
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.787 produtos)
- Apoptose(6.265 produtos)
- Ciclo celular/Ponto de verificação(4.800 produtos)
- Cromatina/Epigenética(2.446 produtos)
- Sinalização Citoesquelética(1.530 produtos)
- Dano de DNA/Reparo de DNA(2.964 produtos)
- Endocrinologia/Hormónios(3.708 produtos)
- Enzima(3.669 produtos)
- GPCR/Proteína-G(9.019 produtos)
- Imunologia e Inflamação(3.883 produtos)
- Vírus da Influenza(301 produtos)
- Sinalização JAK/STAT(414 produtos)
- Sinalização MAPK(1.248 produtos)
- Transportador de Membranas/Canal Iónico(3.038 produtos)
- Metabolismo(10.216 produtos)
- Microbiologia/Virologia(7.607 produtos)
- Neurociência(10.383 produtos)
- Outros inibidores(36.019 produtos)
- Oxidação-Redução(42 produtos)
- Sinalização PI3K/Akt/mTOR(1.442 produtos)
- Proteases/Proteassoma(1.726 produtos)
- Células - tronco e Derivados(823 produtos)
- Tirosina Quinase/Adaptador(2.039 produtos)
- Ubiquitinação(1.718 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66684 produtos de "Inibidores"
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Loxoprofen
CAS:Loxoprofen (Koloxo) is an anti-inflammatory non-steroidal medicine.Fórmula:C15H18O3Pureza:98.59%Cor e Forma:White To Yellowish Crystalline PowderPeso molecular:246.3Ethacridine lactate monohydrate
CAS:Ethacridine lactate hydrate is a topically applied anti-infective agent.Fórmula:C18H23N3O5Pureza:99.00%Cor e Forma:White PowderPeso molecular:361.4Dicoumarol
CAS:<p>Dicoumarol: an anticoagulant from moldy sweet-clover, depletes vitamin K, inhibits clotting enzymes.</p>Fórmula:C19H12O6Pureza:99.75% - 99.9%Cor e Forma:White Or Creamy White Crystalline Powder SolidPeso molecular:336.3Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Fórmula:C46H54N6O8S2Pureza:99.32% - >99.99%Cor e Forma:White Crystalline SolidPeso molecular:883.09Streptomycin sulfate
CAS:Streptomycin sulfate (Phytomycin) is a sulfate salt of streptomycin that is a protein synthesis inhibitor.Fórmula:C21H39N7O12H2SO4Pureza:99.84% - 99.86%Cor e Forma:White To Off-White PowderPeso molecular:728.68NI-42
CAS:NI-42, a BRPFs inhibitor: IC50(BRPF1/2/3)=7.9/48/260 nM, Kd(BRPF1/2/3)=40/210/940 nM; selective for class IV BRDs.Fórmula:C18H15N3O3SPureza:99.18%Cor e Forma:SolidPeso molecular:353.395-Azacytidine
CAS:5-Azacytidine (Ladakamycin) is a cytidine nucleoside analog, a DNA methylation inhibitor with specificity.Fórmula:C8H12N4O5Pureza:98% - 99.79%Cor e Forma:Crystals From Methanol Physical Description White Crystalline Powder (Ntp 1992)Peso molecular:244.2Mizolastine
CAS:Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.Fórmula:C24H25FN6OPureza:98% - 99.75%Cor e Forma:SolidPeso molecular:432.49Incyclinide
CAS:Incyclinide (COL-3) is a matrix metalloproteinase (MMP) inhibitor.Fórmula:C19H17NO7Pureza:97.99%Cor e Forma:SolidPeso molecular:371.34Ref: TM-T15574
1mg88,00€2mgA consultar5mg119,00€10mg188,00€25mg393,00€50mg605,00€100mg847,00€200mg1.159,00€1mL*10mM (DMSO)96,00€Sumatriptan succinate
CAS:Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.Fórmula:C18H27N3O6SPureza:97.53% - 99.51%Cor e Forma:White PowderPeso molecular:413.492',5'-Dideoxyadenosine
CAS:2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).Fórmula:C10H13N5O2Pureza:99.55%Cor e Forma:White SolidPeso molecular:235.24Ref: TM-T10066
1mg39,00€5mg84,00€10mg119,00€25mg210,00€50mg354,00€100mg562,00€500mg1.225,00€1mL*10mM (DMSO)92,00€Pramipexole
CAS:Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not acute liver injury.Fórmula:C10H17N3SPureza:98% - 99.96%Cor e Forma:SolidPeso molecular:211.33Ranitidine Hydrochloride
CAS:Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.Fórmula:C13H23ClN4O3SPureza:99.30% - 99.49%Cor e Forma:SolidPeso molecular:350.86Asaraldehyde
CAS:Asaraldehyde (2,4,5-trimethoxy-Benzaldehyde), a natural COX-2 inhibitor, exhibits 17-fold selectivity than COX-1.Fórmula:C10H12O4Pureza:99.74% - 99.85%Cor e Forma:Physical Description Beige Powder (Ntp 1992)Peso molecular:196.20Fmoc-NH-PEG8-NHS ester
CAS:Fmoc-NH-PEG8-NHS ester is a PEG-based PROTAC linker that can be used in PROTAC synthesis[1].Fórmula:C38H52N2O14Pureza:94.69%Cor e Forma:SolidPeso molecular:760.82Cloxiquine
CAS:Cloxiquine (Dermofongin) is a monohalogenated 8-hydroxyquinoline with activity against bacteria, fungi, and protozoa.Fórmula:C9H6ClNOPureza:99.82% - 99.87%Cor e Forma:Light Yellow CrystalsPeso molecular:179.6Fluorothyl
CAS:Fluorothyl (Bis(2,2,2-trifluoroethyl) ether) is a convulsant used in experimental animals.Fórmula:C4H4F6OPureza:98%Cor e Forma:Clear Colorless LiquidPeso molecular:182.06Sacituzumab
CAS:Sacituzumab is an IgG1 monoclonal antibody, a naked antibody to Sacituzumab govitecan, with potential anti-tumor activity for the study of tumors.Pureza:95% - >95.3% (SEC-HPLC); 96.7% (SDS-PAGE)Cor e Forma:LiquidPeso molecular:145.51 kDaRegorafénib N-oxyde (M2)
CAS:<p>Regorafénib N-oxyde M2 is an active metabolite of Regorafenib.</p>Fórmula:C21H15ClF4N4O4Pureza:98.03% - 98.26%Cor e Forma:SolidPeso molecular:498.81Otilonium bromide
CAS:Otilonium bromide (SP63) , an antimuscarinic, is utilized as a spasmolytic agent.Fórmula:C29H43BrN2O4Pureza:98.88% - 99.78%Cor e Forma:White PowerPeso molecular:563.57Cytidine
CAS:Cytidine (Cytosine-1-β-D-ribofuranoside) is a pyrimidine nucleoside comprised of a cytosine bound to ribose via a beta-N1-glycosidic bond.Fórmula:C9H13N3O5Pureza:98.80% - 99.63%Cor e Forma:Physical Description White Crystalline Powder (Ntp 1992)Peso molecular:243.22Org-26576
CAS:Org-26576 is a positive allosteric modulator of the AMPA receptor.Fórmula:C11H12N2O2Pureza:99.67%Cor e Forma:SolidPeso molecular:204.23Ref: TM-T16402
5mg47,00€10mg70,00€25mg104,00€50mg150,00€100mg256,00€200mg379,00€1mL*10mM (DMSO)50,00€ML-180
CAS:ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .Fórmula:C20H25ClN4O2Pureza:99.74%Cor e Forma:SolidPeso molecular:388.89Ref: TM-T12075
1mg35,00€2mg52,00€5mg77,00€10mg114,00€25mg207,00€50mg363,00€100mg550,00€1mL*10mM (DMSO)86,00€Doxylamine succinate
CAS:Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.Fórmula:C21H28N2O5Pureza:99.61%Cor e Forma:5 1 (Ntp 1992)Peso molecular:388.46Etodolac
CAS:Etodolac (AY-24236), a pyranocarboxylic NSAID, blocks COX-1/2, reducing pain, fever, inflammation, and inhibits platelet aggregation.Fórmula:C17H21NO3Pureza:99.78% - 99.92%Cor e Forma:Crystalline SolidPeso molecular:287.35Moclobemide
CAS:Moclobemide (Ro111163) is a reversible inhibitor of monoamine oxidase type A; (RIMA); (see MONOAMINE OXIDASE INHIBITORS) that has antidepressive properties.Fórmula:C13H17ClN2O2Pureza:99.51% - 99.59%Cor e Forma:White To Off-White SolidPeso molecular:268.74Itraconazole
CAS:Itraconazole (R51211) is a triazole antifungal agent that inhibits cytochrome P-450-dependent enzymes required for ERGOSTEROL synthesis.Fórmula:C35H38Cl2N8O4Pureza:98% - 99.90%Cor e Forma:Off-White Crystalline SolidPeso molecular:705.63BTRX-335140
CAS:<p>BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.</p>Fórmula:C25H32FN5O2Pureza:98% - 99.89%Cor e Forma:SolidPeso molecular:453.55Ref: TM-T14835
1mg105,00€2mg155,00€5mg250,00€10mg406,00€25mg840,00€50mg1.378,00€100mg1.882,00€200mg2.632,00€Alexidine dihydrochloride
CAS:Alexidine dihydrochloride: antifungal, antibiofilm, targets PTPMT1 for mitochondrial apoptosis, potential cancer treatment.Fórmula:C26H58Cl2N10Pureza:99.32% - 99.81%Cor e Forma:SolidPeso molecular:581.71meso-Erythritol
CAS:meso-Erythritol (Phycitol) is a four-carbon sugar that is found in algae, fungi, and lichens. Meso-Erythritol can be used as a coronary vasodilator.Fórmula:C4H10O4Pureza:99.84%Cor e Forma:Bipyramidal Tetragonal Prisms That Of SucrosePeso molecular:122.12Stachyose tetrahydrate
CAS:Stachyose tetrahydrate (D-Stachyose tetrahydrate) is a tetrasaccharide consisting of two α-D-galactose units, one α-D-glucose unit, and one β-D-fructose unitFórmula:C24H50O25Pureza:99.89%Cor e Forma:White To Off White Crystalline PowderPeso molecular:738.64BIX 02565
CAS:BIX 02565 is a potent inhibitor of ribosomal S6 kinase 2 (RSK2, IC50: 1.1 nM).Fórmula:C26H30N6O2Pureza:97.44% - 99.7%Cor e Forma:SolidPeso molecular:458.56Ref: TM-T5428
1mg56,00€2mg79,00€5mg118,00€10mg177,00€25mgA consultar50mgA consultar1mL*10mM (DMSO)145,00€C527
CAS:C527 is a is a pan DUB enzyme inhibitor. Which has a high potency for the USP1/UAF1 complex (IC50=0.88 μM).Fórmula:C17H8FNO3Pureza:97.22%Cor e Forma:SolidPeso molecular:293.25TDI-011536
CAS:TDI-011536: strong Lats kinase blocker, boosts heart cell growth, aids organ repair research.Fórmula:C19H16N4O2SPureza:98.70% - 99.83%Cor e Forma:SoildPeso molecular:364.42GANT 58
CAS:GANT 58 (NSC-75503) is a potent antagonist of Gli. Which inhibits GLI1-induced transcription (IC50: 5 μM).Fórmula:C24H16N4SPureza:99.53%Cor e Forma:SolidPeso molecular:392.48Zonisamide
CAS:Zonisamide (AD 810), a sulfonamide anticonvulsant, is approved for use as an adjunctive treatment in adults with partial-onset seizures.Fórmula:C8H8N2O3SPureza:99.05% - 99.9%Cor e Forma:Off-White PowderPeso molecular:212.23Abexinostat
CAS:Abexinostat (PCI-24781) is a pan-HDAC inhibitor, strongest on HDAC1; less so on HDACs 2, 3, 6, 10. Very select for HDAC8. In Phase 1/2 trials.Fórmula:C21H23N3O5Pureza:98.19% - 98.43%Cor e Forma:SolidPeso molecular:397.42Pepinh-TRIF TFA
Pepinh-TRIF TFA is a 30 aa peptide associated with the immune system that blocks TRIF signaling by interfering with TLR-TRIF interaction (TLR-TRIF interactionFórmula:C180H279F3N58O40S2Pureza:98%Cor e Forma:SolidPeso molecular:4014.09741Brilliant Yellow
CAS:Brilliant Yellow (Direct Yellow 4) is a potent and selective VGLUT inhibitor, a dye that is photodegradable.Fórmula:C26H18N4Na2O8S2Pureza:99.8% - 99.91%Cor e Forma:SolidPeso molecular:624.55Niraparib (R-enantiomer)
CAS:<p>Niraparib R-enantiomer (MK 4827 R-enantiomer) is an inhibitor of PARP1(IC50 of 2.4 nM).</p>Fórmula:C19H20N4OPureza:99.83%Cor e Forma:SolidPeso molecular:320.39Omeprazole sulfide
CAS:Omeprazole sulfide (Ufiprazole), a metabolite of Omeprazole, functions as a proton pump inhibitor.Fórmula:C17H19N3O2SPureza:98.83%Cor e Forma:White To Slightly Collored Solid Solid CrystallinePeso molecular:329.42PROTAC ERRα ligand 1
CAS:<p>PROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).</p>Fórmula:C19H11F3N2O4SPureza:99.45%Cor e Forma:SolidPeso molecular:420.36D-Arabinopyranose
CAS:D-(-)-Arabinose is a reducing sugar useful as a substrate in analysis of arabinose isomerases and synthesis of D-erythroascorbic acid in yeast.Fórmula:C5H10O5Pureza:99.81% - 99.91%Cor e Forma:White Crystalline Powder Crystalline PowderPeso molecular:150.13Dithranol
CAS:Dithranol (cignoline) is an anthracene derivative that disrupts MITOCHONDRIA function and structure and is used for the treatment of DERMATOSES, especiallyFórmula:C14H10O3Pureza:93.49% - 99.33%Cor e Forma:Physical Description Lemon Yellow Leaflets Or Plates Or An Orange Powder MeltingPeso molecular:226.23Hydrocortisone
CAS:Hydrocortisone is a synthetic glucocorticoid that aids in metabolism, immunity, and inflammation control.Fórmula:C21H30O5Pureza:98.4% - 99.95%Cor e Forma:Plates From Alc Or Iso-Propyl Alc SolidPeso molecular:362.46EMD57439
CAS:EMD57439 is a selective PDE-III inhibitor, showing no significant increase in c-AMP concentration and producing little change in Ca(50).Fórmula:C22H23N3O4SPureza:99.35% - 99.57%Cor e Forma:SolidPeso molecular:425.53,5-Diiodothyropropionic acid
CAS:3,5-Diiodothyropropionic acid: thyroid hormone analog, boosts α-myosin mRNA, binds TRα1 & TRβ1 (Ka: 2.40/M, 4.06/M).Fórmula:C15H12I2O4Pureza:98.42%Cor e Forma:SolidPeso molecular:510.06L-741626
CAS:L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3Fórmula:C20H21ClN2OPureza:98.57%Cor e Forma:SolidPeso molecular:340.85Diphylline
CAS:Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.Fórmula:C10H14N4O4Pureza:98.54%Cor e Forma:Crystals From Alcohol SolidPeso molecular:254.24G256 HCl
CAS:<p>G256 HCl has antiarrhythmic and anti-ischemic activity.</p>Fórmula:C14H16Cl3N5Pureza:>99.99% - >99.99%Cor e Forma:SoildPeso molecular:360.67
