
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.519 produtos)
- Apoptose(5.787 produtos)
- Ciclo celular/Ponto de verificação(4.446 produtos)
- Cromatina/Epigenética(2.235 produtos)
- Sinalização Citoesquelética(1.381 produtos)
- Dano de DNA/Reparo de DNA(2.824 produtos)
- Endocrinologia/Hormónios(3.500 produtos)
- Enzima(3.639 produtos)
- GPCR/Proteína-G(8.318 produtos)
- Imunologia e Inflamação(3.516 produtos)
- Vírus da Influenza(296 produtos)
- Sinalização JAK/STAT(404 produtos)
- Sinalização MAPK(1.200 produtos)
- Transportador de Membranas/Canal Iónico(2.787 produtos)
- Metabolismo(9.416 produtos)
- Microbiologia/Virologia(6.968 produtos)
- Neurociência(9.920 produtos)
- Outros inibidores(37.928 produtos)
- Oxidação-Redução(41 produtos)
- Sinalização PI3K/Akt/mTOR(1.400 produtos)
- Proteases/Proteassoma(1.596 produtos)
- Células - tronco e Derivados(831 produtos)
- Tirosina Quinase/Adaptador(2.015 produtos)
- Ubiquitinação(1.649 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66627 produtos de "Inibidores"
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Opromazine hydrochloride
CAS:<p>Opromazine hydrochloride, a phenothiazine antipsychotic, blocks brain dopamine receptors to treat schizophrenia and psychosis.</p>Fórmula:C17H20Cl2N2OSPureza:98.03%Cor e Forma:SolidPeso molecular:371.32Diallyl Trisulfide
CAS:<p>Diallyl Trisulfide is an organic polysulfide compound found in garlic that acts as an H2S donor.</p>Fórmula:C6H10S3Pureza:95% - ≥98%Cor e Forma:LiquidPeso molecular:178.34MSX-127
CAS:<p>MSX-127 elicites positive response in peptide CXCR4.</p>Fórmula:C16H24N2O4Pureza:98.43%Cor e Forma:SolidPeso molecular:308.37MK 212 hydrochloride
CAS:<p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>Fórmula:C8H11ClN4·HClPureza:99.88%Cor e Forma:SolidPeso molecular:235.12Etretinate
CAS:<p>Etretinate (Ro 10-9359), an oral retinoid, treats psoriasis by promoting cell differentiation and reducing cell growth and inflammation.</p>Fórmula:C23H30O3Pureza:97.89%Cor e Forma:Crystals Crystalline SolidPeso molecular:354.48NNC-0640
CAS:<p>NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.</p>Fórmula:C29H31N7O4SPureza:97.04%Cor e Forma:SolidPeso molecular:573.67Fluorescein-5-maleimide
CAS:<p>Fluorescein-5-maleimide (N-(5-Fluoresceinyl)maleimide) is a fluorescent thiol-reactive dye (excitation: 494 nm, emission: 519 nm).</p>Fórmula:C24H13NO7Pureza:97% - 97.42%Cor e Forma:SolidPeso molecular:427.36orcinol
CAS:<p>orcinol (5-Methylresorcin) is anxiolytic agent without sedative effect.</p>Fórmula:C7H8O2Pureza:99.86%Cor e Forma:Pink-Grey To Pink-Brown Cryst Powder Or CrystalsPeso molecular:124.141,4-D-Gulonolactone
CAS:<p>1,4-D-Gulonolactone, precursor to vitamin C, is an enzyme substrate linked to oxidative stress and absent in scurvy-susceptible species.</p>Fórmula:C6H10O6Pureza:99.69%Cor e Forma:White Or Off-White Crystalline PowderPeso molecular:178.14Bimiralisib
CAS:<p>Bimiralisib (PI3K-IN-2) is an orally bioavailable pan inhibitor of PI3K and inhibitor of the mTOR, with potential antineoplastic activity.</p>Fórmula:C17H20F3N7O2Pureza:97.58% - 98.92%Cor e Forma:SolidPeso molecular:411.38Lasiodonin
CAS:<p>Lasiodonin is a natural product isolated from the leaves of Isodon parvifolius.</p>Fórmula:C20H28O6Pureza:93.00%Cor e Forma:SolidPeso molecular:364.43GW 405833
CAS:<p>GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selective</p>Fórmula:C23H24Cl2N2O3Pureza:99.82% - 99.93%Cor e Forma:SolidPeso molecular:447.35L-Hyoscyamine sulfate
CAS:<p>L-Hyoscyamine sulfate (Levsin Sulfate) is a belladonna alkaloid derivative and the levorotatory form of racemic atropine which exhibits anticholinergic effect.</p>Fórmula:C34H48N2O10SPureza:96.7% - 99.61%Cor e Forma:Long Orthorhombic Prisms From Acetone SolidPeso molecular:676.8(-)-α-Terpineol
CAS:<p>(-)-α-Terpineol has antitumour, anti-inflammatory, and antimicrobial activities, it inhibits tumour cells growth through inhibition of the NF-κB pathway.</p>Fórmula:C10H18OPureza:99.85%Cor e Forma:Liquid Clear Colorless LiquidPeso molecular:154.25Phosphorylcholine chloride calcium salt tetrahydrate
CAS:<p>Phosphocholine chloride Ca salt tetrahydrate: found in many organisms; elevated in human liver tumors; precursor in glycine/serine metabolism.</p>Fórmula:C5H21CaClNO8PPureza:99.95%Cor e Forma:White PowderPeso molecular:329.73DUB-IN-2
CAS:<p>Dub-in-2, with an IC50 value of 0.28 for USP8, is an effective deubiquitinase inhibitor.</p>Fórmula:C15H9N5OPureza:98.96%Cor e Forma:SolidPeso molecular:275.26Tetradehydrothalictrifoline
CAS:<p>Tetradehydrothalictrifoline is a nature product.</p>Fórmula:C21H20NO4Pureza:99.26%Cor e Forma:SolidPeso molecular:350.39Oxalic acid dihydrate
CAS:<p>Oxalic acid dihydrate is a plant-derived strong dicarboxylic acid, excreted in urine, used as a reagent and reducing agent.</p>Fórmula:C2H6O6Pureza:98.04% - 99.39%Cor e Forma:White Solid CrystallinePeso molecular:126.07Thalidomide-propargyl
CAS:<p>Thalidomide-propargyl, a Cereblon ligand, links proteins in PROTAC formation.</p>Fórmula:C16H12N2O5Pureza:95.14%Cor e Forma:SolidPeso molecular:312.28Skp2 Inhibitor C1
CAS:<p>Skp2 Inhibitor C1 (SKPin C1)(SKPin C1) is a specific small molecule inhibitor of Skp2-mediated p27 degradation.</p>Fórmula:C18H13BrN2O4S2Pureza:97.36%Cor e Forma:SolidPeso molecular:465.34JMJD7-IN-1
CAS:<p>JMJD7-IN-1 (Benzoic acid, 2,4-dichloro-, 5-nitro-8-quinolinyl ester) is a potent JMJD7 inhibitor, with an IC50 of 6.62 μM.</p>Fórmula:C16H8Cl2N2O4Pureza:99.66%Cor e Forma:SolidPeso molecular:363.15H3B-5942
CAS:<p>H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).</p>Fórmula:C31H34N4O2Pureza:99.21% - ≥95%Cor e Forma:SolidPeso molecular:494.63Ethyl linoleate
CAS:<p>Ethyl linoleate is a natural product and can inhibit the expression of inflammatory mediators and the development of atherosclerotic lesions.</p>Fórmula:C20H36O2Pureza:97.24% - 99.69%Cor e Forma:Pale Yellow LiquidPeso molecular:308.50Boc-NH-PEG3
CAS:<p>Boc-NH-PEG3 (PROTAC Linker 10) is a PEG derivative containing a hydroxyl group and Boc-protected amino group, and is a PROTAC linker.</p>Fórmula:C11H23NO5Pureza:≥95%Cor e Forma:SolidPeso molecular:249.3Levomefolate calcium
CAS:<p>Levomefolate calcium is an artificial form of folate. It is a coenzymated form of folic acid and a more bioavailable alternative in dietary supplements.</p>Fórmula:C20H23CaN7O6Pureza:97.35%Cor e Forma:Off-White To Pale Yellow SolidPeso molecular:497.52Mesaconine
CAS:<p>Mesaconine is an ingredient from Aconitum carmichaelii Debx..</p>Fórmula:C24H39NO9Pureza:98%Cor e Forma:SolidPeso molecular:485.573PO
CAS:<p>3PO inhibits PFKFB3 (IC50: 22.9 µM) and cancer cell growth (IC50: 1.4-24 µM), reducing glucose uptake and key cellular metabolites.</p>Fórmula:C13H10N2OPureza:99.56% - 99.67%Cor e Forma:SolidPeso molecular:210.23VPC-13163
CAS:<p>VPC-13566 inhibits growth in LNCaP, Enzalutamide-resistant MR49F, lowers AR gene, PSA, TMPRSS2 expression, but not in AR-independent PC3 cells.</p>Fórmula:C16H14N2Pureza:98.02%Cor e Forma:SolidPeso molecular:234.3Eurycomanol 2-O-β-D-glucopyranoside
CAS:<p>Eurycomanol 2-O-β-D-glucopyranoside is a natural compound belonging to the class of diterpenoids, extracted from Tongkat Ali.</p>Fórmula:C26H36O14Pureza:99.79%Cor e Forma:SolidPeso molecular:572.56Toosendanin
CAS:<p>Toosendanin is hepatotoxic, inhibits HL-6 cell growth, induces apoptosis, and is an insecticide for Ae.</p>Fórmula:C30H38O11Pureza:98% - ≥98%Cor e Forma:White Crystalline PowderPeso molecular:574.62Padmatin
CAS:<p>Padmatin (Blumeatin C) is a component of the heartwood of Prunus puddum.</p>Fórmula:C16H14O7Pureza:98.46% - 99.82%Cor e Forma:SolidPeso molecular:318.28PNU-120596
CAS:<p>PNU-120596 (NSC-216666) is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.</p>Fórmula:C13H14ClN3O4Pureza:99.82%Cor e Forma:SolidPeso molecular:311.72methyl 5-(3,4-dimethoxyphenyl)isoxazole-3-carboxylate
CAS:<p>methyl 5-(3,4-dimethoxyphenyl)isoxazole-3-carboxylate is a biochemical.</p>Fórmula:C13H13NO5Pureza:97.69%Cor e Forma:SolidPeso molecular:263.25Bimatoprost
CAS:<p>Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular</p>Fórmula:C25H37NO4Pureza:98% - >99.99%Cor e Forma:Crystalline SolidPeso molecular:415.57Alisertib
CAS:<p>Alisertib (MLN 8237) is a specific Aurora A inhibitor (IC50: 1.2 nM). The selectivity of Alisertib(MLN 8237) is >200-fold higher for Aurora A than Aurora B.</p>Fórmula:C27H20ClFN4O4Pureza:98.31% - >99.99%Cor e Forma:SolidPeso molecular:518.92VU0155094
CAS:<p>VU0155094 (ML 397) is a positive allosteric modulator with differential activity at the various group III mGluRs.</p>Fórmula:C24H24N2O4SPureza:97.21%Cor e Forma:SolidPeso molecular:436.52Poziotinib
CAS:<p>Poziotinib (NOV120101)(NOV120101; HM781-36B) is an irreversible HER1/2/4 inhibitor (IC50s: 3/5/23 nM).</p>Fórmula:C23H21Cl2FN4O3Pureza:98.69% - 99.78%Cor e Forma:SolidPeso molecular:491.34(E/Z)-Zotiraciclib citrate
<p>(E/Z)-Zotiraciclib ((E/Z)-TG02) citrate is a potent inhibitor of CDK2, JAK2 and FLT3 and can be used in cancer research.</p>Fórmula:C29H32N4O8Cor e Forma:SolidPeso molecular:564.59Rucaparib Phosphate
CAS:<p>Rucaparib Phosphate (PF-01367338 phosphate) is an inhibitor of PARP that is used in clinical therapy to sensitize cancer cells to chemotherapy.</p>Fórmula:C19H18FN3O·H3PO4Pureza:99.37%Cor e Forma:SolidPeso molecular:421.36Tiagabine hydrochloride
CAS:<p>Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.</p>Fórmula:C20H25NO2S2·HClPureza:99.09% - 99.77%Cor e Forma:White To Off-White SolidPeso molecular:412.01B2
CAS:<p>B2 (Linazolamide intermediate B impurity 2) promotes inclusion formation in cellular models of Huntington's disease and Parkinson's disease</p>Fórmula:C20H17ClN4O3Pureza:99.66%Cor e Forma:SolidPeso molecular:396.83Cannabidivarin
CAS:<p>Cannabidivarin (GWP42006) inhibits GABAA receptors, potentially controlling childhood absence epilepsy.</p>Fórmula:C19H26O2Pureza:98.06% - 98.51%Cor e Forma:SolidPeso molecular:286.41Fosfluconazole
CAS:<p>Fosfluconazole is water-soluble phosphate prodrug of fluconazole. Fluconazole is an antifungal drug.</p>Fórmula:C13H13F2N6O4PPureza:99.12%Cor e Forma:SolidPeso molecular:386.25D-(-)-Mandelic acid
CAS:<p>D-(-)-Mandelic acid ((R)-(-)-Mandelic acid) has the function of killing sperm, inhibiting bacteria, anti-inflammation and enhancing vagina self-cleaning.</p>Fórmula:C8H8O3Pureza:97.15%Cor e Forma:White CrystalsPeso molecular:152.15GSK1379725A
CAS:<p>GSK1379725A is a selective BPTF ligand (Kd = 2.8 μM).</p>Fórmula:C23H23FN6O3Pureza:99.51%Cor e Forma:SolidPeso molecular:450.47Omadacycline HCl
CAS:<p>Omadacycline, a first-class aminomethylcycline, treats pneumonia and skin infections including MRSA, and overcomes tetracycline resistance.</p>Fórmula:C29H41ClN4O7Cor e Forma:SolidPeso molecular:593.118Aldicarb sulfone
CAS:<p>Aldicarb sulfone is a cholinesterase inhibitor .</p>Fórmula:C7H14N2O4SPureza:99.05%Cor e Forma:Aldicarb Sulfone Is A White Crystalline Solid InsecticidePeso molecular:222.265'-N-Ethylcarboxamidoadenosine
CAS:<p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>Fórmula:C12H16N6O4Pureza:98.95% - ≥95%Cor e Forma:PowderPeso molecular:308.29Tideglusib
CAS:<p>Tideglusib (NP031112), a non-ATP competitive inhibitor of glycogen synthase kinase 3 (GSK-3), is with anti-inflammatory and neuroprotective activities.</p>Fórmula:C19H14N2O2SPureza:98.40% - 99.35%Cor e Forma:SolidPeso molecular:334.39Heparan Sulfate
CAS:<p>Heparan sulfate is a natural product, a linear polysaccharide. Heparan sulfate occurs as a proteoglycan (HSPG). Cost effective and quality assured.</p>Fórmula:C12H19NO20S3(monomer)Pureza:98%Cor e Forma:SolidPeso molecular:593.47(monomer)

