Forma:SolidPeso molecular:387.43Ref: TM-T12643
1mg44,00€2mg60,00€5mg90,00€10mg138,00€25mg227,00€50mg334,00€100mg469,00€500mgA consultar1mL*10mM (DMSO)100,00€Clobetasol propionate
CAS:Clobetasol propionate (CGP9555) exerts its effect by binding to cytoplasmic glucocorticoid receptors and subsequently activates glucocorticoid receptor-mediatedFórmula:C25H32ClFO5Pureza:99.41%Cor e Forma:White Crystalline PowderPeso molecular:466.97Lactose
CAS:Lactose is a disaccharide derived from galactose and glucose that is found in milk.Fórmula:C12H22O11Pureza:98% - 99.63%Cor e Forma:White Crystals Or PowderPeso molecular:342.30Captopril
CAS:Captopril (SA333) is a potent and specific inhibitor of peptidyl-dipeptidase A.Fórmula:C9H15NO3SPureza:98.34% - 99.85%Cor e Forma:White To Off-White Crystalline Powder SolidPeso molecular:217.29Acetohexamide
CAS:Acetohexamide (Acetohexamid) is an intermediate-acting, first-generation sulfonylurea with hypoglycemic activity.Fórmula:C15H20N2O4SPureza:99.19% - 99.85%Cor e Forma:Crystals From 90% Aq EthanolPeso molecular:324.402-(1-Piperazinyl)pyrimidine
CAS:2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.Fórmula:C8H12N4Pureza:98.46%Cor e Forma:Liquid - Crystal - LumpPeso molecular:164.21VU0359595
CAS:VU0359595 (ML-270) is a selective PLD1 inhibitor with 3.7 nM IC50; >1700x more selective over PLD2, for cancer/diabetes/neurodegenerative research.Fórmula:C25H29BrN4O2Pureza:99.79%Cor e Forma:SolidPeso molecular:497.434-Nonylphenol polyethoxylate
CAS:4-Nonylphenol polyethoxylate (Nonoxinol-9) is a typical surfactant used as a vaginal spermicide. Spermicides are locally acting non-hormonal contraceptives.Fórmula:(C2H4O)nC15H24OPureza:98%Cor e Forma:Compounds With N20 Are Pale-Yellow To Off-White Pastes Or Waxes Liquid LiquidPeso molecular:514.69Penicillin V Potassium
CAS:Penicillin V Potassium (Phenoxymethylpenicillin potassium salt) is a broad-spectrum penicillin antibiotic used orally in the treatment of infections.Fórmula:C16H17KN2O5SPureza:97.71%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:388.48Ac2-26 ammonium
Ac2-26 ammonium is an N-terminal derivative peptide of Annexin-A1 (AnxA1) with anti-inflammatory activity.Fórmula:C141H210N32O44S·xNH3Pureza:95.58%Cor e Forma:SolidPeso molecular:3089.43 (free base)Clindamycin phosphate
CAS:Clindamycin phosphate: a broad-spectrum chlorinated antibiotic, modified from lincomycin, used topically.Fórmula:C18H34ClN2O8PSPureza:98.15%Cor e Forma:White SolidPeso molecular:504.96Imazamox
CAS:Imazamox: a selective, safe, broad-spectrum systemic herbicide inhibiting ALS, stops plant growth, causing death.Fórmula:C15H19N3O4Pureza:97.07%Cor e Forma:SolidPeso molecular:305.33Rimonabant
CAS:Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Fórmula:C22H21Cl3N4OPureza:98% - 99.91%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:463.796-Iodopravadoline
CAS:6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.Fórmula:C23H25IN2O3Pureza:99.29%Cor e Forma:Off-White SolidPeso molecular:504.36Ref: TM-T14204
1mg38,00€2mg52,00€5mg70,00€10mg90,00€25mg198,00€50mg326,00€100mg520,00€1mL*10mM (DMSO)99,00€Tenalisib
CAS:Tenalisib (RP6530) (RP6530) is a potent and selective inhibitor of PI3Kδ and PI3Kγ(IC50 values of 25 and 33 nM, respectively.)Fórmula:C23H18FN5O2Pureza:99.71%Cor e Forma:SolidPeso molecular:415.42Ref: TM-T13119
1mg38,00€2mg49,00€5mg81,00€10mg111,00€25mg188,00€50mg304,00€100mg457,00€1mL*10mM (DMSO)88,00€Zoxazolamine
CAS:Zoxazolamine (NSC-24995) is a uricosuric and muscle relaxant.Fórmula:C7H5ClN2OPureza:99.54%Cor e Forma:Light Brown To Yellow-Brown PowderPeso molecular:168.58Aluminum Hydroxide
CAS:Aluminum Hydroxide: oral adjuvant, aids vaccine potency, enhances immune response.Fórmula:AlH3O3Pureza:98%Cor e Forma:White Solid PowderPeso molecular:78BRD6989
CAS:BRD6989, a cortistatin A analog, inhibits CDK8/19, enhances IL-10, and binds CDK8 with a 200 nM IC50.Fórmula:C16H16N4Pureza:99.43%Cor e Forma:SolidPeso molecular:264.33Ref: TM-T14778
1mg34,00€5mg66,00€10mg92,00€25mg177,00€50mg268,00€100mg398,00€200mg575,00€1mL*10mM (DMSO)73,00€Cloperastine hydrochloride
CAS:Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.Fórmula:C20H25Cl2NOPureza:97.74% - 99.42%Cor e Forma:SolidPeso molecular:366.334-Methylumbelliferone
CAS:4-Methylumbelliferone: coumarin derivative, used as spasmolytic, choleretic, light-protective agent, and to detect nitric acid.Fórmula:C10H8O3Pureza:97.32% - 97.70%Cor e Forma:Less Crystals Insoluble In Water (Ntp 1992) Physical Description Colorless Crystals Insoluble In Water (Ntp 1992)Peso molecular:176.17Olsalazine disodium
CAS:Olsalazine disodium (Dipentum) is bioconverted to 5-aminosalicylic acid (5-ASA) in the colon and has anti-inflammatory activity in ulcerative colitis.Fórmula:C14H8N2Na2O6Pureza:99.47% - 99.52%Cor e Forma:Yellow Crystalline PowderPeso molecular:346.2NE 10790
CAS:NE 10790, similar to risedronate, is a mild bone resorption inhibitor but poorly blocks FPP synthase.Fórmula:C8H10NO6PPureza:>99.99%Cor e Forma:SolidPeso molecular:247.14ZEN-3694
CAS:ZEN-3694 (ZEN 3694) is a bromo-structural domain extra-terminal inhibitor (BETi) with activity in androgen signaling inhibitor (ASI) resistance models and canFórmula:C19H19N5OPureza:98.94% - 99.76%Cor e Forma:SolidPeso molecular:333.39Entasobulin
CAS:Entasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity.Fórmula:C26H18ClN3O2Pureza:98.40%Cor e Forma:SolidPeso molecular:439.894-Fluoroanisole
CAS:4-Fluoroanisole is a intermediates in medicine, pesticide, liquid crystal materials.Fórmula:C7H7FOPureza:98.62%Cor e Forma:Less To Light Yellow Liquid Colorless To Light Yellow LiquidPeso molecular:126.13HLY78
CAS:HLY78, a Wnt/β-catenin activator, enhances Axin-LRP6 binding by targeting Axin's DIX domain.Fórmula:C17H17NO2Pureza:99.548%Cor e Forma:SolidPeso molecular:267.32Emeramide
CAS:Emeramide (BDTH2) is a thiol-redox antioxidant. It is also a heavy metal chelator.Fórmula:C12H16N2O2S2Pureza:98.73%Cor e Forma:SolidPeso molecular:284.4Ranolazine dihydrochloride
CAS:Ranolazine 2HCl, an antianginal, treats arrhythmia by inhibiting sodium current without changing blood pressure or heart rate.Fórmula:C24H35Cl2N3O4Pureza:99.30% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:500.46GR 103691
CAS:GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).Fórmula:C30H35N3O3Pureza:98.94% - 99.29%Cor e Forma:SolidPeso molecular:485.62Ref: TM-T11463
2mg42,00€5mg62,00€10mg97,00€25mg187,00€50mg305,00€100mg487,00€200mg692,00€1mL*10mM (DMSO)66,00€STL127705
CAS:STL127705 inhibits Ku 70/80 protein & DNA-PKCS kinase, IC50s: 3.5 μM & 2.5 μM.Fórmula:C22H20FN5O4Pureza:99.53% - 99.81%Cor e Forma:SolidPeso molecular:437.42Ref: TM-T13017
1mg73,00€5mg159,00€10mg230,00€25mg390,00€50mg582,00€100mg762,00€1mL*10mM (DMSO)178,00€Quinacrine dihydrochloride
CAS:Quinacrine dihydrochloride (Mepacrine dihydrochloride) is the dihydrochloride salt of the 9-aminoacridine derivative quinacrine with potential antineoplasticFórmula:C23H30CLN3O·2HClPureza:98.24% - 99.80%Cor e Forma:Yellow Crystals Or PowderPeso molecular:472.88

