
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.523 produtos)
- Apoptose(5.792 produtos)
- Ciclo celular/Ponto de verificação(4.449 produtos)
- Cromatina/Epigenética(2.238 produtos)
- Sinalização Citoesquelética(1.383 produtos)
- Dano de DNA/Reparo de DNA(2.825 produtos)
- Endocrinologia/Hormónios(3.507 produtos)
- Enzima(3.640 produtos)
- GPCR/Proteína-G(8.333 produtos)
- Imunologia e Inflamação(3.526 produtos)
- Vírus da Influenza(296 produtos)
- Sinalização JAK/STAT(404 produtos)
- Sinalização MAPK(1.202 produtos)
- Transportador de Membranas/Canal Iónico(2.790 produtos)
- Metabolismo(9.448 produtos)
- Microbiologia/Virologia(6.981 produtos)
- Neurociência(9.926 produtos)
- Outros inibidores(37.926 produtos)
- Oxidação-Redução(41 produtos)
- Sinalização PI3K/Akt/mTOR(1.400 produtos)
- Proteases/Proteassoma(1.597 produtos)
- Células - tronco e Derivados(831 produtos)
- Tirosina Quinase/Adaptador(2.016 produtos)
- Ubiquitinação(1.650 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66641 produtos de "Inibidores"
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Propargyl-PEG5-Ms
CAS:<p>Propargyl-PEG5-Ms (Propargyl-PEG6-Ms) is a PEG-based PROTAC linker. Propargyl-PEG5-Ms can be used in the synthesis of PROTACs.</p>Fórmula:C14H26O8SPureza:≥98%Cor e Forma:SolidPeso molecular:354.42Mal-PEG5-Boc
CAS:<p>Mal-PEG5-Boc (Mal-PEG5-COOtBu) is a PEG-based PROTAC linker. Mal-PEG5-Boc can be used in the synthesis of PROTACs.</p>Fórmula:C21H35NO9Pureza:99.72%Cor e Forma:SolidPeso molecular:445.5Capadenoson
CAS:<p>Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.</p>Fórmula:C25H18ClN5O2S2Pureza:98.85% - 99.57%Cor e Forma:SolidPeso molecular:520.03Magainin 1 acetate
<p>Magainin 1 acetate is an antimicrobial peptide. Magainin 1 acetate exhibits antibiotic activity against numerous Gram-negative and Gram-positive bacteria.</p>Fórmula:C114H181N29O30SPureza:96.65%Cor e Forma:SolidPeso molecular:2469.9Boc-NH-C6-Br
CAS:<p>Boc-NH-C6-Br is a cleavable linker used for antibody-drug conjugates (ADC).</p>Fórmula:C11H22BrNO2Pureza:95.09%Cor e Forma:SolidPeso molecular:280.2S-23
CAS:<p>S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (</p>Fórmula:C18H13ClF4N2O3Pureza:99.55%Cor e Forma:SolidPeso molecular:416.75γ-Linolenic Acid methyl ester
CAS:<p>γ-Linolenic Acid methyl ester (Methyl gamma-linolenate) is a weak leukotriene B4 (LTB4) receptor antagonist.</p>Fórmula:C19H32O2Pureza:98%Cor e Forma:SolidPeso molecular:292.46Lvguidingan
CAS:<p>Lvguidingan is an Anticonvulsant agent.</p>Fórmula:C13H15Cl2NOPureza:99.53% - 99.87%Cor e Forma:SolidPeso molecular:272.17Syringaresinol diglucoside
CAS:<p>Syringaresinol diglucoside (Syringaresinol-di-O-glucoside) protects the animals from the stress-induced decreases in sex behaviours and in rectal temperature.</p>Fórmula:C34H46O18Pureza:98.59% - 99.77%Cor e Forma:SolidPeso molecular:742.72GSK2334470
CAS:<p>GSK2334470 is a novel PDK1 inhibitor (IC50: ~10 nM, in a cell-free assay), with no inhibitory at other close related AGC-kinases.</p>Fórmula:C25H34N8OPureza:99.57% - 99.87%Cor e Forma:SolidPeso molecular:462.595(6)-CFDA
CAS:<p>5(6)-CFDA: cell-permeable, esterase-responsive viability probe; fluoresces upon activation, indicating enzymatic activity and membrane integrity.</p>Fórmula:C50H32O18Pureza:95.25%Cor e Forma:SolidPeso molecular:920.78PRE-084 hydrochloride
CAS:<p>PRE-084 hydrochloride is a selective agonist of σ1(IC50:44 nM, in the sigma receptor assay).</p>Fórmula:C19H28ClNO3Pureza:99.54%Cor e Forma:SolidPeso molecular:353.88Thalidomide-NH-CH2-COOH
CAS:<p>Thalidomide-NH-CH2-COOH ((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)glycine) is a synthesized E3 ligase ligand-linker conjugate containing a</p>Fórmula:C15H13N3O6Pureza:96.3800%Cor e Forma:SolidPeso molecular:331.28Eribulin mesylate
CAS:<p>Eribulin mesylate (E7389), a microtubule inhibitor, treats metastatic breast cancer by halting cell division.</p>Fórmula:C41H63NO14SPureza:97.02% - >99.99%Cor e Forma:SolidPeso molecular:826TPT-260 Dihydrochloride
CAS:<p>TPT-260 Dihydrochloride (NSC55712) is a thiophene thiourea derivative with molecule weight 260.00 in free base form.</p>Fórmula:C8H14Cl2N4S3Pureza:92.87% - 97.32%Cor e Forma:SolidPeso molecular:333.32Orsellinic acid
CAS:<p>Orsellinic acid is a phenolic acid extracted from lichens.</p>Fórmula:C8H8O4Pureza:97.01% - 98.4%Cor e Forma:SolidPeso molecular:168.15D-Lyxose
CAS:<p>D-Lyxose (D-(-)-Lyxose) is used as a chiral building block.</p>Fórmula:C5H10O5Pureza:98.84% - 99.35%Cor e Forma:White Crystalline PowderPeso molecular:150.13Heparan Sulfate
CAS:<p>Heparan sulfate is a natural product, a linear polysaccharide. Heparan sulfate occurs as a proteoglycan (HSPG). Cost effective and quality assured.</p>Fórmula:C12H19NO20S3(monomer)Pureza:98%Cor e Forma:SolidPeso molecular:593.47(monomer)5'-N-Ethylcarboxamidoadenosine
CAS:<p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>Fórmula:C12H16N6O4Pureza:98.95% - ≥95%Cor e Forma:PowderPeso molecular:308.29Sucrose
CAS:<p>Sucrose (D-(+)-Saccharose) is a nonreducing disaccharide composed of glucose and fructose linked via their anomeric carbons.</p>Fórmula:C12H22O11Pureza:99.87% - 99.88%Cor e Forma:White Crystals Or PowderPeso molecular:342.30CEF27, Epstein-Barr Virus BRLF-1 lytic 148-156 acetate
<p>CEF27 is an EBV BRLF-1 lytic 148-156 acetate, a transcriptional activator targeting GC-rich motifs in EBV gene promoters.</p>Fórmula:C53H86N16O16Pureza:99.94%Cor e Forma:SolidPeso molecular:1203.35Bentamapimod
CAS:<p>Bentamapimod (AS 602801) is a novel, orally active inhibitor of JNK.</p>Fórmula:C25H23N5O2SPureza:97.04% - 99.92%Cor e Forma:SolidPeso molecular:457.558-Epideoxyloganic acid
CAS:<p>8-Epideoxyloganic acid offers pain relief, stabilizes bodily functions, reduces inflammation, and may inhibit ROS via NOX activity.</p>Fórmula:C16H24O9Pureza:99.41% - 99.96%Cor e Forma:SolidPeso molecular:360.36GSK2018682
CAS:<p>GSK2018682 is an agonist of sphingosine-1-phosphate receptor (s1p1) and (s1p5) agonist(pEC50s of 7.7 and 7.2,respectively).</p>Fórmula:C22H21ClN4O4Pureza:99.04%Cor e Forma:SolidPeso molecular:440.88GSK-2256098 HCl
CAS:<p>GSK-2256098 HCl is a focal adhesion kinase-1 (FAK) inhibitor with potential antiangiogenic and antineoplastic activities.</p>Fórmula:C20H24Cl2N6O2Cor e Forma:SolidPeso molecular:451.35[Gln8]-C517 (LH-RH), chicken acetate
<p>Avian peptide [Gln8]-C517 (LH-RH) triggers gonadotropin release, regulating reproduction.</p>Fórmula:C56H75N15O16Pureza:99.83%Cor e Forma:SolidPeso molecular:1214.31Preladenant
CAS:<p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine</p>Fórmula:C25H29N9O3Pureza:98.02% - 99.68%Cor e Forma:SolidPeso molecular:503.56Inauhzin
CAS:<p>Inauhzin (INZ) reactivates p53, inhibits SIRT1, induces Y cell apoptosis without genotoxic stress (IC50=3 uM in A549).</p>Fórmula:C25H19N5OS2Pureza:98% - 99.36%Cor e Forma:SolidPeso molecular:469.58NDI-091143
CAS:<p>NDI-091143 is a potent and high-affinity human ATP-citrate lyase (ACLY) inhibitor with an IC50 of 2.1 nM (ADP-Glo assay),indirectly disrupting citrate binding</p>Fórmula:C20H14ClF2NO5SPureza:97.03% - ≥95%Cor e Forma:SolidPeso molecular:453.84Methyl picolinate
CAS:<p>Methyl picolinate (Methyl picolinate) is used as pharmaceutical intermediate.</p>Fórmula:C7H7NO2Pureza:99.42%Cor e Forma:SolidPeso molecular:137.14PFI-3
CAS:<p>PFI-3 is a selective chemical inhibitor for SMARCA (2/4) (Kd = 89 nM)and PBI (5) bromodomains which may result in the delay and prevention of breast cancer.</p>Fórmula:C19H19N3O2Pureza:99.58% - 99.94%Cor e Forma:SolidPeso molecular:321.37Novokinin acetate
<p>Novokinin acetate binds AT2 receptor (Ki=7 nM); antihypertensive effect blocked by PD123319.</p>Fórmula:C41H65N11O9Pureza:99.37%Cor e Forma:SoildPeso molecular:856.02Saccharin 1-methylimidazole
CAS:<p>Saccharin 1-methylimidazole (SMI) is a general-purpose activator used for DNA and RNA synthesis.</p>Fórmula:C7H5NO3S·C4H6N2Pureza:98.21%Cor e Forma:SolidPeso molecular:265.29Angeloylgomisin Q
CAS:<p>Angeloylgomisin Q is a natural product from Schizandra chinensis BAILL.</p>Fórmula:C29H38O9Pureza:99.83%Cor e Forma:SolidPeso molecular:530.61MRTX9768
CAS:<p>MRTX-9768 is a synthetic lethal-based inhibitor designed to bind the PRMT5-MTA complex and selectively target MTAP/CDKN2A-deleted tumors.</p>Fórmula:C24H17FN6OPureza:97.02%Cor e Forma:SolidPeso molecular:424.43Lactobionic acid
CAS:<p>Lactobionic acid with antioxidant, antimicrobial and moisturizing propertie</p>Fórmula:C12H22O12Pureza:99.6%Cor e Forma:White PowderPeso molecular:358.3UNC2541
CAS:<p>UNC2541 is a potent and Mer tyrosine kinase (MerTK)-specific inhibitor.</p>Fórmula:C24H34FN7O2Pureza:98.33%Cor e Forma:SolidPeso molecular:471.57TED-347
CAS:<p>TED-347 is an irreversible and covalent inhibitor of TEAD4-Yap1 protein-protein interaction(EC50 of 5.9 μM), and inhibits glioblastoma cell viability.</p>Fórmula:C15H11ClF3NOPureza:99.9%Cor e Forma:SolidPeso molecular:313.72-Iodobenzenamine
CAS:<p>2-Iodobenzenamine (NSC-34544) is an agent of biochemical.</p>Fórmula:C6H6INPureza:99.95%Cor e Forma:Brown - Yellow NeedlesPeso molecular:219.02Neobavaisoflavone
CAS:<p>Neobavaisoflavone: DNA polymerase inhibitor, potential for treating bone loss, anti-inflammatory, reduces ROS, RNS, cytokines in macrophages.</p>Fórmula:C20H18O4Pureza:99.31% - 99.87%Cor e Forma:SolidPeso molecular:322.35Xanthotoxol
CAS:<p>Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.</p>Fórmula:C11H6O4Pureza:99.97%Cor e Forma:SolidPeso molecular:202.16DD1
CAS:<p>DD1 (HUN85111) is a proteasome inhibitor that induces human myeloid tumor-selective apoptosis.</p>Fórmula:C16H14N2O3Pureza:99.57%Cor e Forma:SolidPeso molecular:282.29D-α-Methylbenzyl isothiocyanate
CAS:<p>D-alpha-Methylbenzyl isothiocyanate, an antioxidant and a chiral agent, induces phase II enzyme activity.</p>Fórmula:C9H9NSPureza:99.80%Cor e Forma:SolidPeso molecular:163.24FPH2
CAS:<p>FPH2 (BRD-9424) (BRD-9424) is a small molecule promoting differentiation of iPS-derived hepatocytes.</p>Fórmula:C14H16ClN5O2SPureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:353.83Zingibroside R1
CAS:<p>Zingibroside R1 (Ginsenoside Z-R1) has anti-HIV-1 activity.</p>Fórmula:C42H66O14Pureza:99.13% - 99.96%Cor e Forma:SolidPeso molecular:794.97CTPI-2
CAS:<p>CTPI-2 inhibits SLC25A1 (KD: 3.5 μM), glycolysis, PPARγ, GLUT4, has anti-tumor effects, and combats NASH and diet-induced obesity.</p>Fórmula:C13H9ClN2O6SPureza:97.23%Cor e Forma:SolidPeso molecular:356.74Davercin
CAS:<p>Davercin (Erythromycin Cyclocarbonate), a Erythromycin derivative, exhibits efficacy against both Gram-positive and select Gram-negative microorganisms.</p>Fórmula:C38H65NO14Pureza:97.55% - 98.732%Cor e Forma:SolidPeso molecular:759.925-Methylfurfural
CAS:<p>5-Methylfurfural (5-Methyl-2-furaldehyde) has been identified as one of the volatile flavor compounds in tamarind, Dutch Coffee and barrel-aged wines.</p>Fórmula:C6H6O2Pureza:98.48%Cor e Forma:Less To Light Yellow Liquid Colorless To Light Yellow LiquidPeso molecular:110.11BMS-5
CAS:<p>BMS-5 (LIMKi 3) is a potent LIMK inhibitor with IC50s of 7 nM and 8 nM for LIMK1 and LIMK2, respectively.</p>Fórmula:C17H14Cl2F2N4OSPureza:98.01% - 99.88%Cor e Forma:SolidPeso molecular:431.29Acetyl-PHF6 amide acetate
<p>Acetyl-PHF6 amide acetate(878663-43-5 freebase) (AcPHF6 acetate) is a tau derived hexapeptide.</p>Fórmula:C40H67N9O11Pureza:>99.99%Cor e Forma:SolidPeso molecular:850.01
