
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.519 produtos)
- Apoptose(5.787 produtos)
- Ciclo celular/Ponto de verificação(4.446 produtos)
- Cromatina/Epigenética(2.235 produtos)
- Sinalização Citoesquelética(1.381 produtos)
- Dano de DNA/Reparo de DNA(2.824 produtos)
- Endocrinologia/Hormónios(3.500 produtos)
- Enzima(3.639 produtos)
- GPCR/Proteína-G(8.317 produtos)
- Imunologia e Inflamação(3.516 produtos)
- Vírus da Influenza(296 produtos)
- Sinalização JAK/STAT(404 produtos)
- Sinalização MAPK(1.200 produtos)
- Transportador de Membranas/Canal Iónico(2.787 produtos)
- Metabolismo(9.416 produtos)
- Microbiologia/Virologia(6.968 produtos)
- Neurociência(9.919 produtos)
- Outros inibidores(37.928 produtos)
- Oxidação-Redução(41 produtos)
- Sinalização PI3K/Akt/mTOR(1.400 produtos)
- Proteases/Proteassoma(1.596 produtos)
- Células - tronco e Derivados(831 produtos)
- Tirosina Quinase/Adaptador(2.015 produtos)
- Ubiquitinação(1.649 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66626 produtos de "Inibidores"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Ciamexon
CAS:<p>Ciamexon: novel immunomodulator, shows promise in autoimmune models, low toxicity, may improve ophthalmic disease.</p>Fórmula:C11H13N3OPureza:99.71%Cor e Forma:SolidPeso molecular:203.24Lentinan
CAS:<p>Lentinan, isolated and purified from a hot water extract of Lentinula edodes fruit bodies, is a fungal polysaccharide immunomodulator with anti-tumor effects.</p>Fórmula:C42H72O36Cor e Forma:SolidPeso molecular:1153Ciprofloxacin
CAS:<p>Ciprofloxacin (Bay-09867) mainly targets bacterial DNA Gyrase (IC50=0.22-0.31 µM) and topoisomerase IV (IC50=0.3-1.9 µM). antibiotic. High-Quality, Low-Cost!</p>Fórmula:C17H18FN3O3Pureza:98.77% - 99.91%Cor e Forma:White PowderPeso molecular:331.34KukoaMine B
CAS:<p>Kukoamine B, as a constituent of Lycii Cortex, exhibits anti-acute inflammatory, anti-oxidant, and anti-diabetic characteristics.</p>Fórmula:C28H42N4O6Pureza:95% - 99.59%Cor e Forma:SolidPeso molecular:530.66Nufenoxole
CAS:<p>Nufenoxole is an orally active and antidiarrhoeal compound that inhibits fluid secretion in the human jejunum.</p>Fórmula:C25H29N3OPureza:98.84%Cor e Forma:SolidPeso molecular:387.52Oxolinic acid
CAS:<p>Oxolinic acid (Nidantin) is a synthetic antimicrobial related to NALIDIXIC ACID and used in URINARY TRACT INFECTIONS.</p>Fórmula:C13H11NO5Pureza:98.39% - 99.72%Cor e Forma:Crystals From Dimethylformamide White Crystalline PowderPeso molecular:261.23Lysipressin acetate(50-57-7(fb_acetate))
CAS:<p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.</p>Fórmula:C48H69N13O14S2Pureza:98.08%Cor e Forma:SolidPeso molecular:1116.28Tirbanibulin Mesylate
CAS:<p>Tirbanibulin Mesylate (KX01 Mesylate) is an inhibitor of Src that targets the peptide substrate site of Src (GI50: 9-60 nM in cancer cell lines).</p>Fórmula:C27H33N3O6SPureza:99%Cor e Forma:SolidPeso molecular:527.63Metaraminol tartrate
CAS:<p>Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>Fórmula:C13H19NO8Pureza:99.68%Cor e Forma:White PowderPeso molecular:317.29Reserpine
CAS:<p>Reserpine, an alkaloid from Rauwolfia roots, depletes neurotransmitters, used in treating hypertension and psychosis, but side effects restrict use.</p>Fórmula:C33H40N2O9Pureza:98.85% - 99.81%Cor e Forma:White Or Pale Buff To Slightly Yellowish Powder With A Bitter Taste (Ntp 1992)Peso molecular:608.68Aliskiren hemifumarate
CAS:<p>Aliskiren hemifumarate (CGP60536B) is an orally active nonpeptide renin inhibitor with antihypertensive activity.</p>Fórmula:C30H53N3O6C4H4O4Pureza:96.18% - 99.21%Cor e Forma:SolidPeso molecular:1219.6Ascorbyl palmitate
CAS:<p>Ascorbyl palmitate (L-Ascorbic acid 6-hexadecanoate), an ester formed from ascorbic acid and palmitic acid, produces a fat-soluble form of vitamin C.</p>Fórmula:C22H38O7Pureza:99.52%Cor e Forma:White Or Yellowish White Powder White Or Yellowish-White Powder With A Citrus-Like OdourPeso molecular:414.53MK-8719
CAS:<p>MK-8719 is a highly potent and selective inhibitor of O-GlcNAcase (OGA) (hOGA, Ki=7.9 nM) .</p>Fórmula:C9H14F2N2O3SPureza:99.67%Cor e Forma:SolidPeso molecular:268.28Deoxycholic acid
CAS:<p>Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate.</p>Fórmula:C24H40O4Pureza:99.91% - 99.91%Cor e Forma:Crystals From Alc SolidPeso molecular:392.57Promethazine
CAS:<p>Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .</p>Fórmula:C17H20N2SPureza:99.76%Cor e Forma:CrystalsPeso molecular:284.42(E/Z)-BCI
CAS:<p>(E/Z)-BCI (NSC-150117), a dual-specificity phosphatase 6 (DUSP6) inhibitor with anti-inflammatory properties, reduces LPS-induced inflammatory mediators and ROS</p>Fórmula:C22H23NOPureza:99.94%Cor e Forma:SolidPeso molecular:317.42Protamine sulfate
CAS:<p>Protamine sulfate: polycationic peptide, antiheparin, neutralizes anticoagulant effect, aids gene transfer.</p>Pureza:99.87%Cor e Forma:SolidNampt activator-1
CAS:<p>NAMPT Activator-1, EC50: 3.3-3.7 µM, specific niacinamide phosphotransferase stimulant, shields cells, potential neuroprotectant.</p>Fórmula:C16H17N3O3Pureza:99.84% - 99.98%Cor e Forma:SoildPeso molecular:299.32Mepiroxol
CAS:<p>Mepiroxol (Lysateril), an antihyperlipidemic, is also called 3-PYRIDINEMETHANOL N-OXIDE.</p>Fórmula:C6H7NO2Pureza:98.67%Cor e Forma:SolidPeso molecular:125.13trans-C75
CAS:<p>trans-C75 ((±)-C75) is an enantiomer of C75. C75 is an inhibitor of fatty-acid synthase (FASN).</p>Fórmula:C14H22O4Pureza:98.88% - 99.57%Cor e Forma:White To Off-White SolidPeso molecular:254.32Enoxacin
CAS:<p>Enoxacin (NSC-629661) is a broad-spectrum 6-fluoronaphthyridinone antibacterial agent (fluoroquinolones) structurally related to nalidixic acid.</p>Fórmula:C15H17FN4O3Pureza:98.68% - 99.89%Cor e Forma:Off-White To Yellow CrystalsPeso molecular:320.32Sodium citrate dihydrate
CAS:<p>Sodium citrate dihydrate (Trisodium citrate dihydrate) is an anticoagulant, and also used as a buffer and food preservatives.</p>Fórmula:C6H9Na3O9Pureza:≥98%Cor e Forma:Solid CrystallinePeso molecular:294.1Procodazole
CAS:<p>Procodazole (2-Benzimidazolepropionic acid) is a non-specific active immunoprotective agent against viral and bacterial infections.</p>Fórmula:C10H10N2O2Pureza:98% - 99.35%Cor e Forma:White To Tan Powder Crystals Or Crystalline Powder And/Or ChunksPeso molecular:190.2Moguisteine
CAS:<p>Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.</p>Fórmula:C16H21NO5SPureza:99.98%Cor e Forma:SolidPeso molecular:339.41T-0156
CAS:<p>T-0156 is a PEG5 inhibitor that inhibits the hydrolysis of cyclic guanosine monophosphate (cGMP) with low affinity for PDE6, PDE1, PDE2, PDE3 and PDE4.</p>Fórmula:C31H29N5O7Pureza:98.53% - 98.76%Cor e Forma:SoildPeso molecular:583.59Cyclamic acid
CAS:<p>Cyclamic acid, a synthetic sweetener (NSC-220327), often used as Na/Ca cyclamate. Banned in USA over disputed cancer risk.</p>Fórmula:C6H13NO3SPureza:98.42%Cor e Forma:White CrystalsPeso molecular:179.24Zileuton
CAS:<p>Zileuton (A 64077) inhibits 5-lipoxygenase, reduces leukotrienes, aids bronchodilation, lessens mucus/edema, and helps manage asthma symptoms.</p>Fórmula:C11H12N2O2SPureza:98.72% - 99.43%Cor e Forma:Crystalline SolidPeso molecular:236.29ZT 52656A hydrochloride
CAS:<p>ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.</p>Fórmula:C19H26ClF3N2OPureza:98.78%Cor e Forma:SolidPeso molecular:390.87Inobrodib
CAS:<p>Inobrodib (CBP-IN-1) is a potent inhibitor of p300/CBP bromodomain.</p>Fórmula:C30H32F2N4O3Pureza:98.91% - 99.18%Cor e Forma:SolidPeso molecular:534.6Articaine hydrochloride
CAS:<p>Articaine hydrochloride (Hoe-045) is a thiophene-containing local anesthetic pharmacologically similar to MEPIVACAINE.</p>Fórmula:C13H21ClN2O3SPureza:99.76%Cor e Forma:White Crystalline PowderPeso molecular:320.844-Nonylphenol polyethoxylate
CAS:<p>4-Nonylphenol polyethoxylate (Nonoxinol-9) is a typical surfactant used as a vaginal spermicide. Spermicides are locally acting non-hormonal contraceptives.</p>Fórmula:(C2H4O)nC15H24OPureza:98%Cor e Forma:Compounds With N20 Are Pale-Yellow To Off-White Pastes Or Waxes Liquid LiquidPeso molecular:514.69Niclosamide olamine
CAS:<p>Niclosamide olamine (Niclosamide Ethanolamine salt) is an Repellent, Insect Attractant and Chemosterilant.</p>Fórmula:C15H15Cl2N3O5Pureza:99.89%Cor e Forma:Bright Yellow Crystalline Physical Description Yellow Solid Insoluble In Water (Ntp 1992)Peso molecular:388.20Hydrocortisone
CAS:<p>Hydrocortisone is a synthetic glucocorticoid that aids in metabolism, immunity, and inflammation control.</p>Fórmula:C21H30O5Pureza:98.4% - 99.95%Cor e Forma:Plates From Alc Or Iso-Propyl Alc SolidPeso molecular:362.46Diaveridine
CAS:<p>Diaveridine (AI3-23935) (DVD) is a popular antibacterial synergist that is widely used in combination with sulfonamide.</p>Fórmula:C13H16N4O2Pureza:99.10%Cor e Forma:White SolidPeso molecular:260.29Orlistat
CAS:<p>Orlistat (Tetrahydrolipstatin) is a lipase inhibitor and a FASN inhibitor. Orlistat has been shown to promote weight loss. Cost effective and quality assured.</p>Fórmula:C29H53NO5Pureza:99.58% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:495.73Pseudobaptigenin
CAS:<p>Pseudobaptigenin (Psi-baptigenin) is an isoflavone, a flavonoid lipid molecule that is a natural product found in Pterocarpus marsupium, Dalbergia spruceana.</p>Fórmula:C16H10O5Pureza:98.61%Cor e Forma:SolidPeso molecular:282.25Diclofenac sodium
CAS:<p>Diclofenac sodium (GP 45840) is a non-steroidal anti-inflammatory agent (NSAID) with antipyretic and analgesic actions.</p>Fórmula:C14H10Cl2NNaO2Pureza:98.21% - 99.73%Cor e Forma:White Or Off-White PowderPeso molecular:318.13Capsaicin
CAS:<p>Capsaicin ((E)-Capsaicin) is a natural product extracted from Capsicum annuum, and is a TRPV1 agonist (EC50=0.29 μM).</p>Fórmula:C18H27NO3Pureza:98.24% - 99.88%Cor e Forma:Pure Dark Red Solid SolidPeso molecular:305.41Q-VD-OPH
CAS:<p>Q-VD-OPh is an irreversible caspase inhibitor with an IC50 value of 48 nM against caspase-7 and between 25 and 400 nM against caspase-1, 3, 8, 9, 10, 12.</p>Fórmula:C26H25F2N3O6Pureza:97.8% - 98.95%Cor e Forma:SolidPeso molecular:513.5Desbenzyl Donepezil Hydrochloride
CAS:<p>Desbenzyl Donepezil Hydrochloride is an impurity of Donepezil.</p>Fórmula:C17H24ClNO3Pureza:99.39%Cor e Forma:SolidPeso molecular:325.83Maltose monohydrate
CAS:<p>D-(+)-Maltose monohydrate (D-(+)-Maltose monohydrate), a dextrodisaccharide from starch and malt, is used as a fermentable intermediate and sweetening agent in</p>Fórmula:C12H2201·H2OPureza:98.41%Cor e Forma:PowderPeso molecular:360.31BRD4 Inhibitor-10
CAS:<p>BRD4 Inhibitor-10 is an inhibitor of BRD4-BD1 (IC50: 8 nM).</p>Fórmula:C25H27N5O2Pureza:99.53%Cor e Forma:SolidPeso molecular:429.51Icopezil
CAS:<p>Icopezil: small molecule, AChE inhibitor, treats neurological disorders, used in Alzheimer's research.</p>Fórmula:C23H25N3O2Pureza:99.35%Cor e Forma:SolidPeso molecular:375.46Citalopram hydrobromide
CAS:<p>Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal reuptake of serotonin, thereby</p>Fórmula:C20H22BrFN2OPureza:99.81%Cor e Forma:White Crystalline PowderPeso molecular:405.304BI-1935
CAS:<p>BI-1935 is an inhibitor of soluble epoxide hydrolase (sEH). For diseases related to cardiovascular disease.</p>Fórmula:C24H21F3N6O3Pureza:97.55%Cor e Forma:SolidPeso molecular:498.46α-Lipoic Acid
CAS:<p>α-Lipoic Acid, a sulfur-containing octanoic acid derivative, is biosynthesized from linoleic acid and used in dietary supplements.</p>Fórmula:C8H14O2S2Pureza:98.39% - 99.73%Cor e Forma:Forms Yellowish Flakes Light Yellow To Yellow PowderPeso molecular:206.33IK-930
CAS:<p>IK-930 is an orally active TEAD inhibitor (EC50 < 0.1 µM) with potent potency.</p>Fórmula:C19H19F3N4O2SPureza:99.89%Cor e Forma:SoildPeso molecular:424.44CHK1-IN-4 hydrochloride
<p>CHK1-IN-4 hydrochloride is a potent inhibitor of checkpoint kinase 1 (chk1).</p>Fórmula:C18H19BrClN7O2Pureza:99.29%Cor e Forma:SoildPeso molecular:480.75Aminophylline
CAS:<p>Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.</p>Fórmula:C7H8O2·C2H8N2Pureza:99.31%Cor e Forma:White Or Slightly Yellowish Granules Or Powder SolidPeso molecular:420.43Dansylamide
CAS:<p>Dansyl amide is a fluorescent dye used in biochemistry and chemistry to label substances with the fluorescent dansyl group.</p>Fórmula:C12H14N2O2SPureza:98.72%Cor e Forma:White To Light Yellow Fine Crystalline PowderPeso molecular:250.32
