CAS 152477-89-9

PRAZEPAM-D5

Description:

Prazepam-D5 is a deuterated derivative of prazepam, which is a benzodiazepine used primarily for its anxiolytic properties. The incorporation of deuterium atoms in its molecular structure alters its pharmacokinetic profile, potentially affecting its metabolism and duration of action compared to non-deuterated prazepam. As a benzodiazepine, prazepam-D5 functions by enhancing the effect of the neurotransmitter gamma-aminobutyric acid (GABA) at the GABA-A receptor, leading to increased inhibitory neurotransmission in the central nervous system. This results in anxiolytic, sedative, muscle relaxant, and anticonvulsant effects. The deuterated form is often utilized in research to study drug metabolism and pharmacodynamics, as the presence of deuterium can provide insights into metabolic pathways and the drug's behavior in biological systems. While specific therapeutic applications may vary, the general characteristics of prazepam-D5 align with those of other benzodiazepines, including potential side effects such as drowsiness, dizziness, and dependence with prolonged use.

Formula:C₁₉H₁₂ClD₅N₂O

InChI:InChI=1S/C19H17ClN2O/c20-15-8-9-17-16(10-15)19(14-4-2-1-3-5-14)21-11-18(23)22(17)12-13-6-7-13/h1-5,8-10,13H,6-7,11-12H2/i1D,2D,3D,4D,5D

InChI key:MWQCHHACWWAQLJ-RALIUCGRSA-N

SMILES:[2H]C1=C(C(=C(C(=C1[2H])[2H])C2=NCC(=O)N(C3=C2C=C(C=C3)Cl)CC4CC4)[2H])[2H]

Synonyms:

2H-1,4-Benzodiazepin-2-one, 7-chloro-1-(cyclopropylmethyl)-1,3-dihydro-5-(phenyl-d5)-
Prazepam-D5,100/Mlinmethanol
PRAZEPAM (D5, 98%) 100 UG/ML IN METHANOL
7-chloro-1-(cyclopropylmethyl)-5-(2,3,4,5,6-pentadeuteriophenyl)-3H-1,4-benzodiazepin-2-one
PRAZEPAM-D5
Prazepam-d5 solution
Prazepam-d5 (100 μg/mL in Methanol)

Found 7 products.

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Prazepam-d5 (phenyl-d5)
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 152477-89-9
- 2955-38-6
Purity:99 atom % D
Color and Shape:White To Yellow Wolid
Molecular weight:329.84
Ref: 3U-D7148
10mg
1,278.00€
VAT not included
+ Info
Prazepam-D5, 0.1mg/ml in Methanol
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 152477-89-9
Formula:C₁₉₂H₅H₁₂ClN₂O
Color and Shape:Colourless
Molecular weight:329.83
Ref: 61-AMP1258.80-02
1ml
60.00€
VAT not included
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Prazepam-D5, 0.1mg/ml in Methanol
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 152477-89-9
Formula:C₁₉₂H₅H₁₂ClN₂O
Color and Shape:Colourless
Molecular weight:329.83
Ref: LP-PRA-1691-0.1LM
1ml
60.00€
VAT not included
+ Info
Prazepam-D5
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 152477-89-9
Formula:C₁₉₂H₅H₁₂ClN₂O
Color and Shape:Neat
Molecular weight:329.83
Ref: LP-PRA-1691
10mg
1,022.00€
VAT not included
50mg
3,066.00€
VAT not included
100mg
5,519.00€
VAT not included
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Prazepam-d5
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 152477-89-9
Applications Prazepam-d5, is the labeled analogue of Prazepam (P702250), a benzodiazepine derivative drug having anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant properties.
References Shader R. I., et al.: Ciba. Found. Symp., (74), 141 (1979); Jacqmin, P., et al.: Neuropsychobiology, 19 (4), 186 (1988);
Formula:C₁₉₂H₅H₁₂ClN₂O
Color and Shape:Neat
Molecular weight:329.83
Ref: TR-P702252
1mg
163.00€
VAT not included
10mg
438.00€
VAT not included
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Prazepam-d5 (100 µg/mL in Methanol)
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 152477-89-9
Formula:C₁₉₂H₅H₁₂ClN₂O
Color and Shape:Single Solution
Molecular weight:329.83
Ref: TR-KIT1767
5x1ml
432.00€
VAT not included
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Prazepam-d5 (1 mg/ml in Acetonitrile)
Controlled ProductPlease note that this is a controlled product in some countries, and needs to be treated in accordance with the relevant regulations. Be aware this might entail additional expenses and documentation.
CAS:
- 152477-89-9
Formula:C₁₉₂H₅H₁₂ClN₂O
Color and Shape:Single Solution
Molecular weight:329.83
Ref: TR-KIT7030
1x1ml
933.00€
VAT not included