
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.523 produtos)
- Apoptose(5.792 produtos)
- Ciclo celular/Ponto de verificação(4.449 produtos)
- Cromatina/Epigenética(2.238 produtos)
- Sinalização Citoesquelética(1.383 produtos)
- Dano de DNA/Reparo de DNA(2.825 produtos)
- Endocrinologia/Hormónios(3.507 produtos)
- Enzima(3.640 produtos)
- GPCR/Proteína-G(8.333 produtos)
- Imunologia e Inflamação(3.526 produtos)
- Vírus da Influenza(296 produtos)
- Sinalização JAK/STAT(404 produtos)
- Sinalização MAPK(1.202 produtos)
- Transportador de Membranas/Canal Iónico(2.790 produtos)
- Metabolismo(9.448 produtos)
- Microbiologia/Virologia(6.981 produtos)
- Neurociência(9.926 produtos)
- Outros inibidores(37.926 produtos)
- Oxidação-Redução(41 produtos)
- Sinalização PI3K/Akt/mTOR(1.400 produtos)
- Proteases/Proteassoma(1.597 produtos)
- Células - tronco e Derivados(831 produtos)
- Tirosina Quinase/Adaptador(2.016 produtos)
- Ubiquitinação(1.650 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66641 produtos de "Inibidores"
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[Sar9,Met(O2)11]-Substance P acetate
<p>[Sar9,Met(O2)11]-Substance P acetate is an NK1 agonist, raising MAP and HR equally to septide but with unique timing and behaviors.</p>Fórmula:C66H106N18O18SPureza:>99.99%Cor e Forma:SolidPeso molecular:1471.75DHBP
CAS:<p>DHBP (Benzoresorcinol) is an WalKR TCS activator.</p>Fórmula:C13H10O3Pureza:99.95%Cor e Forma:Light-Yellow Solid CrystallinePeso molecular:214.22Methyl 2,6-dichlorobenzoate
CAS:<p>Methyl 2,6-dichlorobenzoate (2,6-Dichlorobenzoic acid methyl ester), a biochemical compound, is used for proteomics research.</p>Fórmula:C8H6Cl2O2Pureza:99.03%Cor e Forma:SolidPeso molecular:205.04SKLB-163
CAS:<p>SKLB-163 acts by downregulating RhoGDI, activating JNK-1 signaling pathway and caspase-3, and reducing phosphorylated Akt and p44/42 MAPK.</p>Fórmula:C18H16ClN3O2S2Pureza:99.23%Cor e Forma:SolidPeso molecular:405.92Histamine Phosphate
CAS:<p>Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.</p>Fórmula:C5H9N·2H3O4PPureza:>99.99%Cor e Forma:White Crystal PowderPeso molecular:307.14L-Serine
CAS:<p>L-Serine, a non-essential amino acid, vital in proteins and active in serine proteases like trypsin.</p>Fórmula:C3H7NO3Pureza:99.20% - 99.78%Cor e Forma:Hexagonal Plates Or Prisms SolidPeso molecular:105.09FICZ
CAS:<p>FICZ (6-Formylindolo[3,2-b]carbazole) is a potent aryl agonist for the hydrocarbon receptor (AhR, Kd: 70 pM).</p>Fórmula:C19H12N2OPureza:98.97%Cor e Forma:SolidPeso molecular:284.31Leteprinim potassium
CAS:<p>Leplinine (AIT-082, SPI-205) is a neurotrophic agent that may be used to treat Alzheimer's disease and spinal cord injury.</p>Fórmula:C15H13KN5O4Cor e Forma:SolidPeso molecular:366.398Oxoadipic acid
CAS:<p>Oxoadipic acid: metabolite from tryptophan and lysine, links TCA cycle to lysine synthesis, studied for mitochondrial transport.</p>Fórmula:C6H8O5Pureza:96.61% - >99.99%Cor e Forma:SolidPeso molecular:160.12DPN
CAS:<p>DPN (Diarylpropionitrile) is an selective agonist of estrogen receptor β (ERβ) .</p>Fórmula:C15H13NO2Pureza:99.01%Cor e Forma:Off-White SolidPeso molecular:239.27Rosiptor
CAS:<p>Rosiptor (AQX-1125) (AQX-1125) is an orally-active and specific phosphatase SHIP1 activator with anti-inflammatory effects.</p>Fórmula:C20H35NO2Pureza:99.53% - 99.73%Cor e Forma:SolidPeso molecular:321.5Columbamine
CAS:<p>Columbamine (Columbamin) shows strong activity with IC5 48.1 μM.Columbamine exerts anti-proliferative and anti-vasculogenic effects on metastatic human</p>Fórmula:C20H20NO4Pureza:99.16% - 99.65%Cor e Forma:SolidPeso molecular:338.387-methoxy-8-hydroxy-4-methylcoumarin
CAS:<p>7-methoxy-8-hydroxy-4-methylcoumarin is a compound isolated from Citrus aurantium.</p>Fórmula:C11H10O4Pureza:99.89%Cor e Forma:SolidPeso molecular:206.19Lesinurad
CAS:<p>Lesinurad (RDEA594), a selective uric acid reabsorption inhibitor, is used to treat gout without causing liver damage.</p>Fórmula:C17H14BrN3O2SPureza:99.83% - 99.86%Cor e Forma:SolidPeso molecular:404.28Dimethyl lithospermate B
CAS:<p>Dimethyl lithospermate B (dmLSB) is a selective Na+ channel agonist.</p>Fórmula:C38H34O16Pureza:98.34% - 99.62%Cor e Forma:SolidPeso molecular:746.67Cilofexor tromethamine
CAS:<p>Cilofexor (GS-9674), a nonsteroidal FXR agonist, reduces cholestasis and liver damage in PSC, showing safety and efficacy in trials.</p>Fórmula:C32H33Cl3N4O8Cor e Forma:SolidPeso molecular:707.99Tempol
CAS:<p>Tempol (Tanol) is a superoxide scavenger. It has anti-inflammatory, neuroprotective and analgesic effects.</p>Fórmula:C9H18NO2Pureza:97% - 99.74%Cor e Forma:4-Hydroxy-Tempo Appears As Orange Flakes Solid FlakesPeso molecular:172.25Fibronectin CS1 Peptide acetate
<p>CS1 peptide in IIICS and C-274 lacks RGD, inhibits tumor metastasis.</p>Fórmula:C40H68N8O17Pureza:98.09%Cor e Forma:SolidPeso molecular:933.014-Methyl-2-oxopentanoic acid
CAS:<p>4-Methyl-2-oxopentanoic acid, an abnormal metabolite and neurotoxin, results from improper branched-chain amino acid metabolism.</p>Fórmula:C6H10O3Pureza:99.09%Cor e Forma:LiquidPeso molecular:130.14Potassium thioacetate
CAS:<p>Potassium thioacetate: a sulfur donor for creating polymers, heterocycles, nanoparticles, ligands, bioactives, and complexes.</p>Fórmula:C2H3KOSPureza:98.69%Cor e Forma:White CrystalPeso molecular:114.21CORM-3
CAS:<p>CORM-3 is a carbon monoxide-releasing molecule with anti-inflammatory and cardioprotective activity.</p>Fórmula:C5H4ClNO5RuPureza:98%Cor e Forma:SolidPeso molecular:294.61Lys-SMCC-DM1
CAS:<p>Lys-SMCC-DM1 (Lys-Nε-MCC-DM1) inhibits microtubule polymerization and is commonly used in breast cancer research. Cost-effective and quality-assured.</p>Fórmula:C53H75ClN6O15SPureza:≥98%Cor e Forma:SolidPeso molecular:1103.71Sinapyl alcohol
CAS:<p>Technical grade is a natural from Magnolia sieboldii</p>Fórmula:C11H14O4Pureza:99.66% - 99.67%Cor e Forma:SolidPeso molecular:210.23Apabetalone
CAS:<p>Apabetalone (RVX000222) , an effective BET bromodomain inhibitor, has been investigated for the treatment of diabetes, atherosclerosis, and coronary artery</p>Fórmula:C20H22N2O5Pureza:98.08% - ≥98%Cor e Forma:SolidPeso molecular:370.4E7449
CAS:<p>E7449 is a potent inhibitor of PARP1, PARP2, TNKS1, and TNKS2 with IC50s of 2, 1, ~50, and ~50 nM respectively.</p>Fórmula:C18H15N5OPureza:97.13%Cor e Forma:SolidPeso molecular:317.34Fmoc-1,6-diaminohexane
CAS:<p>Fmoc-1,6-diaminohexane has the potential for Alzheimer's disease and cancer treatment.Fmoc-1,6-diaminohexane is an analog of Osw-1.</p>Fórmula:C21H26N2O2Pureza:98%Cor e Forma:SolidPeso molecular:338.44Kaempferol-3-O-glucorhamnoside
CAS:<p>Kaempferol-3-O-glucorhamnoside (Kaempferol 3-glucorhamnoside), a flavonoid derived from plant Thesium chinense Turcz, inhibits inflammatory responses via MAPK</p>Fórmula:C27H30O15Pureza:96.96% - 98.17%Cor e Forma:SolidPeso molecular:594.54-Hydroxyacetophenone
CAS:<p>4-Hydroxyacetophenone (4-Acetylphenol) is a potent xanthine oxidase inhibitor.</p>Fórmula:C8H8O2Pureza:99.94%Cor e Forma:SolidPeso molecular:136.15Entinostat
CAS:<p>Entinostat (MS-275) is an HDAC class I with oral activity. Entinostat has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C21H20N4O3Pureza:98% - 99.74%Cor e Forma:SolidPeso molecular:376.41Benzyl isothiocyanate
CAS:<p>BITC, found in cruciferous veggies, exhibits anticancer, antimicrobial, and immunomodulatory effects.</p>Fórmula:C8H7NSPureza:99.25% - 99.83%Cor e Forma:Clear Yellow LiquidPeso molecular:149.212,2-Dihydroxy-1-phenylethan-1-one
CAS:<p>2,2-Dihydroxy-1-phenylethan-1-one (Phenylglyoxal hydrate) has antioxidant activity.</p>Fórmula:C8H8O3Pureza:97.10%Cor e Forma:SolidPeso molecular:152.15Fmoc-NH-PEG10-acid
CAS:<p>Fmoc-NH-PEG10-acid is a PEG-based PROTAC linker. Fmoc-NH-PEG10-acid can be used in the synthesis of PROTACs.</p>Fórmula:C38H57NO14Pureza:98.00%Cor e Forma:SolidPeso molecular:751.86BPC 157 acetate(137525-51-0 free base)
<p>BPC 157 acetate(137525-51-0 free base) is a 15-amino acid fragment of a gastric peptide (BPC) which has hepatoprotective effects.</p>Fórmula:C64H102N16O24Pureza:>99.99%Cor e Forma:SolidPeso molecular:1479.61(E)-2-Decenoic acid
CAS:<p>(E)-2-Decenoic acid (trans-2-Decenoic acid) is an unsaturated fatty acid found in royal jelly produced from the mandibular gland secretions of honeybees.</p>Fórmula:C10H18O2Pureza:98%Cor e Forma:SolidPeso molecular:170.25gypenoside A
CAS:<p>anticancer</p>Fórmula:C46H74O17Pureza:99.73% - 99.79%Cor e Forma:SolidPeso molecular:899.07Dinotefuran
CAS:<p>Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.</p>Fórmula:C7H14N4O3Pureza:99.89%Cor e Forma:White Crystalline PowderPeso molecular:202.21L-Leucyl-L-alanine
CAS:<p>L-Leucyl-L-alanine is a simple dipeptide composed of L-leucine and L-alanine>[1].</p>Fórmula:C9H18N2O3Pureza:98% - ≥98%Cor e Forma:SolidPeso molecular:202.253,5,7,3′,4′-Pentamethoxyflavone
CAS:<p>3,5,7,3′,4′-Pentamethoxyflavone (Quercetin 3,5,7,3,4-pentamethyl ether) is a natural product. It can induce adipogenesis on 3T3-L1 preadipocytes.</p>Fórmula:C20H20O7Pureza:98.87%Cor e Forma:SolidPeso molecular:372.37Cytidine 5'-diphosphate disodium
CAS:<p>Cytidine 5'-diphosphate disodium (CDP sodium salt) produces CTP to support DNA and RNA biosynthesis and ribonucleotide reductase to produce dCMP.</p>Fórmula:C9H13N3Na2O11P2Pureza:99.78%Cor e Forma:SolidPeso molecular:447.14Nicardipine
CAS:Nicardipine (Cardene), a calcium channel blockers belonging to the dihydropyridine class, is a drug used to treat angina and high blood pressure.Fórmula:C26H29N3O6Pureza:99.56%Cor e Forma:SolidPeso molecular:479.52Methyl pentadecanoate
CAS:<p>Methyl pentadecanoate is a natural product.Methyl pentadecanoate is a saturated fatty acid methyl ester obtained from the esterification of myristic acid.</p>Fórmula:C16H32O2Pureza:98.61%Cor e Forma:SolidPeso molecular:256.422-Di-1-ASP
CAS:<p>2-Di-1-ASP: mono-stryryl dye, stains mitochondria, binds DNA. Selective for G-quadruplex and double-stranded DNA.</p>Fórmula:C16H19IN2Pureza:99.98%Cor e Forma:SolidPeso molecular:366.24mAChR-IN-1 hydrochloride
CAS:<p>mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.</p>Fórmula:C23H26ClIN2O2Pureza:99.87%Cor e Forma:SolidPeso molecular:524.82Protein kinase inhibitors 1 hydrochlorid
<p>Protein kinase inhibitors 1 hydrochlorid (Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base))) is a novel inhibitor of HIPK2 with an IC50 of 74</p>Fórmula:C18H18ClN5O3SPureza:98.00% - 98.78%Cor e Forma:SolidPeso molecular:419.88NSC-87877 disodium
CAS:<p>NSC-87877 disodium (NSC87877) is a cell-permeable inhibitor of both SHP-1 and SHP-2. NSC-87877 also inhibits EGF-induced Erk1/2 activation in HEK293 cells.</p>Fórmula:C19H13N3O7S2·2NaPureza:97.89%Cor e Forma:SolidPeso molecular:503.42NT157
CAS:<p>NT157, a small tyrphostin, inhibits IRS, IGF-1R, and STAT3 in TME, reducing cancer cell survival.</p>Fórmula:C16H14BrNO5SPureza:99.64%Cor e Forma:SolidPeso molecular:412.263-AP
CAS:<p>3-AP (Triapine) is a novel inhibitor of the M2 subunit of ribonucleotide reductase (RR).</p>Fórmula:C7H9N5SPureza:97.33% - 99.87%Cor e Forma:SolidPeso molecular:195.24Duloxetine
CAS:<p>Duloxetine is an inhibitor of serotonin-norepinephrine reuptake(Ki of 4.6 nM),with treatment of major depressive disorder and generalized anxiety disorder.</p>Fórmula:C18H19NOSPureza:99.71% - 99.89%Cor e Forma:SolidPeso molecular:297.41Lenalidomide hydrochloride
CAS:<p>Lenalidomide HCl, a Thalidomide derivative, modulates immunity, targets CRBN, and selectively impedes B-cell lymphomas.</p>Fórmula:C13H14ClN3O3Cor e Forma:SolidPeso molecular:295.72Vicine
CAS:<p>Vicine, an alkaloid found in fava beans, is toxic in individuals and may cause haemolytic anaemia.</p>Fórmula:C10H16N4O7Pureza:99.82% - >99.99%Cor e Forma:SolidPeso molecular:304.26
