CAS 207572-68-7

RILMENIDINE HEMIFUMARATE SALT

Description:

Rilmenidine hemifumarate salt is a pharmaceutical compound primarily used as an antihypertensive agent. It acts as an agonist at imidazoline receptors, which plays a crucial role in regulating blood pressure by reducing sympathetic nervous system activity. The substance is typically presented as a hemifumarate salt, enhancing its solubility and stability for therapeutic use. Rilmenidine is known for its selective action, which minimizes side effects commonly associated with other antihypertensive medications. In terms of physical characteristics, it is usually a white to off-white crystalline powder. The compound is soluble in water and exhibits a moderate pH range, making it suitable for oral administration. Its pharmacokinetics involve rapid absorption and a relatively short half-life, necessitating careful dosing to maintain effective blood pressure control. As with any medication, potential side effects may include dizziness, dry mouth, or fatigue, and it is essential to monitor patients for any adverse reactions during treatment.

Formula: C₁₀H₁₆N₂O·C₄H₄O₄

Synonyms:

• RILMENIDINE HEMIFUMARATE SALT
• n-(dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine hemifumarate salt
• LZFATBMLSYHRTC-WXXKFALUSA-N
• Oxaminozoline hemifumarate salt, Rilmenidene hemifumarate salt, N-(Dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine hemifumarate salt

N-(Dicyclopropylmethyl)-4,5-dihydrooxazol-2-amine hemifumarate

CAS: 207572-68-7

N-(Dicyclopropylmethyl)-4,5-dihydrooxazol-2-amine hemifumarate

Formula: C₂₄H₃₆N₄O₆

Purity: 98%

Molecular weight: 476.57

Ref: 54-OR1063662

Rilmenidine hemifumarate

CAS: 207572-68-7

Formula: C₂₄H₃₆N₄O₆

Purity: 98%

Color and Shape: Solid

Molecular weight: 476.5658

Ref: IN-DA002J59

Rilmenidine hemifumarate salt

CAS: 207572-68-7

Formula: C₁₀H₁₆N₂O·5C₄H₄O₄

Purity: ≥ 98.5%

Color and Shape: White solid

Molecular weight: 238.28

Ref: 7W-GP9411

Rilmenidine hemifumarate

CAS: 207572-68-7

Rilmenidine hemifumarate (S-3341 hemifumarate) is an I1 imidazoline receptor and α2-adrenergic receptor agonist that induces autophagy.

Formula: C₁₀H₁₆N₂OC₄H₄O₄

Purity: 98.14%

Color and Shape: Solid

Molecular weight: 238.28

Ref: TM-T21911

Rilmenidine Hemifumarate

CAS: 207572-68-7

Applications Rilmenidine hemifumarate  is an antihypertensive agent that selectively binds nonadrenergic imidazoline-binding site I1 receptor.
References Reis, D.J., and Piletz, J.E. Am J Physiol 273, R1569 (1997); Piletz, J. E., et al.: Neuropsychopharmacology 23, 697 (2000)

Formula: C₁₀H₁₆N₂O·C₄H₄O₄

Color and Shape: Neat

Molecular weight: 476.566

Ref: TR-R509705

Rilmenidine hemifumarate

CAS: 207572-68-7

Agonist of ?2-adrenoceptor

Formula: C₁₀H₁₆N₂O•(C₄H₄O₄)₀

Purity: Min. 95%

Molecular weight: 238.28 g/mol

Ref: 3D-BR162477