
Inibidores
Subcategorias de "Inibidores"
- Angiogénese(2.805 produtos)
- Apoptose(6.292 produtos)
- Ciclo celular/Ponto de verificação(4.820 produtos)
- Cromatina/Epigenética(2.490 produtos)
- Sinalização Citoesquelética(1.544 produtos)
- Dano de DNA/Reparo de DNA(2.940 produtos)
- Endocrinologia/Hormónios(3.706 produtos)
- Enzima(3.670 produtos)
- GPCR/Proteína-G(9.024 produtos)
- Imunologia e Inflamação(3.902 produtos)
- Vírus da Influenza(302 produtos)
- Sinalização JAK/STAT(417 produtos)
- Sinalização MAPK(1.247 produtos)
- Transportador de Membranas/Canal Iónico(3.078 produtos)
- Metabolismo(10.178 produtos)
- Microbiologia/Virologia(7.618 produtos)
- Neurociência(10.367 produtos)
- Outros inibidores(35.951 produtos)
- Oxidação-Redução(41 produtos)
- Sinalização PI3K/Akt/mTOR(1.442 produtos)
- Proteases/Proteassoma(1.716 produtos)
- Células - tronco e Derivados(801 produtos)
- Tirosina Quinase/Adaptador(2.030 produtos)
- Ubiquitinação(1.722 produtos)
Foram encontrados 66630 produtos de "Inibidores"
Neohesperidin Dihydrochalcone
CAS:Neohesperidin Dihydrochalcone (Neohesperidin DC) is an artificial sweetener derived from citrus.Fórmula:C28H36O15Pureza:99.37% - 99.97%Cor e Forma:White To Off-White Solid Solid Particulate/PowderPeso molecular:612.58Narsoplimab
CAS:Narsoplimab (OMS 721) is an IgG4 monoclonal antibody that inhibits MASP-2, blocking the lectin pathway in adult stem cell transplant studies.
Pureza:SDS-PAGE:95% SEC-HPLC:98.56%Cor e Forma:LiquidPeso molecular:143.1 kDaRilzabrutinib
CAS:Rilzabrutinib (PRN1008) is a reversible covalent, selective and oral active inhibitor of Bruton’s Tyrosine Kinase (BTK)(IC50 of 1.3 nM).Fórmula:C36H40FN9O3Pureza:98.28% - 99.76%Cor e Forma:SolidPeso molecular:665.76Ref: TM-T12542
1mg99,00€5mg235,00€10mg376,00€25mg655,00€50mg944,00€100mg1.320,00€500mg2.642,00€1mL*10mM (DMSO)344,00€Dirithromycin
CAS:Dirithromycin (LY237216), a macrolide antibiotic, treats bacterial infections like bronchitis and pneumonia.Fórmula:C42H78N2O14Pureza:98% - 98.89%Cor e Forma:CrystalsPeso molecular:835.07Coumarin102
CAS:Coumarin102 (Exciton 480) is a fluorescent dye.Coumarin102 has weak inhibitory activity against Monoamine oxidase B, MAO-B and MAO-A and can be used to studyFórmula:C16H17NO2Pureza:98.4%Cor e Forma:SolidPeso molecular:255.31Dazolicin HCl
CAS:Dazolicin HCl (Dazolicine HCl) is an orally available antiarrhythmic compound.Fórmula:C17H25Cl2N3SPureza:98.83%Cor e Forma:SoildPeso molecular:374.37NVS-PAK1-1
CAS:NVS-PAK1-1 is an effective and selective allosteric PAK1 inhibitor (IC50: 5 nM).Fórmula:C23H25ClF3N5OPureza:99.35%Cor e Forma:SolidPeso molecular:479.93Miconazole
CAS:Miconazole (R18134) is an imidazole antifungal agent that is used topically and by intravenous infusion.Fórmula:C18H14Cl4N2OPureza:98% - 99.89%Cor e Forma:SolidPeso molecular:416.13Oxyclozanide
CAS:Oxyclozanide (Oxyclozanid) is a salicylanilide anthelmintic used in grazing animals for fasciola and cestode infestations.Fórmula:C13H6Cl5NO3Pureza:99.28%Cor e Forma:White To Yellowish PowderPeso molecular:401.46Tripelennamine hydrochloride
CAS:Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.Fórmula:C16H21N3·HClPureza:99.54% - 99.81%Cor e Forma:White SolidPeso molecular:291.82DUPA(OtBu)-OH
CAS:DUPA(OtBu)-OH, a DUPA precursor, targets PSMA with high affinity (Ki=8nM) to deliver Docetaxel for prostate cancer therapy.Fórmula:C23H40N2O9Pureza:97.29%Cor e Forma:SolidPeso molecular:488.57Ref: TM-T11122
2mg35,00€5mg52,00€10mg87,00€25mg130,00€50mg173,00€100mg248,00€200mg351,00€1mL*10mM (DMSO)57,00€Regorafénib N-oxyde (M2)
CAS:Regorafénib N-oxyde M2 is an active metabolite of Regorafenib.
Fórmula:C21H15ClF4N4O4Pureza:98.03% - 98.26%Cor e Forma:SolidPeso molecular:498.81Tubulin inhibitor 6
CAS:Tubulin inhibitor 6 (iHAP1) is an inhibitor of tubulin and a potent inhibitor of multiple cancer cell lines.Fórmula:C20H14ClNO2SPureza:99.05%Cor e Forma:SolidPeso molecular:367.85Captopril
CAS:Captopril (SA333) is a potent and specific inhibitor of peptidyl-dipeptidase A.Fórmula:C9H15NO3SPureza:98.34% - 99.85%Cor e Forma:White To Off-White Crystalline Powder SolidPeso molecular:217.29Phenformin hydrochloride
CAS:Phenformin hydrochloride (Phenformin HCl) is an agent belonging to the biguanide class of antidiabetics with antihyperglycemic activity.Fórmula:C10H16ClN5Pureza:97.11% - 99.80%Cor e Forma:Lactic AcidosisPeso molecular:241.72(R)-ADX-47273
CAS:(R)-ADX-47273 is a potent mGluR5 positive allosteric modulator(EC50 of 168 nM for potentiation ).
Fórmula:C20H17F2N3O2Pureza:99.87%Cor e Forma:SolidPeso molecular:369.36Vitamin B6
CAS:Vitamin B6 aids metabolism, especially for amino acids, and helps prevent pregnancy-induced and radiation sickness vomiting.Fórmula:C8H12NO6PPureza:97.81%Cor e Forma:PowderPeso molecular:249.15Opevesostat
CAS:Opevesostat (ODM-208) is an inhibitor of lyase (CYP11A1) (the enzyme cleavage cholesterol side chain).Fórmula:C21H26N2O5SPureza:99.67%Cor e Forma:SoildPeso molecular:418.51trans-C75
CAS:trans-C75 ((±)-C75) is an enantiomer of C75. C75 is an inhibitor of fatty-acid synthase (FASN).Fórmula:C14H22O4Pureza:98.88% - 99.57%Cor e Forma:White To Off-White SolidPeso molecular:254.32Ref: TM-T10656
1mg52,00€2mg69,00€5mg96,00€10mg160,00€25mg335,00€50mg537,00€100mg753,00€1mL*10mM (DMSO)108,00€Clorprenaline hydrochloride
CAS:Clorprenaline hydrochloride (Clorprenaline HCl) is a beta-2 adrenergic agonist with bronchodilator activity.Fórmula:C11H17Cl2NOPureza:99.59% - >99.99%Cor e Forma:SolidPeso molecular:250.165-Methyltetrahydrofolic acid
CAS:5-Methyl THF is a bioactive, dominant dietary folate and main blood/CSF form.Fórmula:C20H25N7O6Pureza:99.47%Cor e Forma:SolidPeso molecular:459.46DBCO-PEG4-NHS ester
CAS:DBCO-PEG4-NHS ester is a PEG-based PROTAC linker that can be used in PROTAC synthesis[1].Fórmula:C34H39N3O10Pureza:≥98%Cor e Forma:SolidPeso molecular:649.69GSTO1-IN-1
CAS:GSTO1-IN-1 is a potent glutathione S-transferase omega 1 inhibitor (GSTO1; IC50: 31 nM).Fórmula:C10H12Cl2N2O3SPureza:98.11% - 98.45%Cor e Forma:SolidPeso molecular:311.18Ref: TM-T11505
2mg35,00€5mg50,00€10mg80,00€25mg89,00€50mg105,00€100mg178,00€500mg437,00€1mL*10mM (DMSO)71,00€FSEN1
CAS:FSEN1 is a novel and highly effective non-competitive FSP1 inhibitor with an IC50 value of 313 nM.Fórmula:C22H22BrN5OSPureza:99.54% - 99.97%Cor e Forma:SolidPeso molecular:484.411-EBIO
CAS:1-EBIO (1-EBIO) is a calium channel agonist.Fórmula:C9H10N2OPureza:98.75%Cor e Forma:SolidPeso molecular:162.19Asaraldehyde
CAS:Asaraldehyde (2,4,5-trimethoxy-Benzaldehyde), a natural COX-2 inhibitor, exhibits 17-fold selectivity than COX-1.Fórmula:C10H12O4Pureza:99.74% - 99.85%Cor e Forma:Physical Description Beige Powder (Ntp 1992)Peso molecular:196.20NSP-805
CAS:NSP-805 is a potent and selective guinea pig cardiac phosphodiesterase 3 (PDE3) inhibitor.Fórmula:C17H19N3O2Pureza:99.85%Cor e Forma:SolidPeso molecular:297.35Ref: TM-T12267
1mg38,00€5mg86,00€10mg129,00€25mg216,00€50mg309,00€100mg427,00€200mg577,00€1mL*10mM (DMSO)94,00€AA147
CAS:AA147 is an ER proteostasis regulator that selectively activates the ATF6 arm of UPR as a prodrug.Fórmula:C16H17NO2Pureza:99.24%Cor e Forma:SolidPeso molecular:255.31Ref: TM-T14080
5mg63,00€10mg96,00€25mg178,00€50mg265,00€100mg395,00€500mg894,00€1mL*10mM (DMSO)69,00€MBQ-167
CAS:MBQ-167 is a dual inhibitor of Rac/Cdc42 (IC50s: 103 nM for Rac 1/2/3 and 78 nM for Cdc42 in MDA-MB-231 cells, respectively).Fórmula:C22H18N4Pureza:98.07% - 99.52%Cor e Forma:SolidPeso molecular:338.41Ref: TM-T16021
1mg37,00€2mg52,00€5mg79,00€10mg111,00€25mg208,00€50mg376,00€100mg567,00€1mL*10mM (DMSO)87,00€BI-671800
CAS:BI-671800 (AP-761) is a DP2/CRTH2 antagonist with IC50 values of 4.5 nM and 3.7 nM, potential for treating asthma.Fórmula:C25H26F3N5O3Pureza:99.19%Cor e Forma:SolidPeso molecular:501.5Ref: TM-T14565
1mg55,00€5mg124,00€10mg197,00€25mg353,00€50mg502,00€100mg680,00€200mg888,00€1mL*10mM (DMSO)137,00€Aminophylline
CAS:Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.
Fórmula:C7H8O2·C2H8N2Pureza:99.31%Cor e Forma:White Or Slightly Yellowish Granules Or Powder SolidPeso molecular:420.43CC-90003
CAS:CC-90003 is a selective inhibitor of ERK 1/2. It has antitumor activity.Fórmula:C22H21F3N6O2Pureza:99.42%Cor e Forma:SolidPeso molecular:458.44BI-1935
CAS:BI-1935 is an inhibitor of soluble epoxide hydrolase (sEH). For diseases related to cardiovascular disease.Fórmula:C24H21F3N6O3Pureza:97.55%Cor e Forma:SolidPeso molecular:498.46Ref: TM-T14557
1mg46,00€5mg94,00€10mg148,00€25mg259,00€50mg360,00€100mg465,00€200mg625,00€1mL*10mM (DMSO)103,00€Perphenazine
CAS:Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
Fórmula:C21H26ClN3OSPureza:99.3% - 99.99%Cor e Forma:SolidPeso molecular:403.97Procaine
CAS:Procaine (Vitamin H3) is a slow-acting ester local anesthetic with a short effect, used for infiltration, nerve, and spinal blocks.
Fórmula:C13H20N2O2Pureza:99.57% - 99.73%Cor e Forma:Anhydrous Plates Tables From Ligroin Or Ether SolidPeso molecular:236.31Lucitanib
CAS:Lucitanib (E-3810) is a VEGFR/FGFR inhibitor targeting VEGFR1-3 and FGFR1-2 with IC50s 7-82.5 nM.Fórmula:C26H25N3O4Pureza:96.13%Cor e Forma:SolidPeso molecular:443.49Ref: TM-T15185
1mg46,00€2mg59,00€5mg93,00€10mg137,00€25mg255,00€50mg462,00€100mg672,00€1mL*10mM (DMSO)90,00€MR-L2
CAS:MR-L2 is a reversible and noncompetitive allosteric activator of long-isoform phosphodiesterase-4 (PDE4).Fórmula:C19H16Cl3FN4OPureza:98.09% - 98.94%Cor e Forma:SolidPeso molecular:441.71Ref: TM-T12103
1mg145,00€2mg207,00€5mg354,00€10mg528,00€25mg852,00€50mg1.159,00€100mg1.568,00€500mg3.125,00€1mL*10mM (DMSO)378,00€4,4'-Iminodiphenol
CAS:4,4'-Iminodiphenol (Leucoindophenol) is an inactive estrogen receptor ligand with a diphenylamine backbone.Fórmula:C12H11NO2Pureza:98.68%Cor e Forma:SolidPeso molecular:201.22Cytidine
CAS:Cytidine (Cytosine-1-β-D-ribofuranoside) is a pyrimidine nucleoside comprised of a cytosine bound to ribose via a beta-N1-glycosidic bond.Fórmula:C9H13N3O5Pureza:98.80% - 99.63%Cor e Forma:Physical Description White Crystalline Powder (Ntp 1992)Peso molecular:243.22Oxaprozin
CAS:Oxaprozin (Oxaprozinum) is a Nonsteroidal Anti-inflammatory Drug.
Fórmula:C18H15NO3Pureza:98.53%Cor e Forma:SolidPeso molecular:293.32ML-180
CAS:ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .Fórmula:C20H25ClN4O2Pureza:99.74%Cor e Forma:SolidPeso molecular:388.89Ref: TM-T12075
1mg35,00€2mg52,00€5mg77,00€10mg114,00€25mg207,00€50mg363,00€100mg550,00€1mL*10mM (DMSO)86,00€Doxylamine succinate
CAS:Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.Fórmula:C21H28N2O5Pureza:99.61%Cor e Forma:5 1 (Ntp 1992)Peso molecular:388.46Moclobemide
CAS:Moclobemide (Ro111163) is a reversible inhibitor of monoamine oxidase type A; (RIMA); (see MONOAMINE OXIDASE INHIBITORS) that has antidepressive properties.Fórmula:C13H17ClN2O2Pureza:99.51% - 99.59%Cor e Forma:White To Off-White SolidPeso molecular:268.74Tegafur
CAS:Tegafur (FT 207) is a congener of the antimetabolite fluorouracil with antineoplastic activity.
Fórmula:C8H9FN2O3Pureza:99.16% - 99.89%Cor e Forma:White Crystalline PowderPeso molecular:200.17Inobrodib
CAS:Inobrodib (CBP-IN-1) is a potent inhibitor of p300/CBP bromodomain.Fórmula:C30H32F2N4O3Pureza:98.91% - 99.18%Cor e Forma:SolidPeso molecular:534.6Ref: TM-T10717
1mg70,00€2mg92,00€5mg153,00€10mg264,00€25mg557,00€50mg797,00€100mg1.074,00€1mL*10mM (DMSO)173,00€4-Nonylphenol polyethoxylate
CAS:4-Nonylphenol polyethoxylate (Nonoxinol-9) is a typical surfactant used as a vaginal spermicide. Spermicides are locally acting non-hormonal contraceptives.Fórmula:(C2H4O)nC15H24OPureza:98%Cor e Forma:Compounds With N20 Are Pale-Yellow To Off-White Pastes Or Waxes Liquid LiquidPeso molecular:514.69INH154
CAS:INH154 is a potent Nek2 and Hec1 binding (INH) inhibitor with IC50s of 120 nM in MB468 cells and 200 nM in Hela cells for INH.Fórmula:C22H24N4OSPureza:99.95%Cor e Forma:SolidPeso molecular:392.52Ref: TM-T11657
2mg34,00€5mg54,00€10mg82,00€25mg136,00€50mg203,00€100mg299,00€200mg416,00€1mL*10mM (DMSO)59,00€Iron(II) fumarate
CAS:Iron(II) fumarate (Iron Fumarate) is the iron(II) salt of fumaric acid, a reddish-orange powder, applied to supply iron intake.Fórmula:C4H2FeO4Pureza:98%Cor e Forma:Red To Brown PowderPeso molecular:169.9Articaine hydrochloride
CAS:Articaine hydrochloride (Hoe-045) is a thiophene-containing local anesthetic pharmacologically similar to MEPIVACAINE.Fórmula:C13H21ClN2O3SPureza:99.76%Cor e Forma:White Crystalline PowderPeso molecular:320.84Sultamicillin
CAS:Sultamicillin is an orally active double prodrug of Ampicillin/Sulbactan. Sulbactam is a semisynthetic β-Lactamase inhibitor.Fórmula:C25H30N4O9S2Pureza:99.34%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:594.66

