
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.523 produtos)
- Apoptose(5.792 produtos)
- Ciclo celular/Ponto de verificação(4.449 produtos)
- Cromatina/Epigenética(2.238 produtos)
- Sinalização Citoesquelética(1.383 produtos)
- Dano de DNA/Reparo de DNA(2.825 produtos)
- Endocrinologia/Hormónios(3.507 produtos)
- Enzima(3.640 produtos)
- GPCR/Proteína-G(8.333 produtos)
- Imunologia e Inflamação(3.526 produtos)
- Vírus da Influenza(296 produtos)
- Sinalização JAK/STAT(404 produtos)
- Sinalização MAPK(1.202 produtos)
- Transportador de Membranas/Canal Iónico(2.790 produtos)
- Metabolismo(9.448 produtos)
- Microbiologia/Virologia(6.981 produtos)
- Neurociência(9.926 produtos)
- Outros inibidores(37.926 produtos)
- Oxidação-Redução(41 produtos)
- Sinalização PI3K/Akt/mTOR(1.400 produtos)
- Proteases/Proteassoma(1.597 produtos)
- Células - tronco e Derivados(831 produtos)
- Tirosina Quinase/Adaptador(2.016 produtos)
- Ubiquitinação(1.650 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66641 produtos de "Inibidores"
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Andromedoside
CAS:<p>Andromedoside is a useful organic compound for research related to life sciences. The catalog number is T124272 and the CAS number is 75044-72-3.</p>Fórmula:C25H28O13Cor e Forma:SolidPeso molecular:536.4865,7-Diacetoxyflavone
CAS:<p>5,7-Diacetoxyflavone is a natural product from Oroxylum indicum.</p>Fórmula:C19H14O6Pureza:98%Cor e Forma:SolidPeso molecular:338.313-Methoxy-9H-Carbazole
CAS:<p>3-methoxy-9H-carbazole: photosensitizer, anti-breast cancer, from Klauseneria spp., induces apoptosis.</p>Fórmula:C13H11NOPureza:99.24%Cor e Forma:SolidPeso molecular:197.23Anhydrotetracycline hydrochloride
CAS:<p>Anhydrotetracycline (hydrochloride) is a potent competitive inhibitor of broad-spectrum tetracycline destructase enzymes.</p>Fórmula:C22H23ClN2O7Pureza:98.90%Cor e Forma:SolidPeso molecular:462.88UFP-101 acetate
<p>UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.</p>Fórmula:C84H142N32O23Pureza:95.92%Cor e Forma:SolidPeso molecular:1968.23(-)-Holostyligone
CAS:<p>(-)-Holostyligone is a natural product</p>Fórmula:C21H24O5Pureza:98%Cor e Forma:SolidPeso molecular:356.41Sikokianin C
CAS:<p>Sikokianin C, a biflavonoid from Wikstroemia sikokiana, inhibits cystathionine β-synthase, showing anti-colon cancer potential.</p>Fórmula:C31H24O10Pureza:98%Cor e Forma:SolidPeso molecular:556.52MC-Val-Cit-PAB-duocarmycin chloride
CAS:<p>MC-Val-Cit-PAB-duocarmycin: ADC drug-linker with potent anticancer activity; duocarmycin-based, DNA-targeting.</p>Fórmula:C54H65ClN9O9Pureza:98%Cor e Forma:SolidPeso molecular:1019.6Amino-PEG23-amine
<p>Amino-PEG23-amine is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>Fórmula:C48H100N2O23Pureza:98%Cor e Forma:SolidPeso molecular:1073.31CDK ligand for PROTAC
<p>CDK ligand for PROTAC is a CDK inhibitor with antitumor activity. It has been used to design PROTAC CDK4/6 degraders.</p>Fórmula:C25H28F2N8OPureza:98%Cor e Forma:SolidPeso molecular:494.54HKSOX-1
CAS:<p>HKSOX-1 is a fluorescent probe for superoxide detection in live cells and in vivo, with high selectivity and sensitivity.</p>Fórmula:C23H6F10O11S2Cor e Forma:SolidPeso molecular:712.40Tacrine hydrochloride
CAS:<p>Tacrine: a cholinergic agonist, anticholinesterase; inhibits AChE/BChE with IC50s of 31/25.6 nM.</p>Fórmula:C13H15ClN2Pureza:98%Cor e Forma:SolidPeso molecular:234.73Saccharocarcin A
CAS:<p>Saccharocarcin A, an antibiotic from S. aerocolonigenes, combats various bacteria and inhibits C. trachomatis at 0.5 μg/ml, non-toxic to McCoy cells.</p>Fórmula:C67H101NO20Cor e Forma:SolidPeso molecular:1240.532Biotin-PEG24-acid
<p>Biotin-PEG24-acid is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>Fórmula:C61H117N3O28SPureza:98%Cor e Forma:SolidPeso molecular:1372.65Swietemahalactone
CAS:<p>Swietemahalactone exhibits antibacterial activity.</p>Fórmula:C27H30O10Pureza:98%Cor e Forma:SolidPeso molecular:514.527Aplanin
CAS:<p>Aplanin is an Oligosaccharide containing glucose as monomeric unit with an additional N-containing moiety.</p>Fórmula:C25H44O19Cor e Forma:SolidPeso molecular:648.61ent-Labda-8(17),13E-diene-3β,15,18-triol
CAS:<p>ent-Labda-8(17),13E-diene-3beta,15,18-triol is a natural product for research related to life sciences.</p>Fórmula:C20H34O3Pureza:98%Cor e Forma:SolidPeso molecular:322.48Acetanilide, 5'-amino-2'-(octyloxy)-
CAS:<p>Acetanilide, 5'-amino-2'-(octyloxy)- is a bioactive chemical.</p>Fórmula:C16H26N2O2Cor e Forma:SolidPeso molecular:278.39MC 1046
CAS:<p>MC 1046 is an impurity of Calcipotriol. Calcipotriol is a ligand of VDR-like receptors.</p>Fórmula:C27H38O3Pureza:98%Cor e Forma:SolidPeso molecular:410.59Girinimbine
CAS:<p>Girinimbine, a carbazole alkaloid from M. koenigii, exhibits antitumor, antioxidant, anti-inflammatory, antimicrobial effects.</p>Fórmula:C18H17NOPureza:99.23%Cor e Forma:SolidPeso molecular:263.33KuWal151
CAS:<p>CLK inhibitor effective on CLK4, 1, 2 (IC50: 28-510 nM), inactive on CLK3/DYRK/CDK/GSK3 (>10 μM), halts cancer cell growth in vitro.</p>Fórmula:C16H11ClN2OCor e Forma:SolidPeso molecular:282.72Cy5-PEG6-NHS ester
<p>Cy5-PEG6-NHS ester (chloride) is a PEG-based PROTAC linker utilized for PROTACs[1] synthesis.</p>Fórmula:C51H71ClN4O11Pureza:98%Cor e Forma:SolidPeso molecular:951.58Gimatecan HCl
<p>Gimatecan HCl (ST1481 HCL) is a potent topoisomerase I inhibitor. Gimatecan is an orally bioavailable camptothecin analogue with antitumor activity.</p>Fórmula:C25H26ClN3O5Pureza:97.04%Cor e Forma:SoildPeso molecular:483.94ent-11α,16α-Epoxy-15α-hydroxykauran-19-oic acid
CAS:<p>ent-11α,16α-Epoxy-15α-hydroxykauran-19-oic acid is a natural product for research related to life sciences.</p>Fórmula:C20H30O4Pureza:98%Cor e Forma:SolidPeso molecular:334.456Antibacterial agent 43
CAS:<p>Antibacterial agent 43 from patent WO2013030735A1 shows strong activity against infections and has research potential.</p>Fórmula:C12H11N4NaO7SCor e Forma:SolidPeso molecular:378.29Uvarigranol B
CAS:<p>Uvarigranol B is a natural product</p>Fórmula:C23H22O8Pureza:98%Cor e Forma:SolidPeso molecular:426.42RG 13647
CAS:<p>RG 13647 is an agonist of angiotensin II peptide.</p>Fórmula:C30H27N3O5Pureza:98%Cor e Forma:SolidPeso molecular:509.55iE-DAP
CAS:<p>iE-DAP is a biologically active peptide that functions as a NOD1 agonist.</p>Fórmula:C12H21N3O7Pureza:98%Cor e Forma:SolidPeso molecular:319.31N-Methyl-N'-(azido-PEG2-C5)-Cy5
<p>N-Methyl-N'-(azido-PEG2-C5)-Cy5 is an azide-functional PEG-based linker for PROTAC synthesis.</p>Fórmula:C38H51ClN6O3Pureza:98%Cor e Forma:SolidPeso molecular:675.3Imaprelimab
CAS:<p>Imaprelimab (PRX-003) is a humanized IgG1 κmonoclonal antibody against melanoma cell adhesion molecule (MCAM).</p>Pureza:> 95%Cor e Forma:LiquidPeso molecular:144.74 kDa6-Formyl-1,2,9,10-tetramethoxy-6a,7-dehydroaporphine
CAS:<p>6-Formyl-1,2,9,10-tetramethoxy-6a,7-dehydroaporphine is a natural product from Aconitum carmichaelii.</p>Fórmula:C21H21NO5Pureza:98%Cor e Forma:SolidPeso molecular:367.4p-Menth-8-ene-1,2-diol
CAS:<p>p-Menth-8-ene-1,2-diol is a natural product for research related to life sciences. The catalog number is TN4729 and the CAS number is 57457-97-3.</p>Fórmula:C10H18O2Pureza:98%Cor e Forma:SolidPeso molecular:170.257-Deoxyadriamycinol aglycone
CAS:<p>7-Deoxyadriamycinol aglycone is an adriamycin metabolite.</p>Fórmula:C21H20O8Cor e Forma:SolidPeso molecular:400.382: PN: US20040072744 SEQID: 2 claimed protein
CAS:<p>2: PN: US20040072744 SEQID: 2 claimed protein is a synthetic peptide, used for the research of Down' syndrome and schizophrenia.</p>Fórmula:C43H67N13O17SPureza:98%Cor e Forma:SolidPeso molecular:1070.132',3'-Dehydromarmesin
CAS:<p>2',3'-Dehydromarmesin is a useful organic compound for research related to life sciences and the catalog number is T125118.</p>Fórmula:C14H12O4Cor e Forma:SolidPeso molecular:244.25MAC-VC-PABC-ST7612AA1
<p>MAC-VC-PABC-ST7612AA1 is a part of antibody drug conjugates (ADCs) charged with HDAC inhibitor by a linker, shows antitumor activity[1].</p>Fórmula:C44H65N9O8SPureza:98%Cor e Forma:SolidPeso molecular:880.11ent-11α-Hydroxyabieta-8(14),13(15)-dien-16,12α-olide
CAS:<p>ent-11alpha-Hydroxyabieta-8(14),13(15)-dien-16,12alpha-olide is cytotoxic to ANA-1 and Jurkat cells; IC50: 7.12 & 17.9 nM.</p>Fórmula:C20H28O3Pureza:98%Cor e Forma:SolidPeso molecular:316.43(+)-Norlirioferine
CAS:<p>(+)-Norlirioferine is an alkaloid compound that exhibits cell growth inhibitory effects on macrophages and VERO cells.</p>Fórmula:C19H21NO4Cor e Forma:SolidPeso molecular:327.37Pseudohypericin
CAS:<p>Pseudohypericin has photocytotoxic, and antiretroviral activities, it has potential therapeutic value in diseases such as AIDS.</p>Fórmula:C30H16O9Pureza:98%Cor e Forma:SolidPeso molecular:520.44Laurycolactone B
CAS:<p>Laurycolactone B is a useful organic compound for research related to life sciences. The catalog number is T124085 and the CAS number is 85643-77-2.</p>Fórmula:C18H20O5Cor e Forma:SolidPeso molecular:316.353D-myo-Inositol-1,4,5,6-tetraphosphate (sodium salt)
CAS:<p>Ins(1,4,5,6)-P4, a signal-transducing inositol oligophosphate, increases 2-14x in cells post-Salmonella infection and modulates EGF signaling.</p>Fórmula:C6H12Na4O18P4Cor e Forma:SolidPeso molecular:588BACE1-IN-6
CAS:<p>BACE1-IN-6 is a BACE1 inhibitor with an IC 50 value of 1.5 nM.</p>Fórmula:C25H23F2N5O2SCor e Forma:SolidPeso molecular:495.55Mebeverine acid
CAS:<p>Mebeverine acid (Mebeverine metabolite Mebeverine acid) is a secondary metabolite of Mebeverine and can be used as a marker of oral exposure to Mebeverine.</p>Fórmula:C16H25NO3Pureza:99.66%Cor e Forma:SolidPeso molecular:279.37Dihydrocurcumenone
<p>Dihydrocurcumenone is a useful organic compound for research related to life sciences and the catalog number is T125888.</p>Fórmula:C15H24O2Cor e Forma:SolidPeso molecular:236.355PKCθ pseudosubstrate peptide inhibitor,myristoylated
<p>Myristoylated PKCθ pseudosubstrate peptide inhibitor is a synthetic peptide utilized to investigate the mechanism of action of protein kinase C theta (PKCθ) [1</p>Fórmula:C105H184N36O21SPureza:98%Cor e Forma:SolidPeso molecular:2318.88Mezerein
CAS:<p>Mezerein: antileukemic, activates PKC, inhibits yeast growth with PKC alpha, beta1, delta (IC50s: 1190, 908, 141 nM), not affecting PKC+ yeast.</p>Fórmula:C38H38O10Cor e Forma:White SolidPeso molecular:654.70m-Acetotoluidide, 4'-chloro-2-(diethylamino)-α,α,α-trifluoro-, hydrochloride
CAS:<p>m-Acetotoluidide, 4'-chloro-2-(diethylamino)-alpha,alpha,alpha-trifluoro-, hydrochloride is a bioactive chemical.</p>Fórmula:C13H17Cl2F3N2OCor e Forma:SolidPeso molecular:345.19KT5823
CAS:<p>KT5823 is a cGMP-dependent protein kinase (PKG) inhibitor that increases iodide ion uptake by regulating the expression of sodium iodide symporter protein.</p>Fórmula:C29H25N3O5Pureza:95%Cor e Forma:SolidPeso molecular:495.53m-PEG6-Tos
CAS:<p>m-PEG6-Tos is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>Fórmula:C20H34O9SPureza:98%Cor e Forma:SolidPeso molecular:450.54[12]-Dehydrogingerdione
CAS:<p>[12]-Dehydrogingerdione is a natural product found in ginger that has anti-neuroinflammatory activity.Cost-effective and quality-assured.</p>Fórmula:C23H34O4Pureza:98%Cor e Forma:SolidPeso molecular:374.51

